Degradation of Janus kinases in CRLF2-rearranged acute lymphoblastic leukemia
Chang, Yunchao, Min, Jaeki, Jarusiewicz, Jamie A., Actis, Marisa, Yu-Chen Bradford, Shanshan, Mayasundari, Anand, Yang, Lei, Chepyala, Divyabharathi, Alcock, Lisa J., Roberts, Kathryn G., Nithianantham, Stanley, Maxwell, Dylan, Rowland, Lauren, Larsen, Randolph, Seth, Aman, Goto, Hiroaki, Imamura, Toshihiko, Akahane, Koshi, Hansen, Baranda S., Pruett-Miller, Shondra M., Paietta, Elisabeth M., Litzow, Mark R., Qu, Chunxu, Yang, Jun J., Fischer, Marcus, Rankovic, Zoran, Mullighan, Charles G.
Published in Blood (09.12.2021)
Published in Blood (09.12.2021)
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Journal Article
Discovery of a Diaminopyrimidine FLT3 Inhibitor Active against Acute Myeloid Leukemia
Jarusiewicz, Jamie A, Jeon, Jae Yoon, Connelly, Michele C, Chen, Yizhe, Yang, Lei, Baker, Sharyn D, Guy, R. Kiplin
Published in ACS omega (31.05.2017)
Published in ACS omega (31.05.2017)
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Identification of Potent, Selective, and Orally Bioavailable Small-Molecule GSPT1/2 Degraders from a Focused Library of Cereblon Modulators
Nishiguchi, Gisele, Keramatnia, Fatemeh, Min, Jaeki, Chang, Yunchao, Jonchere, Barbara, Das, Sourav, Actis, Marisa, Price, Jeanine, Chepyala, Divyabharathi, Young, Brandon, McGowan, Kevin, Slavish, P. Jake, Mayasundari, Anand, Jarusiewicz, Jamie A, Yang, Lei, Li, Yong, Fu, Xiang, Garrett, Shalandus H, Papizan, James B, Kodali, Kiran, Peng, Junmin, Pruett Miller, Shondra M, Roussel, Martine F, Mullighan, Charles, Fischer, Marcus, Rankovic, Zoran
Published in Journal of medicinal chemistry (10.06.2021)
Published in Journal of medicinal chemistry (10.06.2021)
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Journal Article
Development of an Orally Bioavailable LCK PROTAC Degrader as a Potential Therapeutic Approach to T‑Cell Acute Lymphoblastic Leukemia
Jarusiewicz, Jamie A., Yoshimura, Satoshi, Actis, Marisa, Li, Yong, Fu, Xiang, Yang, Lei, Narina, Shilpa, Pruett-Miller, Shondra M., Zhou, Suiping, Wang, Xusheng, High, Anthony A., Nishiguchi, Gisele, Yang, Jun J., Rankovic, Zoran
Published in Journal of medicinal chemistry (25.07.2024)
Published in Journal of medicinal chemistry (25.07.2024)
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Journal Article
Phenyl Dihydrouracil: An Alternative Cereblon Binder for PROTAC Design
Jarusiewicz, Jamie A., Yoshimura, Satoshi, Mayasundari, Anand, Actis, Marisa, Aggarwal, Anup, McGowan, Kevin, Yang, Lei, Li, Yong, Fu, Xiang, Mishra, Vibhor, Heath, Richard, Narina, Shilpa, Pruett-Miller, Shondra M., Nishiguchi, Gisele, Yang, Jun J., Rankovic, Zoran
Published in ACS medicinal chemistry letters (09.02.2023)
Published in ACS medicinal chemistry letters (09.02.2023)
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Journal Article
Development of Potent and Selective Janus Kinase 2/3 Directing PG–PROTACs
Alcock, Lisa J, Chang, Yunchao, Jarusiewicz, Jamie A, Actis, Marisa, Nithianantham, Stanley, Mayasundari, Anand, Min, Jaeki, Maxwell, Dylan, Hunt, Jeremy, Smart, Brandon, Yang, Jun J, Nishiguchi, Gisele, Fischer, Marcus, Mullighan, Charles G, Rankovic, Zoran
Published in ACS medicinal chemistry letters (10.03.2022)
Published in ACS medicinal chemistry letters (10.03.2022)
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Chemical scaffold recycling: Structure-guided conversion of an HIV integrase inhibitor into a potent influenza virus RNA-dependent RNA polymerase inhibitor designed to minimize resistance potential
Slavish, Peter J., Cuypers, Maxime G., Rimmer, Mary Ashley, Abdolvahabi, Alireza, Jeevan, Trushar, Kumar, Gyanendra, Jarusiewicz, Jamie A., Vaithiyalingam, Sivaraja, Jones, Jeremy C., Bowling, John J., Price, Jeanine E., DuBois, Rebecca M., Min, Jaeki, Webby, Richard J., Rankovic, Zoran, White, Stephen W.
Published in European journal of medicinal chemistry (05.02.2023)
Published in European journal of medicinal chemistry (05.02.2023)
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Identification of Small Molecules Exhibiting Oxacillin Synergy through a Novel Assay for Inhibition of vraTSR Expression in Methicillin-Resistant Staphylococcus aureus
Lee, Hyun, Boyle-Vavra, Susan, Ren, Jinhong, Jarusiewicz, Jamie A, Sharma, Lalit Kumar, Hoagland, Daniel T, Yin, Shaohui, Zhu, Tian, Hevener, Kirk E, Ojeda, Isabel, Lee, Richard E, Daum, Robert S, Johnson, Michael E
Published in Antimicrobial agents and chemotherapy (01.09.2019)
Published in Antimicrobial agents and chemotherapy (01.09.2019)
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Journal Article
Inhibition of the function of class IIa HDACs by blocking their interaction with MEF2
Jayathilaka, Nimanthi, Han, Aidong, Gaffney, Kevin J, Dey, Raja, Jarusiewicz, Jamie A, Noridomi, Kaori, Philips, Michael A, Lei, Xiao, He, Ju, Ye, Jun, Gao, Tao, Petasis, Nicos A, Chen, Lin
Published in Nucleic acids research (01.07.2012)
Published in Nucleic acids research (01.07.2012)
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Journal Article
Thin layer chromatographic analysis of glucose and maltose in estivated Biomphalaria glabrata snails and those infected with Schistosoma mansoni
Jarusiewicz, Jamie A., Sherma, Joseph, Fried, Bernard
Published in Comparative Biochemistry and Physiology Part B: Biochemistry and Molecular Biology (01.11.2006)
Published in Comparative Biochemistry and Physiology Part B: Biochemistry and Molecular Biology (01.11.2006)
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Journal Article
Effects of diet on the carotenoid pigment and lipid content of Pomacea bridgesii as determined by quantitative high performance thin layer chromatography
Jarusiewicz, Jamie A., Fried, Bernard, Sherma, Joseph
Published in Comparative Biochemistry and Physiology Part B: Biochemistry and Molecular Biology (01.02.2006)
Published in Comparative Biochemistry and Physiology Part B: Biochemistry and Molecular Biology (01.02.2006)
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Journal Article
Chemical scaffold recycling: Structure-guided conversion of an HIV integrase inhibitor into a potent influenza virus RNA-dependent RNA polymerase inhibitor designed to minimize resistance potential
Slavish, Peter J., Cuypers, Maxime G., Rimmer, Mary Ashley, Abdolvahabi, Alireza, Jeevan, Trushar, Kumar, Gyanendra, Jarusiewicz, Jamie A., Vaithiyalingam, Sivaraja, Jones, Jeremy C., Bowling, John J., Price, Jeanine E., DuBois, Rebecca M., Min, Jaeki, Webby, Richard J., Rankovic, Zoran, White, Stephen W.
Published in European journal of medicinal chemistry (01.02.2023)
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Published in European journal of medicinal chemistry (01.02.2023)
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