Nanocarrier mediated retinal drug delivery: overcoming ocular barriers to treat posterior eye diseases
Bisht, Rohit, Mandal, Abhirup, Jaiswal, Jagdish K, Rupenthal, Ilva D
Published in Wiley interdisciplinary reviews. Nanomedicine and nanobiotechnology (01.03.2018)
Published in Wiley interdisciplinary reviews. Nanomedicine and nanobiotechnology (01.03.2018)
Get more information
Journal Article
An agent-based model for drug-radiation interactions in the tumour microenvironment: Hypoxia-activated prodrug SN30000 in multicellular tumour spheroids
Mao, Xinjian, McManaway, Sarah, Jaiswal, Jagdish K, Patel, Priyanka B, Wilson, William R, Hicks, Kevin O, Bogle, Gib
Published in PLoS computational biology (01.10.2018)
Published in PLoS computational biology (01.10.2018)
Get full text
Journal Article
The CSF1 receptor inhibitor pexidartinib (PLX3397) reduces tissue macrophage levels without affecting glucose homeostasis in mice
Merry, Troy L, Brooks, Anna E S, Masson, Stewart W, Adams, Shannon E, Jaiswal, Jagdish K, Jamieson, Stephen M F, Shepherd, Peter R
Published in International Journal of Obesity (01.01.2020)
Published in International Journal of Obesity (01.01.2020)
Get full text
Journal Article
In situ gelling system for sustained intraarticular delivery of bupivacaine and ketorolac in sheep
Abdeltawab, Hani, Bolam, Scott M., Jaiswal, Jagdish K., McGlashan, Sue R., Young, Simon W, Hill, Andrew, Svirskis, Darren, Sharma, Manisha
Published in European journal of pharmaceutics and biopharmaceutics (01.05.2022)
Published in European journal of pharmaceutics and biopharmaceutics (01.05.2022)
Get full text
Journal Article
Cellular pharmacology of evofosfamide (TH-302): A critical re-evaluation of its bystander effects
Hong, Cho Rong, Dickson, Benjamin D., Jaiswal, Jagdish K., Pruijn, Frederik B., Hunter, Francis W., Hay, Michael P., Hicks, Kevin O., Wilson, William R.
Published in Biochemical pharmacology (01.10.2018)
Published in Biochemical pharmacology (01.10.2018)
Get full text
Journal Article
Spatially-resolved pharmacokinetic/pharmacodynamic modelling of bystander effects of a nitrochloromethylbenzindoline hypoxia-activated prodrug
Hong, Cho Rong, Mehta, Sunali Y., Liyanage, H. D. Sarath, McManaway, Sarah P., Lee, Ho H., Jaiswal, Jagdish K., Bogle, Gib, Tercel, Moana, Pruijn, Frederik B., Wilson, William R., Hicks, Kevin O.
Published in Cancer chemotherapy and pharmacology (01.10.2021)
Published in Cancer chemotherapy and pharmacology (01.10.2021)
Get full text
Journal Article
Inhibition of the Cytolytic Protein Perforin Prevents Rejection of Transplanted Bone Marrow Stem Cells in Vivo
Spicer, Julie A, Miller, Christian K, O’Connor, Patrick D, Jose, Jiney, Giddens, Anna C, Jaiswal, Jagdish K, Jamieson, Stephen M. F, Bull, Matthew R, Denny, William A, Akhlaghi, Hedieh, Trapani, Joseph A, Hill, Geoff R, Chang, Karshing, Gartlan, Kate H
Published in Journal of medicinal chemistry (12.03.2020)
Published in Journal of medicinal chemistry (12.03.2020)
Get full text
Journal Article
Pharmacokinetic/Pharmacodynamic Modeling Identifies SN30000 and SN29751 as Tirapazamine Analogues with Improved Tissue Penetration and Hypoxic Cell Killing in Tumors
HICKS, Kevin O, SIIM, Bronwyn G, DENNY, William A, HAY, Michael P, WILSON, William R, JAISWAL, Jagdish K, PRUIJN, Frederik B, FRASER, Annie M, PATEL, Rita, HOGG, Alison, SARATH LIYANAGE, H. D, JO DORIE, Mary, BROWN, J. Martin
Published in Clinical cancer research (15.10.2010)
Published in Clinical cancer research (15.10.2010)
Get full text
Journal Article
Substituted arylsulphonamides as inhibitors of perforin-mediated lysis
Spicer, Julie A., Miller, Christian K., O'Connor, Patrick D., Jose, Jiney, Huttunen, Kristiina M., Jaiswal, Jagdish K., Denny, William A., Akhlaghi, Hedieh, Browne, Kylie A., Trapani, Joseph A.
Published in European journal of medicinal chemistry (08.09.2017)
Published in European journal of medicinal chemistry (08.09.2017)
Get full text
Journal Article
Benzenesulphonamide inhibitors of the cytolytic protein perforin
Spicer, Julie A., Miller, Christian K., O'Connor, Patrick D., Jose, Jiney, Huttunen, Kristiina M., Jaiswal, Jagdish K., Denny, William A., Akhlaghi, Hedieh, Browne, Kylie A., Trapani, Joseph A.
Published in Bioorganic & medicinal chemistry letters (15.02.2017)
Published in Bioorganic & medicinal chemistry letters (15.02.2017)
Get full text
Journal Article
Development of a novel stability indicating RP-HPLC method for quantification of Connexin43 mimetic peptide and determination of its degradation kinetics in biological fluids
Bisht, Rohit, Rupenthal, Ilva D., Sreebhavan, Sreevalsan, Jaiswal, Jagdish K.
Published in Journal of pharmaceutical analysis (01.12.2017)
Published in Journal of pharmaceutical analysis (01.12.2017)
Get full text
Journal Article
Effect of fixed space maintainers and removable appliances on oral microflora in children: An in vivo study
Kundu, Ritesh, Tripathi, Abhay, Jaiswal, Jagdish, Ghoshal, Ujjala, Palit, Madhuchanda, Khanduja, Sonali
Published in Journal of the Indian Society of Pedodontics and Preventive Dentistry (01.01.2016)
Published in Journal of the Indian Society of Pedodontics and Preventive Dentistry (01.01.2016)
Get full text
Journal Article
Diarylthiophenes as inhibitors of the pore-forming protein perforin
Miller, Christian K., Huttunen, Kristiina M., Denny, William A., Jaiswal, Jagdish K., Ciccone, Annette, Browne, Kylie A., Trapani, Joseph A., Spicer, Julie A.
Published in Bioorganic & medicinal chemistry letters (15.01.2016)
Published in Bioorganic & medicinal chemistry letters (15.01.2016)
Get full text
Journal Article
The flavoprotein FOXRED2 reductively activates nitro-chloromethylbenzindolines and other hypoxia-targeting prodrugs
Hunter, Francis W., Jaiswal, Jagdish K., Hurley, Daniel G., Liyanage, H.D. Sarath, McManaway, Sarah P., Gu, Yongchuan, Richter, Susan, Wang, Jingli, Tercel, Moana, Print, Cristin G., Wilson, William R., Pruijn, Frederik B.
Published in Biochemical pharmacology (15.05.2014)
Published in Biochemical pharmacology (15.05.2014)
Get full text
Journal Article
Photodegradation of the Benzotriazine 1,4-Di-N-Oxide Hypoxia-Activated Prodrug SN30000 in Aqueous Solution
Gu, Yongchuan, Jaiswal, Jagdish K., Wang, Jingli, Hicks, Kevin O., Hay, Michael P., Wilson, William R.
Published in Journal of pharmaceutical sciences (01.11.2014)
Published in Journal of pharmaceutical sciences (01.11.2014)
Get full text
Journal Article
Reductive Metabolism Influences the Toxicity and Pharmacokinetics of the Hypoxia-Targeted Benzotriazine Di-Oxide Anticancer Agent SN30000 in Mice
Gu, Yongchuan, Chang, Tony T-A, Wang, Jingli, Jaiswal, Jagdish K, Edwards, David, Downes, Noel J, Liyanage, H D Sarath, Lynch, Courtney R H, Pruijn, Frederik B, Hickey, Anthony J R, Hay, Michael P, Wilson, William R, Hicks, Kevin O
Published in Frontiers in pharmacology (11.08.2017)
Published in Frontiers in pharmacology (11.08.2017)
Get full text
Journal Article
Evidence that phospholipase C is involved in the antitumour action of NSC768313, a new thieno[2,3-b]pyridine derivative
Reynisson, Jóhannes, Jaiswal, Jagdish K, Barker, David, D'mello, Stacey A N, Denny, William A, Baguley, Bruce C, Leung, Euphemia Y
Published in Cancer cell international (10.03.2016)
Published in Cancer cell international (10.03.2016)
Get full text
Journal Article
Preclinical Activity and Pharmacokinetic/Pharmacodynamic Relationship for a Series of Novel Benzenesulfonamide Perforin Inhibitors
Gartlan, Kate H., Jaiswal, Jagdish K., Bull, Matthew R., Akhlaghi, Hedieh, Sutton, Vivien R., Alexander, Kylie A., Chang, Karshing, Hill, Geoffrey R., Miller, Christian K., O’Connor, Patrick D., Jose, Jiney, Trapani, Joseph A., Charman, Susan A., Spicer, Julie A., Jamieson, Stephen M. F.
Published in ACS pharmacology & translational science (10.06.2022)
Published in ACS pharmacology & translational science (10.06.2022)
Get full text
Journal Article