Discovery of a First-In-Class Small Molecule Antagonist against the Adrenomedullin‑2 Receptor: Structure–Activity Relationships and Optimization
Zirimwabagabo, Jean-Olivier, Jailani, Ameera B. A, Avgoustou, Paris, Tozer, Matthew J, Gibson, Karl R, Glossop, Paul A, Mills, James E. J, Porter, Roderick A, Blaney, Paul, Wang, Ning, Skerry, Timothy M, Richards, Gareth O, Harrity, Joseph P. A
Published in Journal of medicinal chemistry (25.03.2021)
Published in Journal of medicinal chemistry (25.03.2021)
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Receptor activity-modifying protein modulation of parathyroid hormone-1 receptor function and signaling
Avgoustou, Paris, Jailani, Ameera B A, Desai, Aditya J, Roberts, David J, Lilley, Ewan R, Stothard, Grant W, Skerry, Timothy M, Richards, Gareth O
Published in Frontiers in pharmacology (23.09.2024)
Published in Frontiers in pharmacology (23.09.2024)
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Journal Article
Discovery of a First-in-Class Potent Small Molecule Antagonist against the Adrenomedullin‑2 Receptor
Avgoustou, Paris, Jailani, Ameera B. A, Zirimwabagabo, Jean-Olivier, Tozer, Matthew J, Gibson, Karl R, Glossop, Paul A, Mills, James E. J, Porter, Roderick A, Blaney, Paul, Bungay, Peter J, Wang, Ning, Shaw, Alice P, Bigos, Kamilla J. A, Holmes, Joseph L, Warrington, Jessica I, Skerry, Timothy M, Harrity, Joseph P. A, Richards, Gareth O
Published in ACS pharmacology & translational science (14.08.2020)
Published in ACS pharmacology & translational science (14.08.2020)
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Targeting the adrenomedullin-2 receptor for the discovery and development of novel anti-cancer agents
Jailani, Ameera B. A., Bigos, Kamilla J. A., Avgoustou, Paris, Egan, Joseph L., Hathway, Robert A., Skerry, Timothy M., Richards, Gareth O.
Published in Expert opinion on drug discovery (03.08.2022)
Published in Expert opinion on drug discovery (03.08.2022)
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