The Interleukin‐1 Receptor–Associated Kinase 4 Inhibitor PF‐06650833 Blocks Inflammation in Preclinical Models of Rheumatic Disease and in Humans Enrolled in a Randomized Clinical Trial
Winkler, Aaron, Sun, Weiyong, De, Saurav, Jiao, Aiping, Sharif, M. Nusrat, Symanowicz, Peter T., Athale, Shruti, Shin, Julia H., Wang, Ju, Jacobson, Bruce A., Ramsey, Simeon J., Dower, Ken, Andreyeva, Tatyana, Liu, Heng, Hegen, Martin, Homer, Bruce L., Brodfuehrer, Joanne, Tilley, Mera, Gilbert, Steven A., Danto, Spencer I., Beebe, Jean J., Barnes, Betsy J., Pascual, Virginia, Lin, Lih‐Ling, Kilty, Iain, Fleming, Margaret, Rao, Vikram R.
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.12.2021)
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.12.2021)
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Quantifying NF-κB Activation by Flow Cytometry of IκBα Degradation
Veerasubramanian, Praveen Krishna, Jacobson, Bruce A, Karlsson, Fridrik J, Duffen, Jennifer L
Published in Current protocols (01.05.2024)
Published in Current protocols (01.05.2024)
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Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP)
Sulsky, Richard, Magnin, David R., Huang, Yanting, Simpkins, Ligaya, Taunk, Prakash, Patel, Manorama, Zhu, Yeheng, Stouch, Terry R., Bassolino-Klimas, Donna, Parker, Rex, Harrity, Thomas, Stoffel, Robert, Taylor, David S., Lavoie, Thomas B., Kish, Kevin, Jacobson, Bruce L., Sheriff, Steven, Adam, Leonard P., Ewing, William R., Robl, Jeffrey A.
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
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IL-13 blockade reduces lung inflammation after Ascaris suum challenge in cynomolgus monkeys
Bree, Andrea, BS, Schlerman, Franklin J., BS, Wadanoli, Michael, DVM, Tchistiakova, Lioudmila, PhD, Marquette, Kimberly, BS, Tan, Xiang-Yang, MD, PhD, Jacobson, Bruce A., PhD, Widom, Angela, MS, Cook, Timothy A., BS, Wood, Nancy, BS, Vunnum, Suresh, PhD, Krykbaev, Rustem, PhD, Xu, Xin, PhD, Donaldson, Debra D., MD, Goldman, Samuel J., PhD, Sypek, Joseph, PhD, Kasaian, Marion T., PhD
Published in Journal of allergy and clinical immunology (01.05.2007)
Published in Journal of allergy and clinical immunology (01.05.2007)
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Human Alveolar Macrophage Gene Responses to Mycobacterium tuberculosis Strains H37Ra and H37Rv
Silver, Richard F, Walrath, Jessica, Lee, Hung, Jacobson, Bruce A, Horton, Heidi, Bowman, Michael R, Nocka, Karl, Sypek, Joseph P
Published in American journal of respiratory cell and molecular biology (01.04.2009)
Published in American journal of respiratory cell and molecular biology (01.04.2009)
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Regulation and function of the interleukin 13 receptor alpha 2 during a T helper cell type 2-dominant immune response
Chiaramonte, Monica G, Mentink-Kane, Margaret, Jacobson, Bruce A, Cheever, Allen W, Whitters, Matthew J, Goad, Mary E P, Wong, Anthony, Collins, Mary, Donaldson, Debra D, Grusby, Michael J, Wynn, Thomas A
Published in The Journal of experimental medicine (17.03.2003)
Published in The Journal of experimental medicine (17.03.2003)
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Enhanced interleukin (IL)-13 responses in mice lacking IL-13 receptor alpha 2
Wood, Nancy, Whitters, Matthew J, Jacobson, Bruce A, Witek, JoAnn, Sypek, Joseph P, Kasaian, Marion, Eppihimer, Michael J, Unger, Michelle, Tanaka, Takashi, Goldman, Samuel J, Collins, Mary, Donaldson, Debra D, Grusby, Michael J
Published in The Journal of experimental medicine (17.03.2003)
Published in The Journal of experimental medicine (17.03.2003)
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Efficacy of IL-13 Neutralization in a Sheep Model of Experimental Asthma
Kasaian, Marion T, Donaldson, Debra D, Tchistiakova, Lioudmila, Marquette, Kimberly, Tan, Xiang-Yang, Ahmed, Ashfaq, Jacobson, Bruce A, Widom, Angela, Cook, Timothy A, Xu, Xin, Barry, Anthony B, Goldman, Samuel J, Abraham, William M
Published in American journal of respiratory cell and molecular biology (01.03.2007)
Published in American journal of respiratory cell and molecular biology (01.03.2007)
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Isolation, Cloning, and Localization of Rat PV-1, a Novel Endothelial Caveolar Protein
Stan, Radu-Virgil, Ghitescu, Lucian, Jacobson, Bruce S., Palade, George E.
Published in The Journal of cell biology (14.06.1999)
Published in The Journal of cell biology (14.06.1999)
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Characterization of MMP-9 and -12 KO mice in a model of acute smoke exposure
Schlerman, Franklin J, Kubera, John E, Pazdziorko, Stephen P, Bowman, Michael R, Jacobson, Bruce A, Fleming, Margaret, Williams, Cara MM, Sypek, Joseph P
Published in Journal of inflammation (London, England) (14.08.2013)
Published in Journal of inflammation (London, England) (14.08.2013)
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Solid-phase synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors
SUTTON, James C, BOLTON, Scott A, BISACCHI, Gregory S, DAVIS, Malcolm E, HARTL, Karen S, JACOBSON, Bruce, MATHUR, Arvind, OGLETREE, Martin L, SLUSARCHYK, William A, ZAHLER, Robert, SEILER, Steven M
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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Tumor cells secreting IL‐13 but not IL‐13Rα2 fusion protein have reduced tumorigenicity in vivo
Ma, Hak‐Ling, Whitters, Matthew J., Jacobson, Bruce A., Donaldson, Deborah D., Collins, Mary, Dunussi‐Joannopoulos, Kyriaki
Published in International immunology (01.07.2004)
Published in International immunology (01.07.2004)
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Analysis of Biosensor Chips for Identification of Nucleic Acids
Arlinghaus, Heinrich F, Kwoka, Margaret N, Jacobson, K. Bruce
Published in Analytical chemistry (Washington) (15.09.1997)
Published in Analytical chemistry (Washington) (15.09.1997)
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Cdc42 and RhoA are differentially regulated during arachidonate-mediated HeLa cell adhesion
Roberts, Louis A., Glenn, Honor, Hahn, Chang S., Jacobson, Bruce S.
Published in Journal of cellular physiology (01.07.2003)
Published in Journal of cellular physiology (01.07.2003)
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