Development and Proof of Concept for a Large-Scale Photoredox Additive-Free Minisci Reaction
Graham, Mark A., Noonan, Gary, Cherryman, Janette H., Douglas, James J., Gonzalez, Miguel, Jackson, Lucinda V., Leslie, Kevin, Liu, Zhi-qing, McKinney, David, Munday, Rachel H., Parsons, Chris D., Whittaker, David T. E., Zhang, En-xuan, Zhang, Jun-wang
Published in Organic process research & development (15.01.2021)
Published in Organic process research & development (15.01.2021)
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An Orally Bioavailable, Indole-3-glyoxylamide Based Series of Tubulin Polymerization Inhibitors Showing Tumor Growth Inhibition in a Mouse Xenograft Model of Head and Neck Cancer
Colley, Helen E, Muthana, Munitta, Danson, Sarah J, Jackson, Lucinda V, Brett, Matthew L, Harrison, Joanne, Coole, Sean F, Mason, Daniel P, Jennings, Luke R, Wong, Melanie, Tulasi, Vamshi, Norman, Dennis, Lockey, Peter M, Williams, Lynne, Dossetter, Alexander G, Griffen, Edward J, Thompson, Mark J
Published in Journal of medicinal chemistry (10.12.2015)
Published in Journal of medicinal chemistry (10.12.2015)
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Development and Scale-Up of an Improved Manufacturing Route to the ATR Inhibitor Ceralasertib
Graham, Mark A., Askey, Hannah, Campbell, Andrew D., Chan, Lai, Cooper, Katie G., Cui, Zhaoshan, Dalgleish, Andrew, Dave, David, Ensor, Gareth, Espinosa, Maria Rita Galan, Hamilton, Peter, Heffernan, Claire, Jackson, Lucinda, Jing, Dajiang, Jones, Martin F., Liu, Pengpeng, Mulholland, Keith R., Pervez, Mohammed, Popadynec, Michael, Randles, Emma, Tomasi, Simone, Wang, Shenghua
Published in Organic process research & development (15.01.2021)
Published in Organic process research & development (15.01.2021)
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Synthetic Route Design of AZD4635, an A(2A)R Antagonist
Littleson, Mairi M., Campbell, Andrew D., Clarke, Adam, Dow, Mark, Ensor, Gareth, Evans, Matthew C., Herring, Adam, Jackson, Bethany A., Jackson, Lucinda V., Karlsson, Staffan, Klauber, David J., Legg, Danny H., Leslie, Kevin W., Moravcik, Stefan, Parsons, Chris D., Ronson, Thomas O., Meadows, Rebecca E.
Published in Organic process research & development (01.07.2019)
Published in Organic process research & development (01.07.2019)
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Journal Article
Synthetic Route Design of AZD4635, an A 2A R Antagonist
Littleson, Mairi M., Campbell, Andrew D., Clarke, Adam, Dow, Mark, Ensor, Gareth, Evans, Matthew C., Herring, Adam, Jackson, Bethany A., Jackson, Lucinda V., Karlsson, Staffan, Klauber, David J., Legg, Danny H., Leslie, Kevin W., Moravčík, Štefan, Parsons, Chris D., Ronson, Thomas O., Meadows, Rebecca E.
Published in Organic process research & development (19.07.2019)
Published in Organic process research & development (19.07.2019)
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PHARMACEUTICAL PROCESS AND INTERMEDIATES
INGLESBY PHILLIP ANTHONY, JACKSON LUCINDA V, GRAHAM MARK ANDREW, DAVE DAVID PRANAY, NOONAN GARY MICHAEL, COOPER KATIE G
Year of Publication 30.07.2021
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Year of Publication 30.07.2021
Patent
PROCESSES FOR THE PREPARATION OF 4-{8-AMINO-3-[(2S)-1-(BUT-2-YNOYL)-PYRROLIDIN-2-YL]IMIDAZO[1,5-A]-PYRAZIN-1-YL}N-(PYRIDIN-2-YL)-BENZAMIDE
VAN EIJK PETER J S S, CHAN LAI C, PHILLIPS ANDREW J, COX ROBERT J, EVARTS JERRY, ZIJP ERIC J, BETHEL PAUL A, HUGHES SHAUN A, SHORT DAVID A, GOLDEN MICHAEL D, VERSTAPPEN MATHILDA M H, LITJENS REMY E J N, JACKSON LUCINDA V, GARREY RUSTAM F, LAWLER MICHAEL J, WANG ALEXANDRA, MILLARD KIRSTY J, TELFORD ALEXANDER J, VOS FRANK L M, JUNYING QIU, COOPER KATIE G
Year of Publication 09.04.2021
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Year of Publication 09.04.2021
Patent