Discovery of a Series of Phosphonic Acid-Containing Thiazoles and Orally Bioavailable Diamide Prodrugs That Lower Glucose in Diabetic Animals Through Inhibition of Fructose-1,6-Bisphosphatase
Dang, Qun, Liu, Yan, Cashion, Daniel K, Kasibhatla, Srinivas Rao, Jiang, Tao, Taplin, Frank, Jacintho, Jason D, Li, Haiqing, Sun, Zhili, Fan, Yi, DaRe, Jay, Tian, Feng, Li, Wenyu, Gibson, Tony, Lemus, Robert, van Poelje, Paul D, Potter, Scott C, Erion, Mark D
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
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Discovery of potent and selective PPARα/δ dual antagonists and initial biological studies
Jacintho, Jason D., Baccei, Christopher S., Bravo, Yalda, Broadhead, Alex, Chen, Austin, Correa, Lucia, Fischer, Kim, Laffitte, Bryan, Lee, Catherine, Lorrain, Daniel S., Messmer, Davorka, Prasit, Peppi, Stebbins, Karin J., Stock, Nicholas S.
Published in Bioorganic & medicinal chemistry letters (01.02.2019)
Published in Bioorganic & medicinal chemistry letters (01.02.2019)
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Identification of the first potent, selective and bioavailable PPARα antagonist
Bravo, Yalda, Baccei, Christopher S., Broadhead, Alex, Bundey, Richard, Chen, Austin, Clark, Ryan, Correa, Lucia, Jacintho, Jason D., Lorrain, Daniel S., Messmer, Davorka, Stebbins, Karin, Prasit, Peppi, Stock, Nicholas
Published in Bioorganic & medicinal chemistry letters (15.05.2014)
Published in Bioorganic & medicinal chemistry letters (15.05.2014)
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Synthesis and Biological Evaluation of a Series of Liver-Selective Phosphonic Acid Thyroid Hormone Receptor Agonists and Their Prodrugs
Boyer, Serge H, Jiang, Hongjian, Jacintho, Jason D, Reddy, Mali Venkat, Li, Haiqing, Li, Wenyu, Godwin, Jennifer L, Schulz, William G, Cable, Edward E, Hou, Jinzhao, Wu, Rongrong, Fujitaki, James M, Hecker, Scott J, Erion, Mark D
Published in Journal of medicinal chemistry (27.11.2008)
Published in Journal of medicinal chemistry (27.11.2008)
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A Selective Novel Peroxisome Proliferator-Activated Receptor (PPAR)-α Antagonist Induces Apoptosis and Inhibits Proliferation of CLL Cells In Vitro and In Vivo
Messmer, Davorka, Lorrain, Kymmy, Stebbins, Karin, Bravo, Yalda, Stock, Nicholas, Cabrera, Geraldine, Correa, Lucia, Chen, Austin, Jacintho, Jason, Chiorazzi, Nicholas, Yan, Xiao Jie, Spaner, David, Prasit, Peppi, Lorrain, Daniel
Published in Molecular medicine (Cambridge, Mass.) (09.06.2015)
Published in Molecular medicine (Cambridge, Mass.) (09.06.2015)
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Erratum to: A Selective Novel Peroxisome Proliferator-Activated Receptor (PPAR)-α Antagonist Induces Apoptosis and Inhibits Proliferation of CLL Cells In Vitro and In Vivo
Messmer, Davorka, Lorrain, Kymmy, Stebbins, Karin, Bravo, Yalda, Stock, Nicholas, Cabrera, Geraldine, Correa, Lucia, Chen, Austin, Jacintho, Jason, Chiorazzi, Nicholas, Yan, Xiao Jie, Spaner, David, Prasit, Peppi, Lorrain, Daniel
Published in Molecular medicine (Cambridge, Mass.) (01.01.2015)
Published in Molecular medicine (Cambridge, Mass.) (01.01.2015)
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Inhibition of Fatty Acid Oxidation Leads to Apoptosis of Resting and Proliferating Chronic Lymphocytic Leukemia Cells in Vitro
Messmer, Davorka, Lorrain, Kymmy, Bravo, Yalda, Stock, Nicholas, Bundey, Richard, Correa, Lucia, Poon, Michael M, Stebbins, Karin, Cabrera, Geraldine, Chen, Austin, Jacintho, Jason, Spaner, David, Prasit, Peppi, Lorrain, Daniel
Published in Blood (16.11.2012)
Published in Blood (16.11.2012)
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TRIAZOLONE COMPOUNDS AND USES THEREOF
STOCK NICHOLAS SIMON, BRAVO YALDA MOSTOFI, JACINTHO JASON DUARTE, CHEN AUSTIN CHIH YU
Year of Publication 04.05.2016
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Year of Publication 04.05.2016
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PYRAZOLONE COMPOUNDS AND USES THEREOF
STOCK NICHOLAS SIMON, BRAVO YALDA MOSTOFI, TRUONG YEN, JACINTHO JASON DUARTE, CHEN AUSTIN CHIH YU
Year of Publication 06.10.2016
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Year of Publication 06.10.2016
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TRIAZOLONE COMPOUNDS AND USES THEREOF
STOCK NICHOLAS SIMON, BRAVO YALDA MOSTOFI, CLARK RYAN CHRISTOPHER, STEARNS BRIAN ANDREW, JACINTHO JASON DUARTE, CHEN AUSTIN CHIH YU, BACCEI JILL MELISSA
Year of Publication 31.08.2015
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Year of Publication 31.08.2015
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METALLOENZYMES FOR BIOMOLECULAR RECOGNITION OF N-TERMINAL MODIFIED PEPTIDES
VERESPY, Stephen III, OKERBERG, Eric, MILES, Zachary, GANGULY, Soumya, WISE, Aaron, KLIMA, Jason, C, JACINTHO, Jason, Duarte
Year of Publication 08.11.2023
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Year of Publication 08.11.2023
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Mechanisms of action of DNA intercalating acridine-based drugs: How important are contributions from electron transfer and oxidative stress? : Oxidative stress
BAGULEY, Bruce C, WAKELIN, Laurence P. G, JACINTHO, Jason D, KOVACIC, Peter
Published in Current medicinal chemistry (2003)
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Published in Current medicinal chemistry (2003)
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