Discovery of Orally Active Inhibitors of Brahma Homolog (BRM)/SMARCA2 ATPase Activity for the Treatment of Brahma Related Gene 1 (BRG1)/SMARCA4-Mutant Cancers
Papillon, Julien P. N, Nakajima, Katsumasa, Adair, Christopher D, Hempel, Jonathan, Jouk, Andriana O, Karki, Rajeshri G, Mathieu, Simon, Möbitz, Henrik, Ntaganda, Rukundo, Smith, Troy, Visser, Michael, Hill, Susan E, Hurtado, Felipe Kellermann, Chenail, Gregg, Bhang, Hyo-Eun C, Bric, Anka, Xiang, Kay, Bushold, Geoffrey, Gilbert, Tamara, Vattay, Anthony, Dooley, Julie, Costa, Emily A, Park, Isabel, Li, Ailing, Farley, David, Lounkine, Eugen, Yue, Q. Kimberley, Xie, Xiaoling, Zhu, Xiaoping, Kulathila, Raviraj, King, Daniel, Hu, Tiancen, Vulic, Katarina, Cantwell, John, Luu, Catherine, Jagani, Zainab
Published in Journal of medicinal chemistry (21.11.2018)
Published in Journal of medicinal chemistry (21.11.2018)
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Journal Article
Discovery of Darovasertib (NVP-LXS196), a Pan-PKC Inhibitor for the Treatment of Metastatic Uveal Melanoma
Visser, Michael, Papillon, Julien P. N., Luzzio, Michael, LaMarche, Matthew J., Fan, Jianmei, Michael, Walter, Wang, David, Zhang, Alan, Straub, Christopher, Mathieu, Simon, Kato, Mitsunori, Palermo, Mark, Chen, Christine, Ramsey, Timothy, Joud, Carol, Barrett, Rosemary, Vattay, Anthony, Guo, Ribo, Bric, Anka, Chung, Franklin, Liang, Guiqing, Romanowski, Michael J., Lam, Joni, Thohan, Sanjeev, Atassi, Faraj, Wylie, Andrew, Cooke, Vesselina G.
Published in Journal of medicinal chemistry (25.01.2024)
Published in Journal of medicinal chemistry (25.01.2024)
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Journal Article
Structure–Activity Relationships, Pharmacokinetics, and in Vivo Activity of CYP11B2 and CYP11B1 Inhibitors
Papillon, Julien P. N, Adams, Christopher M, Hu, Qi-Ying, Lou, Changgang, Singh, Alok K, Zhang, Chun, Carvalho, Jose, Rajan, Srinivan, Amaral, Adam, Beil, Michael E, Fu, Fumin, Gangl, Eric, Hu, Chii-Whei, Jeng, Arco Y, LaSala, Daniel, Liang, Guiqing, Logman, Michael, Maniara, Wieslawa M, Rigel, Dean F, Smith, Sherri A, Ksander, Gary M
Published in Journal of medicinal chemistry (11.06.2015)
Published in Journal of medicinal chemistry (11.06.2015)
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Journal Article
Discovery of a novel indole pharmacophore for the irreversible inhibition of myeloperoxidase (MPO)
Patnaik, Anup, Axford, Laura, Deng, Lin, Cohick, Evan, Ren, Xianglin, Loi, Sally, Kecman, Sam, Hollis-Symynkywicz, Micah, Harrison, Tyler J., Papillon, Julien P.N., Dales, Natalie, Hamann, Lawrence G., Lee, Lac, Regard, Jean B., Marcinkeviciene, Jovita, Marro, Martin L., Patterson, Andrew W.
Published in Bioorganic & medicinal chemistry (15.06.2020)
Published in Bioorganic & medicinal chemistry (15.06.2020)
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Journal Article
The Discovery of SWI/SNF Chromatin Remodeling Activity as a Novel and Targetable Dependency in Uveal Melanoma
Rago, Florencia, Elliott, GiNell, Li, Ailing, Sprouffske, Kathleen, Kerr, Grainne, Desplat, Aurore, Abramowski, Dorothee, Chen, Julie T., Farsidjani, Ali, Xiang, Kay X., Bushold, Geoffrey, Feng, Yun, Shirley, Matthew D., Bric, Anka, Vattay, Anthony, Möbitz, Henrik, Nakajima, Katsumasa, Adair, Christopher D., Mathieu, Simon, Ntaganda, Rukundo, Smith, Troy, Papillon, Julien P.N., Kauffmann, Audrey, Ruddy, David A., Bhang, Hyo-eun C., Castelletti, Deborah, Jagani, Zainab
Published in Molecular cancer therapeutics (01.10.2020)
Published in Molecular cancer therapeutics (01.10.2020)
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Journal Article
Discovery of N‑[5-(6-Chloro-3-cyano-1-methyl‑1H‑indol-2-yl)-pyridin-3-ylmethyl]-ethanesulfonamide, a Cortisol-Sparing CYP11B2 Inhibitor that Lowers Aldosterone in Human Subjects
Papillon, Julien P. N, Lou, Changgang, Singh, Alok K, Adams, Christopher M, Ksander, Gary M, Beil, Michael E, Chen, Wei, Leung-Chu, Jennifer, Fu, Fumin, Gan, Lu, Hu, Chii-Whei, Jeng, Arco Y, LaSala, Daniel, Liang, Guiqing, Rigel, Dean F, Russell, Kerry S, Vest, John A, Watson, Catherine
Published in Journal of medicinal chemistry (10.12.2015)
Published in Journal of medicinal chemistry (10.12.2015)
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Journal Article
Ocular Pharmacology and Toxicology of TRPV1 Antagonist SAF312 (Libvatrep)
Mogi, Muneto, Mendonza, Anisha E., Chastain, James, Demirs, John T., Medley, Quintus G., Zhang, Qin, Papillon, Julien P. N., Yang, Junzheng, Gao, Yan, Xu, YongYao, Stasi, Kalliopi
Published in Translational vision science & technology (01.09.2023)
Published in Translational vision science & technology (01.09.2023)
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Journal Article
Discovery and in Vivo Evaluation of Potent Dual CYP11B2 (Aldosterone Synthase) and CYP11B1 Inhibitors
Meredith, Erik L, Ksander, Gary, Monovich, Lauren G, Papillon, Julien P. N, Liu, Qian, Miranda, Karl, Morris, Patrick, Rao, Chang, Burgis, Robin, Capparelli, Michael, Hu, Qi-Ying, Singh, Alok, Rigel, Dean F, Jeng, Arco Y, Beil, Michael, Fu, Fumin, Hu, Chii-Whei, LaSala, Daniel
Published in ACS medicinal chemistry letters (12.12.2013)
Published in ACS medicinal chemistry letters (12.12.2013)
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Journal Article
Discovery of 1-((6-Aminopyridin-3-yl)Methyl)-3-(4-Bromophenyl)Urea as a Potent, Irreversible Myeloperoxidase Inhibitor
Marro, Martin L, Patterson, Andrew W, Lee, Lac, Deng, Lin, Reynolds, Aimee, Ren, Xianglin, Axford, Laura, Patnaik, Anup, Hollis-Symynkywicz, Micah, Casson, Nigel, Custeau, Dominique, Ames, Lisa, Loi, Sally, Zhang, Lihe, Honda, Toshiyuki, Blank, Jutta, Harrison, Tyler J, Papillon, Julien P N, Hamann, Lawrence G, Marcinkeviciene, Jovita, Regard, Jean B
Published in The Journal of pharmacology and experimental therapeutics (01.10.2018)
Published in The Journal of pharmacology and experimental therapeutics (01.10.2018)
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Journal Article
Synthetic phospholipids as specific substrates for plasma endothelial lipase
Papillon, Julien P.N., Pan, Meihui, Brousseau, Margaret E., Gilchrist, Mark A., Lou, Changgang, Singh, Alok K., Stawicki, Todd, Thompson, James E.
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
Published in Bioorganic & medicinal chemistry letters (01.08.2016)
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Journal Article
Formal synthesis of (+)-neooxazolomycin via a Stille cross-coupling/deconjugation route
Bastin, Reyhan, Dale, James W., Edwards, Michael G., Papillon, Julien P.N., Webb, Michael R., Taylor, Richard J.K.
Published in Tetrahedron (23.12.2011)
Published in Tetrahedron (23.12.2011)
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Journal Article
Ru-Catalyzed Alkene−Alkyne Coupling. Total Synthesis of Amphidinolide P
Trost, Barry M, Papillon, Julien P. N, Nussbaumer, Thomas
Published in Journal of the American Chemical Society (21.12.2005)
Published in Journal of the American Chemical Society (21.12.2005)
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Journal Article
Alkene−Alkyne Coupling as a Linchpin: An Efficient and Convergent Synthesis of Amphidinolide P
Trost, Barry M, Papillon, Julien P. N
Published in Journal of the American Chemical Society (27.10.2004)
Published in Journal of the American Chemical Society (27.10.2004)
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Journal Article
New synthetic method for the polymerization of alkylthiophenes
Se´vignon, Marc, Papillon, Julien, Schulz, Emmanuelle, Lemaire, Marc
Published in Tetrahedron letters (06.08.1999)
Published in Tetrahedron letters (06.08.1999)
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Journal Article
Towards the preparation of modified chiral electrodes for heterogeneous asymmetric catalysis: synthesis and electrochemical properties of ( S,S)-5,5′-bis-[3-(3-methyl-pentyl)-thiophen-2-yl]-[2,2′]-bipyridine
Papillon, Julien, Schulz, Emmanuelle, Gélinas, Stéphane, Lessard, Jean, Lemaire, Marc
Published in Synthetic metals (30.07.1998)
Published in Synthetic metals (30.07.1998)
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Journal Article
Formal synthesis of (+)-neooxazolomycin via a Stille cross-coupling/ deconjugation route: Organic Synthesis-2011: Perspective, Journeys, and Accounts
BASTIN, Reyhan, DALE, James W, EDWARDS, Michael G, PAPILLON, Julien P. N, WEBB, Michael R, TAYLOR, Richard J. K
Published in Tetrahedron (2011)
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Published in Tetrahedron (2011)
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