Selective estrogen receptor degraders with novel structural motifs induce regression in a tamoxifen-resistant breast cancer xenograft
Govek, Steven P., Bonnefous, Celine, Julien, Jackaline D., Nagasawa, Johnny Y., Kahraman, Mehmet, Lai, Andiliy G., Douglas, Karensa L., Aparicio, Anna M., Darimont, Beatrice D., Grillot, Katherine L., Joseph, James D., Kaufman, Joshua A., Lee, Kyoung-Jin, Lu, Nhin, Moon, Michael J., Prudente, Rene Y., Sensintaffar, John, Rix, Peter J., Hager, Jeffrey H., Smith, Nicholas D.
Published in Bioorganic & medicinal chemistry letters (01.02.2019)
Published in Bioorganic & medicinal chemistry letters (01.02.2019)
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Journal Article
POLYCYCLIC ESTROGEN RECEPTOR MODULATORS AND USES THEREOF
GOVEK STEVEN P, BONNEFOUS CELINE, JULIEN JACKALINE D, KAHRAMAN MEHMET, SMITH NICHOLAS D
Year of Publication 20.11.2015
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Year of Publication 20.11.2015
Patent
ESTROGEN RECEPTOR MODULATORS AND USES THEREOF
LAI ANDILIY G, GOVEK STEVEN P, BONNEFOUS CELINE, JULIEN JACKALINE D, NAGASAWA JOHNNY Y, KAHRAMAN MEHMET, DOUGLAS KARENSA L, SMITH NICHOLAS D
Year of Publication 03.12.2014
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Year of Publication 03.12.2014
Patent
The selective estrogen receptor downregulator GDC-0810 is efficacious in diverse models of ER+ breast cancer
Joseph, James D, Darimont, Beatrice, Zhou, Wei, Arrazate, Alfonso, Young, Amy, Ingalla, Ellen, Walter, Kimberly, Blake, Robert A, Nonomiya, Jim, Guan, Zhengyu, Kategaya, Lorna, Govek, Steven P, Lai, Andiliy G, Kahraman, Mehmet, Brigham, Dan, Sensintaffar, John, Lu, Nhin, Shao, Gang, Qian, Jing, Grillot, Kate, Moon, Michael, Prudente, Rene, Bischoff, Eric, Lee, Kyoung-Jin, Bonnefous, Celine, Douglas, Karensa L, Julien, Jackaline D, Nagasawa, Johnny Y, Aparicio, Anna, Kaufman, Josh, Haley, Benjamin, Giltnane, Jennifer M, Wertz, Ingrid E, Lackner, Mark R, Nannini, Michelle A, Sampath, Deepak, Schwarz, Luis, Manning, Henry Charles, Tantawy, Mohammed Noor, Arteaga, Carlos L, Heyman, Richard A, Rix, Peter J, Friedman, Lori, Smith, Nicholas D, Metcalfe, Ciara, Hager, Jeffrey H
Published in eLife (13.07.2016)
Published in eLife (13.07.2016)
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Journal Article
ESTROGEN RECEPTOR MODULATORS AND USES THEREOF
LAI ANDILIY G, GOVEK STEVEN P, BONNEFOUS CELINE, NAGASAWA JOHNNY Y, JULIEN JACKALINE D, KAHRAMAN MEHMET, HERBERT MARK R, DOUGLAS KARENSA L, SMITH NICHOLAS D
Year of Publication 13.12.2013
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Year of Publication 13.12.2013
Patent
Estrogen receptor modulators and uses thereof
Julien, Jackaline, D, Govek, Steven, P, Bonnefous, Celine, Douglas, Karensa L, Lai, Andiliy, G, Smith, Nicholas, D, Nagasawa, Johnny, Y, Kahraman, Mehmet, Herbert, Mark R
Year of Publication 15.11.2023
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Year of Publication 15.11.2023
Patent