Cyclodepsipeptides: a rich source of biologically active compounds for drug research
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Toward More Selective Antibiotic Inhibitors: A Structural View of the Complexed Binding Pocket of E. coli Peptide Deformylase
Kirschner, Hendrik, Heister, Nicole, Zouatom, Manuela, Zhou, Tianyi, Hofmann, Eckhard, Scherkenbeck, Jürgen, Stoll, Raphael
Published in Journal of medicinal chemistry (25.04.2024)
Published in Journal of medicinal chemistry (25.04.2024)
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Synthesis, Biological Evaluation, and Binding Mode of a New Class of Oncogenic K‐Ras4b Inhibitors
Jeuken, Stephan, Shkura, Oleksandr, Röger, Marc, Brickau, Victoria, Choidas, Axel, Degenhart, Carsten, Gülden, Daniel, Klebl, Bert, Koch, Uwe, Stoll, Raphael, Scherkenbeck, Jürgen
Published in ChemMedChem (18.11.2022)
Published in ChemMedChem (18.11.2022)
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Structural Insights into Antibacterial Payload Release from Gold Nanoparticles Bound to E. coli Peptide Deformylase
Kirschner, Hendrik, John, Milena, Zhou, Tianyi, Bachmann, Nathalie, Schultz, André, Hofmann, Eckhard, Bandow, Julia Elisabeth, Scherkenbeck, Jürgen, Metzler‐Nolte, Nils, Stoll, Raphael
Published in ChemMedChem (15.03.2024)
Published in ChemMedChem (15.03.2024)
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The Bisphenol A analogue Bisphenol S binds to K‐Ras4B – implications for ‘BPA‐free’ plastics
Schöpel, Miriam, Herrmann, Christian, Scherkenbeck, Jürgen, Stoll, Raphael, Griesinger, Christian
Published in FEBS letters (01.02.2016)
Published in FEBS letters (01.02.2016)
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Sequence‐Selective Covalent CaaX‐Box Receptors Prevent Farnesylation of Oncogenic Ras Proteins and Impact MAPK/PI3 K Signaling
Franz, Matthias, Mörchen, Britta, Degenhart, Carsten, Gülden, Daniel, Shkura, Oleksandr, Wolters, Dirk, Koch, Uwe, Klebl, Bert, Stoll, Raphael, Helfrich, Iris, Scherkenbeck, Jürgen
Published in ChemMedChem (19.08.2021)
Published in ChemMedChem (19.08.2021)
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Small Molecules Antagonise the MIA-Fibronectin Interaction in Malignant Melanoma
Yip, King Tuo, Zhong, Xue Yin, Seibel, Nadia, Pütz, Stefanie, Autzen, Jasmin, Gasper, Raphael, Hofmann, Eckhard, Scherkenbeck, Jürgen, Stoll, Raphael
Published in Scientific reports (06.05.2016)
Published in Scientific reports (06.05.2016)
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Rottlerin: Structure Modifications and KCNQ1/KCNE1 Ion Channel Activity
Lübke, Marco, Schreiber, Julian A., Le Quoc, Thang, Körber, Florian, Müller, Jasmin, Sivanathan, Sivatharushan, Matschke, Veronika, Schubert, Janina, Strutz‐Seebohm, Nathalie, Seebohm, Guiscard, Scherkenbeck, Jürgen
Published in ChemMedChem (17.06.2020)
Published in ChemMedChem (17.06.2020)
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Bisphenol A Binds to Ras Proteins and Competes with Guanine Nucleotide Exchange: Implications for GTPase-Selective Antagonists
Schöpel, Miriam, Jockers, Katharina F. G, Düppe, Peter M, Autzen, Jasmin, Potheraveedu, Veena N, Ince, Semra, Yip, King Tuo, Heumann, Rolf, Herrmann, Christian, Scherkenbeck, Jürgen, Stoll, Raphael
Published in Journal of medicinal chemistry (12.12.2013)
Published in Journal of medicinal chemistry (12.12.2013)
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Anthelmintic PF1022A: stepwise solid-phase synthesis of a cyclodepsipeptide containing N-methyl amino acids
Lüttenberg, Sebastian, Sondermann, Frank, Scherkenbeck, Jürgen
Published in Tetrahedron (25.02.2012)
Published in Tetrahedron (25.02.2012)
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Structural Prerequisites for Receptor Binding of Helicokinin I, a Diuretic Insect Neuropeptide from Helicoverpa zea
Van, Chien Tran, Zdobinsky, Tino, Seebohm, Guiscard, Nennstiel, Dirk, Zerbe, Oliver, Scherkenbeck, Jürgen
Published in European journal of organic chemistry (01.05.2014)
Published in European journal of organic chemistry (01.05.2014)
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The Natural Plant Product Rottlerin Activates Kv7.1/KCNE1 Channels
Matschke, Veronika, Piccini, Ilaria, Schubert, Janina, Wrobel, Eva, Lang, Florian, Matschke, Johann, Amedonu, Elsie, Meuth, Sven G., Strünker, Timo, Strutz-Seebohm, Nathalie, Greber, Boris, Scherkenbeck, Jürgen, Seebohm, Guiscard
Published in Cellular physiology and biochemistry (01.01.2016)
Published in Cellular physiology and biochemistry (01.01.2016)
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Segment Solid-Phase Total Synthesis of the Anthelmintic Cyclooctadepsipeptides PF1022A and Emodepside
Scherkenbeck, Jürgen, Lüttenberg, Sebastian, Ludwig, Monika, Brücher, Karin, Kotthaus, Andreas
Published in European Journal of Organic Chemistry (01.03.2012)
Published in European Journal of Organic Chemistry (01.03.2012)
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