Structure of the PAPP-ABP5 complex reveals mechanism of substrate recognition
Judge, Russell A., Sridar, Janani, Tunyasuvunakool, Kathryn, Jain, Rinku, Wang, John C. K., Ouch, Christna, Xu, Jun, Mafi, Amirhossein, Nile, Aaron H., Remarcik, Clint, Smith, Corey L., Ghosh, Crystal, Xu, Chen, Stoll, Vincent, Jumper, John, Singh, Amoolya H., Eaton, Dan, Hao, Qi
Published in Nature communications (20.09.2022)
Published in Nature communications (20.09.2022)
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Author Correction: Structure of the PAPP-ABP5 complex reveals mechanism of substrate recognition
Judge, Russell A., Sridar, Janani, Tunyasuvunakool, Kathryn, Jain, Rinku, Wang, John C. K., Ouch, Christna, Xu, Jun, Mafi, Amirhossein, Nile, Aaron H., Remarcik, Clint, Smith, Corey L., Ghosh, Crystal, Xu, Chen, Stoll, Vincent, Jumper, John, Singh, Amoolya H., Eaton, Dan, Hao, Qi
Published in Nature communications (28.09.2022)
Published in Nature communications (28.09.2022)
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Identification and structure-based drug design of cell-active inhibitors of interleukin 17A at a novel C-terminal site
Goedken, Eric R, Argiriadi, Maria A, Dietrich, Justin D, Petros, Andrew M, Krishnan, Navasona, Panchal, Sanjay C, Qiu, Wei, Wu, Haihong, Zhu, Haizhong, Adams, Ashley M, Bodelle, Pierre M, Goguen, Lucas, Richardson, Paul L, Slivka, Peter F, Srikumaran, Myron, Upadhyay, Anup K, Wu, Bainan, Judge, Russell A, Vasudevan, Anil, Gopalakrishnan, Sujatha M, Cox, Philip B, Stoll, Vincent S, Sun, Chaohong
Published in Scientific reports (26.08.2022)
Published in Scientific reports (26.08.2022)
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Structure reveals function of the dual variable domain immunoglobulin (DVD-Ig™) molecule
Jakob, Clarissa G, Edalji, Rohinton, Judge, Russell A, DiGiammarino, Enrico, Li, Yingchun, Gu, Jijie, Ghayur, Tariq
Published in mAbs (01.05.2013)
Published in mAbs (01.05.2013)
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Cryo-EM structure of human PAPP-A2 and mechanism of substrate recognition
Sridar, Janani, Mafi, Amirhossein, Judge, Russell A., Xu, Jun, Kong, Kailyn A., Wang, John C. K., Stoll, Vincent S., Koukos, Georgios, Simon, Reyna J., Eaton, Dan, Bratkowski, Matthew, Hao, Qi
Published in Communications chemistry (28.10.2023)
Published in Communications chemistry (28.10.2023)
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Selective MCL-1 inhibitor ABBV-467 is efficacious in tumor models but is associated with cardiac troponin increases in patients
Yuda, Junichiro, Will, Christine, Phillips, Darren C., Abraham, Linu, Alvey, Cory, Avigdor, Abraham, Buck, Wayne, Besenhofer, Lauren, Boghaert, Erwin, Cheng, Dong, Cojocari, Dan, Doyle, Kelly, Hansen, T. Matthew, Huang, Kevin, Johnson, Eric F., Judd, Andrew S., Judge, Russell A., Kalvass, John C., Kunzer, Aaron, Lam, Lloyd T., Li, Rachel, Martin, Ruth L., Mastracchio, Anthony, Mitten, Mike, Petrich, Adam, Wang, Jin, Ward, James E., Zhang, Haichao, Wang, Xilu, Wolff, Johannes E., Bell-McGuinn, Katherine M., Souers, Andrew J.
Published in Communications medicine (25.10.2023)
Published in Communications medicine (25.10.2023)
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Neutron structure of the cyclic glucose-bound xylose isomerase E186Q mutant
Munshi, Parthapratim, Snell, Edward H., van der Woerd, Mark J., Judge, Russell A., Myles, Dean A. A., Ren, Zhong, Meilleur, Flora
Published in Acta crystallographica. Section D, Biological crystallography. (01.02.2014)
Published in Acta crystallographica. Section D, Biological crystallography. (01.02.2014)
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CD40/anti-CD40 antibody complexes which illustrate agonist and antagonist structural switches
Argiriadi, Maria A, Benatuil, Lorenzo, Dubrovska, Ievgeniia, Egan, David A, Gao, Lei, Greischar, Amy, Hardman, Jennifer, Harlan, John, Iyer, Ramesh B, Judge, Russell A, Lake, Marc, Perron, Denise C, Sadhukhan, Ramkrishna, Sielaff, Bernhard, Sousa, Silvino, Wang, Rui, McRae, Bradford L
Published in BMC molecular and cell biology (05.08.2019)
Published in BMC molecular and cell biology (05.08.2019)
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Minimising the payload solvent exposed hydrophobic surface area optimises the antibody-drug conjugate properties
Hobson, Adrian D, Zhu, Haizhong, Qiu, Wei, Judge, Russell A, Longenecker, Kenton
Published in MedChemComm (20.03.2024)
Published in MedChemComm (20.03.2024)
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Microgravity and Macromolecular Crystallography
Kundrot, Craig E, Judge, Russell A, Pusey, Marc L, Snell, Edward H
Published in Crystal growth & design (01.01.2001)
Published in Crystal growth & design (01.01.2001)
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Structure-Guided Design of a Series of MCL‑1 Inhibitors with High Affinity and Selectivity
Bruncko, Milan, Wang, Le, Sheppard, George S, Phillips, Darren C, Tahir, Stephen K, Xue, John, Erickson, Scott, Fidanze, Steve, Fry, Elizabeth, Hasvold, Lisa, Jenkins, Gary J, Jin, Sha, Judge, Russell A, Kovar, Peter J, Madar, David, Nimmer, Paul, Park, Chang, Petros, Andrew M, Rosenberg, Saul H, Smith, Morey L, Song, Xiaohong, Sun, Chaohong, Tao, Zhi-Fu, Wang, Xilu, Xiao, Yu, Zhang, Haichao, Tse, Chris, Leverson, Joel D, Elmore, Steven W, Souers, Andrew J
Published in Journal of medicinal chemistry (12.03.2015)
Published in Journal of medicinal chemistry (12.03.2015)
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Inhibition of MALT1 and BCL2 Induces Synergistic Antitumor Activity in Models of B-Cell Lymphoma
Plotnik, Joshua P., Richardson, Adam E., Yang, Haopeng, Rojas, Estela, Bontcheva, Velitchka, Dowell, Colleen, Parsons, Sydney, Wilson, Ashley, Ravanmehr, Vida, Will, Christine, Jung, Paul, Zhu, Haizhong, Partha, Sarathy Karunan, Panchal, Sanjay C., Mali, Raghuveer Singh, Kohlhapp, Frederick J., McClure, Ryan A., Ramathal, Cyril Y., George, Mariam D., Jhala, Manisha, Elsen, Nathaniel L., Qiu, Wei, Judge, Russell A., Pan, Chin, Mastracchio, Anthony, Henderson, Jared, Meulbroek, Jonathan A., Green, Michael R., Pappano, William N.
Published in Molecular cancer therapeutics (02.07.2024)
Published in Molecular cancer therapeutics (02.07.2024)
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The Effect of Temperature and Solution pH on the Nucleation of Tetragonal Lysozyme Crystals
Judge, Russell A., Jacobs, Randolph S., Frazier, Tyralynn, Snell, Edward H., Pusey, Marc L.
Published in Biophysical journal (01.09.1999)
Published in Biophysical journal (01.09.1999)
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Discovery of a Potent and Selective BCL‑XL Inhibitor with in Vivo Activity
Tao, Zhi-Fu, Hasvold, Lisa, Wang, Le, Wang, Xilu, Petros, Andrew M, Park, Chang H, Boghaert, Erwin R, Catron, Nathaniel D, Chen, Jun, Colman, Peter M, Czabotar, Peter E, Deshayes, Kurt, Fairbrother, Wayne J, Flygare, John A, Hymowitz, Sarah G, Jin, Sha, Judge, Russell A, Koehler, Michael F. T, Kovar, Peter J, Lessene, Guillaume, Mitten, Michael J, Ndubaku, Chudi O, Nimmer, Paul, Purkey, Hans E, Oleksijew, Anatol, Phillips, Darren C, Sleebs, Brad E, Smith, Brian J, Smith, Morey L, Tahir, Stephen K, Watson, Keith G, Xiao, Yu, Xue, John, Zhang, Haichao, Zobel, Kerry, Rosenberg, Saul H, Tse, Chris, Leverson, Joel D, Elmore, Steven W, Souers, Andrew J
Published in ACS medicinal chemistry letters (09.10.2014)
Published in ACS medicinal chemistry letters (09.10.2014)
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Tetragonal Chicken Egg White Lysozyme Solubility in Sodium Chloride Solutions
Forsythe, Elizabeth L, Judge, Russell A, Pusey, Marc L
Published in Journal of chemical and engineering data (01.05.1999)
Published in Journal of chemical and engineering data (01.05.1999)
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Identification of Selective Dual ROCK1 and ROCK2 Inhibitors Using Structure-Based Drug Design
Hobson, Adrian D, Judge, Russell A, Aguirre, Ana L, Brown, Brian S, Cui, Yifang, Ding, Ping, Dominguez, Eric, DiGiammarino, Enrico, Egan, David A, Freiberg, Gail M, Gopalakrishnan, Sujatha M, Harris, Christopher M, Honore, Marie P, Kage, Karen L, Kapecki, Nicolas J, Ling, Christopher, Ma, Junli, Mack, Helmut, Mamo, Mulugeta, Maurus, Stefan, McRae, Bradford, Moore, Nigel S, Mueller, Bernhard K, Mueller, Reinhold, Namovic, Marian T, Patel, Kaushal, Pratt, Steve D, Putman, C. Brent, Queeney, Kara L, Sarris, Kathy K, Schaffter, Lisa M, Stoll, Vincent, Vasudevan, Anil, Wang, Lei, Wang, Lu, Wirthl, William, Yach, Kimberly
Published in Journal of medicinal chemistry (27.12.2018)
Published in Journal of medicinal chemistry (27.12.2018)
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An anti-PD-1-GITR-L bispecific agonist induces GITR clustering-mediated T cell activation for cancer immunotherapy
Chan, Sarah, Belmar, Nicole, Ho, Sun, Rogers, Bryan, Stickler, Marcia, Graham, Michelle, Lee, Eileen, Tran, Ninian, Zhang, Dong, Gupta, Priyanka, Sho, Mien, MacDonough, Tracy, Woolley, Andrew, Kim, Han, Zhang, Hong, Liu, Wei, Zheng, Pingping, Dezso, Zoltan, Halliwill, Kyle, Ceccarelli, Michele, Rhodes, Susan, Thakur, Archana, Forsyth, Charles M, Xiong, Mengli, Tan, Siu Sze, Iyer, Ramesh, Lake, Marc, Digiammarino, Enrico, Zhou, Li, Bigelow, Lance, Longenecker, Kenton, Judge, Russell A, Liu, Cassie, Trumble, Max, Remis, Jonathan P, Fox, Melvin, Cairns, Belinda, Akamatsu, Yoshiko, Hollenbaugh, Diane, Harding, Fiona, Alvarez, Hamsell M
Published in Nature cancer (01.03.2022)
Published in Nature cancer (01.03.2022)
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