Discovery of GSK8612, a Highly Selective and Potent TBK1 Inhibitor
Thomson, Douglas W, Poeckel, Daniel, Zinn, Nico, Rau, Christina, Strohmer, Katrin, Wagner, Anne J, Graves, Alan P, Perrin, Jessica, Bantscheff, Marcus, Duempelfeld, Birgit, Kasparcova, Viera, Ramanjulu, Joshi M, Pesiridis, G. Scott, Muelbaier, Marcel, Bergamini, Giovanna
Published in ACS medicinal chemistry letters (09.05.2019)
Published in ACS medicinal chemistry letters (09.05.2019)
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Journal Article
Design of amidobenzimidazole STING receptor agonists with systemic activity
Ramanjulu, Joshi M, Pesiridis, G Scott, Yang, Jingsong, Concha, Nestor, Singhaus, Robert, Zhang, Shu-Yun, Tran, Jean-Luc, Moore, Patrick, Lehmann, Stephanie, Eberl, H Christian, Muelbaier, Marcel, Schneck, Jessica L, Clemens, Jim, Adam, Michael, Mehlmann, John, Romano, Joseph, Morales, Angel, Kang, James, Leister, Lara, Graybill, Todd L, Charnley, Adam K, Ye, Guosen, Nevins, Neysa, Behnia, Kamelia, Wolf, Amaya I, Kasparcova, Viera, Nurse, Kelvin, Wang, Liping, Puhl, Ana C, Li, Yue, Klein, Michael, Hopson, Christopher B, Guss, Jeffrey, Bantscheff, Marcus, Bergamini, Giovanna, Reilly, Michael A, Lian, Yiqian, Duffy, Kevin J, Adams, Jerry, Foley, Kevin P, Gough, Peter J, Marquis, Robert W, Smothers, James, Hoos, Axel, Bertin, John
Published in Nature (London) (01.12.2018)
Published in Nature (London) (01.12.2018)
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Journal Article
A diamidobenzimidazole STING agonist protects against SARS-CoV-2 infection
Sze-Ling, Ng, Maehr, Rene, Morales, Angel, Ramanjulu, Joshi M
Published in Science Immunology (18.05.2021)
Published in Science Immunology (18.05.2021)
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Journal Article
Web Resource
STING Agonist Induced Innate Immune Responses Drive Anti-Respiratory Virus Activity In Vitro with Limited Antiviral Efficacy In Vivo
Broeckel, Rebecca, Browne, Amanda, Sucoloski, Scott, Cantizani, Juan, Simpson, Juliet. K., Pesiridis, Scott, Ramanjulu, Joshi M., Stokes, Neil, Luthra, Priya
Published in ACS infectious diseases (13.09.2024)
Published in ACS infectious diseases (13.09.2024)
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Journal Article
Overcoming the Pregnane X Receptor Liability: Rational Design to Eliminate PXR-Mediated CYP Induction
Ramanjulu, Joshi M, Williams, Shawn P, Lakdawala, Ami S, DeMartino, Michael P, Lan, Yunfeng, Marquis, Robert W
Published in ACS medicinal chemistry letters (09.09.2021)
Published in ACS medicinal chemistry letters (09.09.2021)
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Journal Article
Titanium(IV) Isopropoxide Mediated Synthesis of Pyrimidin-4-ones
Ramanjulu, Joshi M, DeMartino, Michael P, Lan, Yunfeng, Marquis, Robert
Published in Organic letters (21.05.2010)
Published in Organic letters (21.05.2010)
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Journal Article
Author Correction: Design of amidobenzimidazole STING receptor agonists with systemic activity
Ramanjulu, Joshi M, Pesiridis, G Scott, Yang, Jingsong, Concha, Nestor, Singhaus, Robert, Zhang, Shu-Yun, Tran, Jean-Luc, Moore, Patrick, Lehmann, Stephanie, Eberl, H Christian, Muelbaier, Marcel, Schneck, Jessica L, Clemens, Jim, Adam, Michael, Mehlmann, John, Romano, Joseph, Morales, Angel, Kang, James, Leister, Lara, Graybill, Todd L, Charnley, Adam K, Ye, Guosen, Nevins, Neysa, Behnia, Kamelia, Wolf, Amaya I, Kasparcova, Viera, Nurse, Kelvin, Wang, Liping, Puhl, Ana C, Li, Yue, Klein, Michael, Hopson, Christopher B, Guss, Jeffrey, Bantscheff, Marcus, Bergamini, Giovanna, Reilly, Michael A, Lian, Yiqian, Duffy, Kevin J, Adams, Jerry, Foley, Kevin P, Gough, Peter J, Marquis, Robert W, Smothers, James, Hoos, Axel, Bertin, John
Published in Nature (London) (01.06.2019)
Published in Nature (London) (01.06.2019)
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Journal Article
Total Synthesis of Vancomycin-Part 1: Design and Development of Methodology
Nicolaou, K. C., Li, Hui, Boddy, Christopher N. C., Ramanjulu, Joshi M., Yue, Tai-Yuen, Natarajan, Swaminathan, Chu, Xin-Jie, Bräse, Stefan, Rübsam, Frank
Published in Chemistry : a European journal (03.09.1999)
Published in Chemistry : a European journal (03.09.1999)
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Journal Article
Total Synthesis of Vancomycin Aglycon-Part 1: Synthesis of Amino Acids 4-7 and Construction of the AB-COD Ring Skeleton
Nicolaou, K. C., Natarajan, Swaminathan, Li, Hui, Jain, Nareshkumar F., Hughes, Robert, Solomon, Michael E., Ramanjulu, Joshi M., Boddy, Christopher N. C., Takayanagi, Masaru
Published in Angewandte Chemie (International ed.) (16.10.1998)
Published in Angewandte Chemie (International ed.) (16.10.1998)
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Journal Article
Total Synthesis of Vancomycin-Part 2: Retrosynthetic Analysis, Synthesis of Amino Acid Building Blocks and Strategy Evaluations
Nicolaou, K. C., Boddy, Christopher N. C., Li, Hui, Koumbis, Alexandros E., Hughes, Robert, Natarajan, Swaminathan, Jain, Nareshkumar F., Ramanjulu, Joshi M., Bräse, Stefan, Solomon, Michael E.
Published in Chemistry : a European journal (03.09.1999)
Published in Chemistry : a European journal (03.09.1999)
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Journal Article
Total Synthesis of Vancomycin Aglycon-Part 2: Synthesis of Amino Acids 1-3 and Construction of the AB-COD-DOE Ring Skeleton
Nicolaou, K. C., Jain, Nareshkumar F., Natarajan, Swaminathan, Hughes, Robert, Solomon, Michael E., Li, Hui, Ramanjulu, Joshi M., Takayanagi, Masaru, Koumbis, Alexandros E., Bando, Toshikazu
Published in Angewandte Chemie (International ed.) (16.10.1998)
Published in Angewandte Chemie (International ed.) (16.10.1998)
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Journal Article
HETEROCYCLIC AMIDE USEFUL AS PROTEIN REGULATOR
LI YUE, JOSHI M RAMANJULU, YE GUOSEN, KANG JIANXING, TERRY V HUGHES, LARA KATHRYN LEISTER, ADAM KENNETH CHARNLEY, JOSEPH J ROMANO, GREN Z WANG, DONG XIAOYANG, JASON W DODSON, ZHANG DAOHUA, JOHN F MEHLMANN, NEYSA NEVINS, MICHAEL G DARCY, LIAN YIQIAN
Year of Publication 26.07.2021
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Year of Publication 26.07.2021
Patent
HETEROCYCLIC AMIDES USEFUL AS PROTEIN MODULATORS
LI YUE, JOSHI M RAMANJULU, YE GUOSEN, KANG JIANXING, TERRY V HUGHES, LARA KATHRYN LEISTER, ADAM KENNETH CHARNLEY, JOSEPH J ROMANO, GREN Z WANG, DONG XIAOYANG, JASON W DODSON, ZHANG DAOHUA, JOHN F MEHLMANN, NEYSA NEVINS, MICHAEL G DARCY, LIAN YIQIAN
Year of Publication 02.07.2020
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Year of Publication 02.07.2020
Patent
Inhibition of Protein Synthesis by Didemnins: Cell Potency and SAR
Ahuja, Deepika, Geiger, Adam, Ramanjulu, Joshi M, Vera, Matthew D, SirDeshpande, Bhagyashri, Pfizenmayer, Amy, Abazeed, Mohamed, Krosky, Daniel J, Beidler, David, Joullié, Madeleine M, Toogood, Peter L
Published in Journal of medicinal chemistry (02.11.2000)
Published in Journal of medicinal chemistry (02.11.2000)
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Journal Article
HETEROCYCLIC AMIDES AS KINASE INHIBITORS
JOSHI M RAMANJULU, ROBERT W MARQUIS JR, KANG JIANXING, LARA KATHRYN LEISTER, BRYAN WAYNE KING, JAE U JEONG, RAHMAN ATTIQ, ROBERT SINGHAUS JR, LAKDAWALA SHAH AMI, CLARK A SEHON, ZHANG DAOHUA, PHILIP ANTHONY HARRIS, DEEPAK BANDYOPADHYAY, PATRICK M EIDAM, PETER J GOUGH
Year of Publication 27.09.2018
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Year of Publication 27.09.2018
Patent
HETEROCYCLIC AMIDES AS KINASE INHIBITORS
JOSHI M RAMANJULU, ROBERT W MARQUIS JR, KANG JIANXING, LARA KATHRYN LEISTER, BRYAN WAYNE KING, JAE U JEONG, RAHMAN ATTIQ, ROBERT SINGHAUS JR, LAKDAWALA SHAH AMI, CLARK A SEHON, ZHANG DAOHUA, PHILIP ANTHONY HARRIS, DEEPAK BANDYOPADHYAY, PATRICK M EIDAM, PETER J GOUGH
Year of Publication 19.07.2018
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Year of Publication 19.07.2018
Patent
Synthesis of a Reduced Ring Analog of Didemnin B
Ramanjulu, Joshi M, Ding, Xiaobin, Joullié, Madeleine M, Li, Wen-Ren
Published in Journal of organic chemistry (25.07.1997)
Published in Journal of organic chemistry (25.07.1997)
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Journal Article
Total synthesis of vancomycin - Part 1: Design and development of methodology
Nicolaou, KC, Li, H, Boddy, CNC, Ramanjulu, JM, Yue, TY, Natarajan, S, Chu, XJ, Brase, S, Rubsam, F
Published in Chemistry : a European journal (01.09.1999)
Published in Chemistry : a European journal (01.09.1999)
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Journal Article