1,2-Benzothiazine 1,1-Dioxide P2−P3 Peptide Mimetic Aldehyde Calpain I Inhibitors
Wells, Gregory J, Tao, Ming, Josef, Kurt A, Bihovsky, Ron
Published in Journal of medicinal chemistry (11.10.2001)
Published in Journal of medicinal chemistry (11.10.2001)
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Synthesis of constrained benzocinnolinone analogues of CEP-26401 (irdabisant) as potent, selective histamine H3 receptor inverse agonists
Josef, Kurt A., Aimone, Lisa D., Lyons, Jacquelyn, Raddatz, Rita, Hudkins, Robert L.
Published in Bioorganic & medicinal chemistry letters (15.06.2012)
Published in Bioorganic & medicinal chemistry letters (15.06.2012)
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4-Phenoxypiperidine pyridazin-3-one histamine H3 receptor inverse agonists demonstrating potent and robust wake promoting activity
Hudkins, Robert L., Zulli, Allison L., Dandu, Reddeppa reddy, Tao, Ming, Josef, Kurt A., Aimone, Lisa D., Curtis Haltiwanger, R., Huang, Zeqi, Lyons, Jacquelyn A., Mathiasen, Joanne R., Raddatz, Rita, Gruner, John A.
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
Published in Bioorganic & medicinal chemistry letters (15.02.2012)
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Mixed-Lineage Kinase 1 and Mixed-Lineage Kinase 3 Subtype-Selective Dihydronaphthyl[3,4-a]pyrrolo[3,4-c]carbazole-5-ones: Optimization, Mixed-Lineage Kinase 1 Crystallography, and Oral in Vivo Activity in 1-Methyl-4-phenyltetrahydropyridine Models
Hudkins, Robert L, Diebold, James L, Tao, Ming, Josef, Kurt A, Park, Chung Ho, Angeles, Thelma S, Aimone, Lisa D, Husten, Jean, Ator, Mark A, Meyer, Sheryl L, Holskin, Beverly P, Durkin, John T, Fedorov, Alexander A, Fedorov, Elena V, Almo, Steven C, Mathiasen, Joanne R, Bozyczko-Coyne, Donna, Saporito, Michael S, Scott, Richard W, Mallamo, John P
Published in Journal of medicinal chemistry (25.09.2008)
Published in Journal of medicinal chemistry (25.09.2008)
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4,5-Dihydropyridazin-3-one derivatives as histamine H3 receptor inverse agonists
Hudkins, Robert L., Aimone, Lisa D., Dandu, Reddeppa reddy, Dunn, Derek, Gruner, John A., Huang, Zeqi, Josef, Kurt A., Lyons, Jacquelyn A., Mathiasen, Joanne R., Tao, Ming, Zulli, Allison L., Raddatz, Rita
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
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Journal Article
Identification of pyridazin-3-one derivatives as potent, selective histamine H3 receptor inverse agonists with robust wake activity
Hudkins, Robert L., Aimone, Lisa D., Bailey, Thomas R., Bendesky, Robert J., Dandu, Reddeppa reddy, Dunn, Derek, Gruner, John A., Josef, Kurt A., Lin, Yin-Guo, Lyons, Jacquelyn, Marcy, Val R., Mathiasen, Joanne R., Sundar, Babu G., Tao, Ming, Zulli, Allison L., Raddatz, Rita, Bacon, Edward R.
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
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Discovery of (1R, 6S)-5-[4-(1-cyclobutyl-piperidin-4-yloxy)-phenyl]3,4-diaza-bicyclo[4.1.0] hept-4-en-2-one (R, S-4a): Histamine H3 receptor inverse agonist demonstrating potent cognitive enhancing and wake promoting activity
Hudkins, Robert L., Josef, Kurt A., Becknell, Nadine C., Aimone, Lisa D., Lyons, Jacquelyn A., Mathiasen, Joanne R., Gruner, John A., Raddatz, Rita
Published in Bioorganic & medicinal chemistry letters (01.03.2014)
Published in Bioorganic & medicinal chemistry letters (01.03.2014)
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Peptide Aptamer Microarrays: Bridging the bio-detector interface
Song, Qifeng, Josef Stadler, Lukas Kurt, Peng, Jianhe, Ko Ferrigno, Paul
Published in Faraday discussions (01.01.2011)
Published in Faraday discussions (01.01.2011)
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Conformationally restrained analogs of pravadoline: nanomolar potent, enantioselective, (aminoalkyl)indole agonists of the cannabinoid receptor
D'Ambra, Thomas E, Estep, Kimberly G, Bell, Malcolm R, Eissenstat, Michael A, Josef, Kurt A, Ward, Susan J, Haycock, Dean A, Baizman, Eugene R, Casiano, Frances M
Published in Journal of medicinal chemistry (01.01.1992)
Published in Journal of medicinal chemistry (01.01.1992)
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Potent peptide α-Ketohydroxamate inhibitors of recombinant human calpain I
Josef, Kurt A, Kauer, Frederick W, Bihovsky, Ron
Published in Bioorganic & medicinal chemistry letters (08.10.2001)
Published in Bioorganic & medicinal chemistry letters (08.10.2001)
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Does political and social feasibility matter in energy scenarios?
Schubert, Daniel Kurt Josef, Thuß, Sebastian, Möst, Dominik
Published in Energy research & social science (01.05.2015)
Published in Energy research & social science (01.05.2015)
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1,3,5-Trialkyl-2,4,6-triiodobenzenes: Novel X-ray Contrast Agents for Gastrointestinal Imaging
Estep, Kimberly G, Josef, Kurt A, Bacon, Edward R, Illig, Carl R, Toner, John L, Mishra, Dinesh, Blazak, William F, Miller, Dennis M, Johnson, David K, Allen, Jack M, Spencer, Andy, Wilson, Susan A
Published in Journal of medicinal chemistry (18.05.2000)
Published in Journal of medicinal chemistry (18.05.2000)
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Synthesis and Structure-Activity Relationships of 6-Heterocyclic-Substituted Purines as Inactivation Modifiers of Cardiac Sodium Channels
Estep, Kimberly G, Josef, Kurt A, Bacon, Edward R, Carabateas, Philip M, Rumney, Squire, Pilling, Garry M, Krafte, Douglas S, Volberg, Walter A, Dillon, Kathleen, Dugrenier, Nancy, Briggs, G. Maurice, Canniff, Paul C, Gorczyca, William P, Stankus, Gerald P, Ezrin, Alan M
Published in Journal of medicinal chemistry (01.07.1995)
Published in Journal of medicinal chemistry (01.07.1995)
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Discovery of (1R,6S)-5-[4-(1-cyclobutyl-piperidin-4-yloxy)-phenyl]-3,4-diaza-bi c yclo[4.1.0]hept-4-en-2-one (R,S-4a): Histamine H3 receptor inverse agonist demonstrating potent cognitive enhancing and wake promoting activity
Hudkins, Robert, Josef, Kurt, Becknell, Nadine, Aimone, Lisa, Lyons, Jacquelyn, Mathiasen, Joanne, Gruner, John, Raddatz, Rita
Published in Bioorganic & medicinal chemistry letters (01.03.2014)
Published in Bioorganic & medicinal chemistry letters (01.03.2014)
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Structure−function studies of an engineered scaffold protein derived from Stefin A. II: Development and applications of the SQT variant
Stadler, Lukas Kurt Josef, Hoffmann, Toni, Tomlinson, Darren Charles, Song, Qifeng, Lee, Tracy, Busby, Michael, Nyathi, Yvonne, Gendra, Elisenda, Tiede, Christian, Flanagan, Keith, Cockell, Simon J., Wipat, Anil, Harwood, Colin, Wagner, Simon D., Knowles, Margaret A., Davis, Jason J., Keegan, Neil, Ko Ferrigno, Paul
Published in Protein engineering, design and selection (01.09.2011)
Published in Protein engineering, design and selection (01.09.2011)
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