Crystallographic Evidence for Preformed Dimers of Erythropoietin Receptor Before Ligand Activation
Livnah, Oded, Stura, Enrico A., Middleton, Steven A., Johnson, Dana L., Jolliffe, Linda K., Wilson, Ian A.
Published in Science (American Association for the Advancement of Science) (12.02.1999)
Published in Science (American Association for the Advancement of Science) (12.02.1999)
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Functional Mimicry of a Protein Hormone by a Peptide Agonist: The EPO Receptor Complex at 2.8 Å
Livnah, Oded, Stura, Enrico A., Johnson, Dana L., Middleton, Steven A., Mulcahy, Linda S., Wrighton, Nicholas C., Dower, William J., Jolliffe, Linda K., Wilson, Ian A.
Published in Science (American Association for the Advancement of Science) (26.07.1996)
Published in Science (American Association for the Advancement of Science) (26.07.1996)
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Small Peptides as Potent Mimetics of the Protein Hormone Erythropoietin
Wrighton, Nicholas C., Farrell, Francis X., Chang, Ray, Kashyap, Arun K., Barbone, Francis P., Mulcahy, Linda S., Johnson, Dana L., Barrett, Ronald W., Jolliffe, Linda K., Dower, William J.
Published in Science (American Association for the Advancement of Science) (26.07.1996)
Published in Science (American Association for the Advancement of Science) (26.07.1996)
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Increased potency of an erythropoietin peptide mimetic through covalent dimerization
Wrighton, Nicholas C, Balasubramanian, Palaniappan, Barbone, Francis P, Kashyap, Arun K, Farrell, Francis X, Jolliffe, Linda K, Barrett, Ronald W, Dower, William J
Published in Nature biotechnology (01.11.1997)
Published in Nature biotechnology (01.11.1997)
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Identification of a 13 Amino Acid Peptide Mimetic of Erythropoietin and Description of Amino Acids Critical for the Mimetic Activity of EMP1
Johnson, Dana L, Farrell, Francis X, Barbone, Francis P, McMahon, Frank J, Tullai, Jennifer, Hoey, Kenway, Livnah, Oded, Wrighton, Nicholas C, Middleton, Steven A, Loughney, Deborah A, Stura, Enrico A, Dower, William J, Mulcahy, Linda S, Wilson, Ian A, Jolliffe, Linda K
Published in Biochemistry (Easton) (17.03.1998)
Published in Biochemistry (Easton) (17.03.1998)
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1-Acyl-1H-[1,2,4]triazole-3,5-diamine Analogues as Novel and Potent Anticancer Cyclin-Dependent Kinase Inhibitors: Synthesis and Evaluation of Biological Activities
Lin, Ronghui, Connolly, Peter J, Huang, Shenlin, Wetter, Steven K, Lu, Yanhua, Murray, William V, Emanuel, Stuart L, Gruninger, Robert H, Fuentes-Pesquera, Angel R, Rugg, Catherine A, Middleton, Steven A, Jolliffe, Linda K
Published in Journal of medicinal chemistry (30.06.2005)
Published in Journal of medicinal chemistry (30.06.2005)
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In Vitro Characterization of Five Humanized OKT3 Effector Function Variant Antibodies
Xu, Danlin, Alegre, Maria-Luisa, Varga, Sally S., Rothermel, Annette L., Collins, Alexander M., Pulito, Virginia L., Hanna, Lewis S., Dolan, Kevin P., Parren, Paul W.H.I., Bluestone, Jeffrey A., Jolliffe, Linda K., Zivin, Robert A.
Published in Cellular immunology (25.02.2000)
Published in Cellular immunology (25.02.2000)
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The structure, organization, activation and plasticity of the erythropoietin receptor
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Book Review
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3-Acyl-2,6-diaminopyridines as cyclin-dependent kinase inhibitors: synthesis and biological evaluation
Lin, Ronghui, Lu, Yanhua, Wetter, Steven K., Connolly, Peter J., Turchi, Ignatius J., Murray, William V., Emanuel, Stuart L., Gruninger, Robert H., Fuentes-Pesquera, Angel R., Adams, Mary, Pandey, Niranjan, Moreno-Mazza, Sandra, Middleton, Steven A., Jolliffe, Linda K.
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
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Arylpiperazine substituted heterocycles as Selective α1a adrenergic antagonists
Khatuya, Haripada, Hutchings, Richard H, Kuo, Gee-Hong, Pulito, Virginia L, Jolliffe, Linda K, Li, Xiaobing, Murray, William V
Published in Bioorganic & medicinal chemistry letters (02.09.2002)
Published in Bioorganic & medicinal chemistry letters (02.09.2002)
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Journal Article
An antagonist peptide-EPO receptor complex suggests that receptor dimerization is not sufficient for activation
Jolliffe, Linda K, Wilson, Ian A, Livnah, Oded, Johnson, Dana L, Stura, Enrico A, Farrell, Francis X, Barbone, Francis P, You, Yun, Liu, Kathleen D, Goldsmith, Mark A, He, Wen, Krause, Christopher D, Pestka, Sidney
Published in Nature structural biology (01.11.1998)
Published in Nature structural biology (01.11.1998)
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Journal Article
Shared and Unique Determinants of the Erythropoietin (EPO) Receptor Are Important for Binding EPO and EPO Mimetic Peptide
Middleton, Steven A., Barbone, Francis P., Johnson, Dana L., Thurmond, Robin L., You, Yun, McMahon, Frank J., Jin, Renzhe, Livnah, Oded, Tullai, Jennifer, Farrell, Francis X., Goldsmith, Mark A., Wilson, Ian A., Jolliffe, Linda K.
Published in The Journal of biological chemistry (14.05.1999)
Published in The Journal of biological chemistry (14.05.1999)
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Erythropoietin induces changes in gene expression in PC-12 cells
Renzi, Michael J, Farrell, Francis X, Bittner, Anton, Galindo, Jose E, Morton, Mike, Trinh, Heather, Jolliffe, Linda K
Published in Brain research. Molecular brain research. (15.07.2002)
Published in Brain research. Molecular brain research. (15.07.2002)
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Synthesis and erythropoietin receptor binding affinities of N,N-disubstituted amino acids
Connolly, Peter J, Wetter, Steven K, Murray, William V, Johnson, Dana L, McMahon, Frank J, Farrell, Francis X, Tullai, Jennifer, Jolliffe, Linda K
Published in Bioorganic & medicinal chemistry letters (04.09.2000)
Published in Bioorganic & medicinal chemistry letters (04.09.2000)
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Mutagenesis Studies of the Human Erythropoietin Receptor
Barbone, Francis P., Middleton, Steven A., Johnson, Dana L., McMahon, Frank J., Tullai, Jennifer, Gruninger, Robert H., Schilling, Adriane E., Jolliffe, Linda K., Mulcahy, Linda S.
Published in The Journal of biological chemistry (21.02.1997)
Published in The Journal of biological chemistry (21.02.1997)
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Journal Article
Identification of a Critical Ligand Binding Determinant of the Human Erythropoietin Receptor
Middleton, Steven A., Johnson, Dana L., Jin, Renzhe, McMahon, Frank J., Collins, Alexander, Tullai, Jennifer, Gruninger, Robert H., Jolliffe, Linda K., Mulcahy, Linda S.
Published in The Journal of biological chemistry (14.06.1996)
Published in The Journal of biological chemistry (14.06.1996)
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Journal Article
Amino-terminal dimerization of an erythropoietin mimetic peptide results in increased erythropoietic activity
Johnson, Dana L., Farrell, Francis X., Barbone, Francis P., McMahon, Frank J., Tullai, Jennifer, Kroon, Daniel, Freedy, James, Zivin, Robert A., Mulcahy, Linda S., Jolliffe, Linda K.
Published in Chemistry & biology (01.12.1997)
Published in Chemistry & biology (01.12.1997)
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Erythropoietin mimetic peptides and the future
Johnson, Dana L., Jolliffe, Linda K.
Published in Nephrology, dialysis, transplantation (01.09.2000)
Published in Nephrology, dialysis, transplantation (01.09.2000)
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Journal Article
1-Acyl-1 H -[1,2,4]triazole-3,5-diamine Analogues as Novel and Potent Anticancer Cyclin-Dependent Kinase Inhibitors: Synthesis and Evaluation of Biological Activities
Lin, Ronghui, Connolly, Peter J., Huang, Shenlin, Wetter, Steven K., Lu, Yanhua, Murray, William V., Emanuel, Stuart L., Gruninger, Robert H., Fuentes-Pesquera, Angel R., Rugg, Catherine A., Middleton, Steven A., Jolliffe, Linda K.
Published in Journal of medicinal chemistry (01.06.2005)
Published in Journal of medicinal chemistry (01.06.2005)
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