Allosteric chromenone inhibitors of phosphoinositide 3-kinase (PI3K) for the treatment of disease
Dahlgren, Markus K, Knight, Jennifer Lynn, Kesicki, Edward A, Klippel-Giese, Anke, Mayne, Christopher Glenn, McElligott, David L, Long, Katelyn Frances, Aronow, Sean Douglas, Ravi, Kannan Karukurichi, Feng, Shulu, Widjaja, Tien, Hickey, Eugene R, Kolakowski, Gabrielle R, Severance, Daniel Lee, Irvin, Thomas Combs, Puca, Loredana, Anderson, Erin Danielle, Boyles, Nicholas A, Gerasyuto, Aleksey I, Kumar, Manoj, Welch, Michael Brian, McLean, Johnathan Alexander
Year of Publication 16.05.2023
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Year of Publication 16.05.2023
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THIENO[2,3-C]PYRROL-4-ON-DERIVATER SOM ERK-INHIBITORER
MCMILLEN, William T, CORTEZ, Guillermo S, JOSEPH, Sajan, MCLEAN, Johnathan Alexander, RODRIGUEZ, Michael John, ZHAO, Gaiying
Year of Publication 22.07.2019
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Year of Publication 22.07.2019
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ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR THE TREATMENT OF DISEASE
DAWADI, Surendra, ANDERSON, Erin Danielle, HICKEY, Eugene R, CHEN, Xiaohong, POTOTSCHNIG, Gerit Maria, KOLAKOWSKI, Gabrielle R, MCLEAN, Johnathan Alexander, WIDJAJA, Tien, IRVIN, Thomas Combs, WELCH, Michael Brian, LONG, Katelyn Frances, ARONOW, Sean Douglas, KNIGHT, Jennifer Lynn, WANG, Hua-Yu, BOYLES, Nicholas A, KUMAR, Manoj, MAYNE, Christopher Glenn, KESICKI, Edward A
Year of Publication 30.03.2023
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Year of Publication 30.03.2023
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THIENO[2,3-C]PYRROL-4-ONE DERIVATIVES AS ERK INHIBITORS
RODRIGUEZ, MICHAEL JOHN, CORTEZ, GUILLERMO S, JOSEPH, SAJAN, ZHAO, GAIYING, MCMILLEN, WILLIAM T, MCLEAN, JOHNATHAN ALEXANDER
Year of Publication 18.06.2019
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Year of Publication 18.06.2019
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THIENO[2,3-C]PYRROL-4-ONE DERIVATIVES AS ERK INHIBITORS
MCMILLEN, William T, CORTEZ, Guillermo S, JOSEPH, Sajan, MCLEAN, Johnathan Alexander, RODRIGUEZ, Michael John, ZHAO, Gaiying
Year of Publication 05.06.2019
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Year of Publication 05.06.2019
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ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR THE TREATMENT OF DISEASES ASSOCIATED WITH P13K MODULATION
ANDERSON, Erin Danielle, GERASYUTO, Aleksey I, HICKEY, Eugene R, FENG, Shulu, KOLAKOWSKI, Gabrielle R, MCLEAN, Johnathan Alexander, SEVERANCE, Daniel Lee, WIDJAJA, Tien, MCELLIGOTT, David L, IRVIN, Thomas Combs, PUCA, Loredana, RAVI, Kannan Karukurichi, WELCH, Michael Brian, LONG, Katelyn Frances, ARONOW, Sean Douglas, KNIGHT, Jennifer Lynn, BOYLES, Nicholas A, KUMAR, Manoj, KLIPPEL-GIESE, Anke, MAYNE, Christopher Glenn, DAHLGREN, Markus K, KESICKI, Edward A
Year of Publication 08.02.2023
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Year of Publication 08.02.2023
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THIENO[2,3-C]PYRROL-4-ONE DERIVATIVES AS ERK INHIBITORS
MCMILLEN, William T, CORTEZ, Guillermo S, JOSEPH, Sajan, MCLEAN, Johnathan Alexander, RODRIGUEZ, Michael John, ZHAO, Gaiying
Year of Publication 27.02.2019
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Year of Publication 27.02.2019
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ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR THE TREATMENT OF CANCER
HICKEY, EUGENE R, ANDERSON, ERIN DANIELLE, ARONOW, SEAN DOUGLAS, BOYLES, NICHOLAS A, IRVIN, THOMAS COMBS, LONG, KATELYN FRANCES, WELCH, MICHAEL BRIAN, CHEN, XIAOHONG, KNIGHT, JENNIFER LYNN, MAYNE, CHRISTOPHER GLENN, DAWADI, SURENDRA, POTOTSCHNIG, GERIT MARIA, MCLEAN, JOHNATHAN ALEXANDER, KESICKI, EDWARD A, WIDJAJA, TIEN, KOLAKOWSKI, GABRIELLE R, KUMAR, MANOJ, WANG, HUA-YU
Year of Publication 01.12.2022
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Year of Publication 01.12.2022
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ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR THE TREATMENT OF CANCER
DAWADI, Surendra, ANDERSON, Erin Danielle, HICKEY, Eugene R, CHEN, Xiaohong, POTOTSCHNIG, Gerit Maria, KOLAKOWSKI, Gabrielle R, MCLEAN, Johnathan Alexander, WIDJAJA, Tien, IRVIN, Thomas Combs, WELCH, Michael Brian, LONG, Katelyn Frances, ARONOW, Sean Douglas, KNIGHT, Jennifer Lynn, WANG, Hua-Yu, BOYLES, Nicholas A, KUMAR, Manoj, MAYNE, Christopher Glenn, KESICKI, Edward A
Year of Publication 01.12.2022
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Year of Publication 01.12.2022
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Thieno[2,3-c]pyrrol-4-one derivatives as ERK inhibitors
Zhao, Gaiying, Joseph, Sajan, Rodriguez, Michael John, McMillen, William T, Cortez, Guillermo S, McLean, Johnathan Alexander
Year of Publication 21.02.2019
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Year of Publication 21.02.2019
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ALLOSTERIC CHROMENONE INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE (PI3K) FOR THE TREATMENT OF DISEASE
ANDERSON, Erin Danielle, GERASYUTO, Aleksey I, HICKEY, Eugene R, FENG, Shulu, KOLAKOWSKI, Gabrielle R, MCLEAN, Johnathan Alexander, SEVERANCE, Daniel Lee, WIDJAJA, Tien, MCELLIGOTT, David L, IRVIN, Thomas Combs, PUCA, Loredana, RAVI, Kannan Karukurichi, WELCH, Michael Brian, LONG, Katelyn Frances, ARONOW, Sean Douglas, KNIGHT, Jennifer Lynn, BOYLES, Nicholas A, KUMAR, Manoj, KLIPPEL-GIESE, Anke, MAYNE, Christopher Glenn, DAHLGREN, Markus K, KESICKI, Edward A
Year of Publication 24.11.2022
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Year of Publication 24.11.2022
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Allosteric chromenone inhibitors of phosphoinositide 3-kinase (PI3K) for the treatment of diseases associated with PI3K modulation
ANDERSON, Erin Danielle, GERASYUTO, Aleksey I, HICKEY, Eugene R, FENG, Shulu, KOLAKOWSKI, Gabrielle R, MCLEAN, Johnathan Alexander, SEVERANCE, Daniel Lee, WIDJAJA, Tien, MCELLIGOTT, David L, IRVIN, Thomas Combs, PUCA, Loredana, RAVI, Kannan Karukurichi, WELCH, Michael Brian, LONG, Katelyn Frances, ARONOW, Sean Douglas, KNIGHT, Jennifer Lynn, BOYLES, Nicholas A, KUMAR, Manoj, KLIPPEL-GIESE, Anke, MAYNE, Christopher Glenn, DAHLGREN, Markus K, KESICKI, Edward A
Year of Publication 20.10.2022
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Year of Publication 20.10.2022
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Thieno[2,3-c]pyrrol-4-one derivatives as erk inhibitors
Zhao, Gaiying, Joseph, Sajan, Mcmillen, William T, Rodriguez, Michael John, Mclean, Johnathan Alexander, Cortez, Guillermo S
Year of Publication 21.12.2018
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Year of Publication 21.12.2018
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THIENO[2,3-C]PYRROL-4-ONE DERIVATIVES AS ERK INHIBITORS
MCMILLEN, William T, CORTEZ, Guillermo S, JOSEPH, Sajan, MCLEAN, Johnathan Alexander, RODRIGUEZ, Michael John, ZHAO, Gaiying
Year of Publication 19.10.2018
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Year of Publication 19.10.2018
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ERK INHIBITORS
MCMILLEN, William T, CORTEZ, Guillermo S, JOSEPH, Sajan, MCLEAN, Johnathan Alexander, RODRIGUEZ, Michael John, ZHAO, Gaiying
Year of Publication 26.09.2018
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Year of Publication 26.09.2018
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DERIVADOS DE TIENO[2,3-C]PIRROL-4-ONA COMO INHIBIDORES DE ERK
JOSEPH SAJAN, ZHAO GAIYING, CORTEZ GUILLERMO S, MCLEAN JOHNATHAN ALEXANDER, RODRIGUEZ MICHAEL JOHN
Year of Publication 27.08.2018
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Year of Publication 27.08.2018
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Thieno[2,3-c]pyrrol-4-one derivatives as ERK inhibitors
Zhao, Gaiying, Joseph, Sajan, Rodriguez, Michael John, McMillen, William T, Cortez, Guillermo S, McLean, Johnathan Alexander
Year of Publication 23.08.2018
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Year of Publication 23.08.2018
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PYRAZOLE DERIVATIVES AS RET KINASE INHIBITORS
BOLDRON, CHRISTOPHER PIERRE ALBERT JEAN, MOURET, TIPHAINE, PANCALDI, THOMAS PIERRE DINO, ANDREWS, STEVEN W, MCKENNEY, MEGAN L, PILKINGTON-MIKSA, MICHAEL ALEXANDER, IRVIN, THOMAS C, ANDERSON, ERIN D, MCFADDIN, ELIZABETH A, MUNCHHOF, MICHAEL J, CONDROSKI, KEVIN R, PINTO, MARTA, MCLEAN, JOHNATHAN ALEXANDER, KUMAR, MANOJ, KOLAKOWSKI, GABRIELLE R. A/K/A JODY GABRIELLE RUSTMANN KOLAKOWSKI
Year of Publication 12.05.2022
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Year of Publication 12.05.2022
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RET KINASE INHIBITORS
ANDERSON, Erin D, BOLDON, Christopher Pierre Albert Jean, Andrews, Steven W, CONDROSKI, Kevin R, MCLEAN, Johnathan Alexander, Kolakowski, Gabrielle R, IRVIN, Thomas C, KUMAR, Manoj, PANCALDI, Thomas Pierre Dino, PILKINGTON-MIKSA, Michael Alexander, PINTO, Marta, MCKENNEY, Megan L, MUNCHHOF, Michael J, MOURET, Tiphaine, MCFADDIN, Elizabeth A
Year of Publication 12.05.2022
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Year of Publication 12.05.2022
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ERK inhibitors
Cortez Guillermo S, McLean Johnathan Alexander, Zhao Gaiying, Rodriguez Michael John, Joseph Sajan, McMillen William Thomas
Year of Publication 30.01.2018
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Year of Publication 30.01.2018
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