Cross-Strand Pairing and Amyloid Assembly
Liang, Yan, Pingali, Sai Venkatesh, Jogalekar, Ashutosh S, Snyder, James P, Thiyagarajan, Pappannan, Lynn, David G
Published in Biochemistry (Easton) (23.09.2008)
Published in Biochemistry (Easton) (23.09.2008)
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The Development of a Selective Cyclin-Dependent Kinase Inhibitor That Shows Antitumor Activity
ALI, Simak, HEATHCOTE, Dean A, TOLHURST, Robert S, KANNEGANTI, Seshu K, SNYDER, James P, LIOTTA, Dennis C, ABOAGYE, Eric O, BARRETT, Anthony G. M, COOMBES, R. Charles, KROLL, Sebastian H. B, JOGALEKAR, Ashutosh S, SCHEIPER, Bodo, PATEL, Hetal, BRACKOW, Jan, SIWICKA, Alekasandra, FUCHTER, Matthew J, PERIYASAMY, Manikandan
Published in Cancer research (Chicago, Ill.) (01.08.2009)
Published in Cancer research (Chicago, Ill.) (01.08.2009)
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A Novel Pyrazolo[1,5-a]pyrimidine Is a Potent Inhibitor of Cyclin-Dependent Protein Kinases 1, 2, and 9, Which Demonstrates Antitumor Effects in Human Tumor Xenografts Following Oral Administration
Heathcote, Dean A, Patel, Hetal, Kroll, Sebastian H. B, Hazel, Pascale, Periyasamy, Manikandan, Alikian, Mary, Kanneganti, Seshu K, Jogalekar, Ashutosh S, Scheiper, Bodo, Barbazanges, Marion, Blum, Andreas, Brackow, Jan, Siwicka, Alekasandra, Pace, Robert D. M, Fuchter, Matthew J, Snyder, James P, Liotta, Dennis C, Freemont, Paul. S, Aboagye, Eric O, Coombes, R. Charles, Barrett, Anthony G. M, Ali, Simak
Published in Journal of medicinal chemistry (23.12.2010)
Published in Journal of medicinal chemistry (23.12.2010)
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Journal Article
Dictyostatin Flexibility Bridges Conformations in Solution and in the β-Tubulin Taxane Binding Site
Jogalekar, Ashutosh S, Damodaran, Krishnan, Kriel, Frederik H, Jung, Won-Hyuk, Alcaraz, Ana A, Zhong, Shi, Curran, Dennis P, Snyder, James P
Published in Journal of the American Chemical Society (02.03.2011)
Published in Journal of the American Chemical Society (02.03.2011)
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Journal Article
The Discodermolide Hairpin Structure Flows from Conformationally Stable Modular Motifs
Jogalekar, Ashutosh S, Kriel, Frederik H, Shi, Qi, Cornett, Ben, Cicero, Daniel, Snyder, James P
Published in Journal of medicinal chemistry (14.01.2010)
Published in Journal of medicinal chemistry (14.01.2010)
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알로스테릭 SHP2 억제제로서의 다환식 화합물
WON WALTER S, BUCKL ANDREAS, TZITZILONIS CHRISTOS, PITZEN JENNIFER, BLANK BRIAN R, GILL ADRIAN LIAM, MELLEM KEVIN T, WANG GANG, KOLTUN ELENA S, CREGG JAMES JOSEPH, LI JIE JACK, AAY NAING N, JOGALEKAR ASHUTOSH S
Year of Publication 24.08.2020
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Year of Publication 24.08.2020
Patent
Abstract 4877: Allosteric inhibition of SHP2 variants containing cancer-associated activating mutations
Wildes, David, Aay, Naing, Buckl, Andreas, Hsieh, Daphne, Jogalekar, Ashutosh S., Kiss, Gert, Koltun, Elena S., Marquez, Abby, Mellem, Kevin T., Romero, Jason, Saldajeno-Concar, Mae, Schulze, Christopher J., Semko, Chris M., Won, Walter, Nichols, Robert J., Stahlhut, Carlos, Tzitzilonis, Christos, Gill, Adrian L., Smith, Jacqueline A.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract 4878: RMC-4550, an allosteric inhibitor of SHP2: Synthesis, structure, and anti-tumor activity
Koltun, Elena S., Aay, Naing, Buckl, Andreas, Jogalekar, Ashutosh S., Kiss, Gert, Marquez, Abby, Mellem, Kevin T., Mordec, Kasia, Saldajeno-Concar, Mae, Semko, Chris M., Tibrewal, Nidhi, Tzitzilonis, Christos, Won, Walter, Smith, Jacqueline A., Wilson, Susan E., Nichols, Robert J., Wang, Zhengping, Wilds, David, Singh, Mallika, Gill, Adrian L.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
The development of a selective cyclin-dependent kinase inhibitor which demonstrates anti-tumor activity
Ali, Simak, Heathcote, Dean A., Kroll, Sebastian H. B., Jogalekar, Ashutosh S., Scheiper, Bodo, Patel, Hetal, Brackow, Jan, Siwicka, Alekasandra, Fuchter, Matthew J., Periyasamy, Manikandan, Tolhurst, Robert S., Kanneganti, Seshu K., Snyder, James P., Liotta, Dennis C., Aboagye, Eric O., Barrett, Anthony G. M., Coombes, R. Charles
Published in Cancer research (Chicago, Ill.) (28.07.2009)
Published in Cancer research (Chicago, Ill.) (28.07.2009)
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Journal Article
POLYCYCLIC COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
WON, Walter S, LI, Jie Jack, AAY, Naing N, KOLTUN, Elena S, BLANK, Brian R, TZITZILONIS, Christos, PITZEN, Jennifer, BUCKL, Andreas, WANG, Gang, JOGALEKAR, Ashutosh S, MELLEM, Kevin T, GILL, Adrian Liam, CREGG, James Joseph
Year of Publication 28.03.2024
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Year of Publication 28.03.2024
Patent
POLYCYCLIC COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
WON, Walter S, LI, Jie Jack, AAY, Naing N, KOLTUN, Elena S, BLANK, Brian R, TZITZILONIS, Christos, PITZEN, Jennifer, BUCKL, Andreas, WANG, Gang, JOGALEKAR, Ashutosh S, MELLEM, Kevin T, GILL, Adrian Liam, CREGG, James Joseph
Year of Publication 04.10.2023
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Year of Publication 04.10.2023
Patent
Polycyclic compounds as allosteric SHP2 inhibitors
Koltun, Elena S, Tzitzilonis, Christos, Aay, Naing N, Won, Walter S, Li, Jie Jack, Pitzen, Jennifer, Blank, Brian R, Wang, Gang, Jogalekar, Ashutosh S, Gill, Adrian Liam, Mellem, Kevin T, Buckl, Andreas, Cregg, James Joseph
Year of Publication 13.06.2023
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Year of Publication 13.06.2023
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POLYCYCLIC COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
WON, Walter S, LI, Jie Jack, AAY, Naing N, KOLTUN, Elena S, BLANK, Brian R, TZITZILONIS, Christos, PITZEN, Jennifer, BUCKL, Andreas, WANG, Gang, JOGALEKAR, Ashutosh S, MELLEM, Kevin T, GILL, Adrian Liam, CREGG, James Joseph
Year of Publication 17.05.2021
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Year of Publication 17.05.2021
Patent
POLYCYCLIC COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
WON, Walter S, LI, Jie Jack, AAY, Naing N, KOLTUN, Elena S, BLANK, Brian R, TZITZILONIS, Christos, PITZEN, Jennifer, BUCKL, Andreas, WANG, Gang, JOGALEKAR, Ashutosh S, MELLEM, Kevin T, GILL, Adrian Liam, CREGG, James Joseph
Year of Publication 31.12.2020
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Year of Publication 31.12.2020
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