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The Substrate-Activity-Screening methodology applied to receptor tyrosine kinases: A proof-of-concept study
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Published in European journal of medicinal chemistry (01.11.2012)
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Published in Bioorganic & medicinal chemistry letters (01.02.2014)
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Liniger, Marc, Neuhaus, Christian, Hofmann, Tatjana, Fransioli-Ignazio, Luca, Jordi, Michel, Drueckes, Peter, Trappe, Jörg, Fabbro, Doriano, Altmann, Karl-Heinz
Published in ACS medicinal chemistry letters (13.01.2011)
Published in ACS medicinal chemistry letters (13.01.2011)
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Substrate profiling of IGF-1R and InsR: Identification of a potent pentamer substrate
Chapelat, Julien, Berst, Frédéric, Marzinzik, Andreas L., Moebitz, Henrik, Drueckes, Peter, Fabbro, Doriano, Trappe, Joerg, Seebach, Dieter
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
Published in Bioorganic & medicinal chemistry letters (01.12.2011)
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Targeting Plasmodium phosphatidylinositol 4-kinase to eliminate malaria
McNamara, Case W, Lee, Marcus CS, Lim, Chek Shik, Lim, Siau Hoi, Roland, Jason, Simon, Oliver, Yeung, Bryan KS, Chatterjee, Arnab K, McCormack, Susan L, Manary, Micah J, Zeeman, Anne-Marie, Dechering, Koen J, Kumar, TR Santha, Henrich, Philipp P, Gagaring, Kerstin, Ibanez, Maureen, Kato, Nobutaka, Kuhen, Kelli L, Fischli, Christoph, Nagle, Advait, Rottmann, Matthias, Plouffe, David M, Bursulaya, Badry, Meister, Stephan, Rameh, Lucia, Trappe, Joerg, Haasen, Dorothea, Timmerman, Martijn, Sauerwein, Robert W, Suwanarusk, Rossarin, Russell, Bruce, Renia, Laurent, Nosten, Francois, Tully, David C, Kocken, Clemens HM, Glynne, Richard J, Bodenreider, Christophe, Fidock, David A, Diagana, Thierry T, Winzeler, Elizabeth A
Published in Nature (London) (27.11.2013)
Published in Nature (London) (27.11.2013)
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