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Year of Publication 24.10.2012
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Year of Publication 24.10.2012
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α-Μethylation at benzylic fragment of N-aryl-N'-benzyl ureas provides TRPV1 antagonists with better pharmacokinetic properties and higher efficacy in inflammatory pain model
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Published in Bioorganic & medicinal chemistry letters (2007)
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PROCESS FOR PREPARING METHYL{(2S,3R)-1-[(2S)-2-{5-[(2R,5R)-1-{3,5-DIFLUORO-4-[4-(4-FLUOROPHENYL)PIPERIDINE-1-YL]PHENYL}-5-(6-FLUORO-2-{(2S)-1-[N-(METHOXYCARBONYL)-O-METHYL-L-THREONYL]PYRROLIDINE-2-YL}-1H-BENZIMIDAZOLE-5-YL)pyrrolidinePYRROLIDINE-2-YL]-6-FLUORO-1H-BENZIMIDAZOLE-2-YL}PYRROLIDINE-1-YL]-3-METHOXY-1-OXOBUTANE-2-YL}CARBAMATE
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Year of Publication 30.09.2019
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