Combination therapy with androgen receptor N‐terminal domain antagonist EPI‐7170 and enzalutamide yields synergistic activity in AR‐V7‐positive prostate cancer
Hirayama, Yukiyoshi, Tam, Teresa, Jian, Kunzhong, Andersen, Raymond J., Sadar, Marianne D.
Published in Molecular oncology (01.10.2020)
Published in Molecular oncology (01.10.2020)
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Lessons learned from the metastatic castration-resistant prostate cancer phase I trial of EPI-506, a first-generation androgen receptor N-terminal domain inhibitor
Le Moigne, Ronan, Zhou, Han-Jie, Obst, Jon K., Banuelos, C. Adriana, Jian, Kunzhong, Williams, David, Virsik, Peter, Andersen, Raymond J, Sadar, Marianne, Perabo, Frank, Chi, Kim N.
Published in Journal of clinical oncology (01.03.2019)
Published in Journal of clinical oncology (01.03.2019)
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Characterization of niphatenones that inhibit androgen receptor N-terminal domain
Banuelos, Carmen A, Lal, Aaron, Tien, Amy H, Shah, Neel, Yang, Yu Chi, Mawji, Nasrin R, Meimetis, Labros G, Park, Jacob, Kunzhong, Jian, Andersen, Raymond J, Sadar, Marianne D
Published in PloS one (2014)
Published in PloS one (2014)
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PD05-12 COMBINATION OF AN ANTAGONIST TO THE ANDROGEN RECEPTOR N-TERMINAL DOMAIN WITH ENZALUTAMIDE FOR THE TREATMENT OF CASTRATION RESISTANT PROSTATE CANCER
Hirayama, Yukiyoshi, Jian, Kunzhong, Anderson, Raymond J., Sadar, Marianne D.
Published in The Journal of urology (01.04.2019)
Published in The Journal of urology (01.04.2019)
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MP34-05 COMBINATION THERAPY FOR CASTRATION-RESISTANT PROSTATE CANCER USING ANTAGONISTS OF THE N-TERMINAL DOMAIN OF ANDROGEN RECEPTOR WITH IONIZING RADIATION
Ito, Yusuke, Banuelos, C. Adriana, Hirayama, Yukiyoshi, Jian, Kunzhong, Andersen, Raymond, Sadar, Marianne
Published in The Journal of urology (01.04.2019)
Published in The Journal of urology (01.04.2019)
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Journal Article
Combination therapy with androgen receptor N#8208;terminal domain antagonist EPI#8208;7170 and enzalutamide yields synergistic activity in AR#8208;V7#8208;positive prostate cancer
Hirayama, Yukiyoshi, Tam, Teresa, Jian, Kunzhong, Andersen, Raymond J, Sadar, Marianne D
Published in Molecular oncology (01.10.2020)
Published in Molecular oncology (01.10.2020)
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Synthetic Analogs of the Sponge Sesterterpenoid Alotaketal C are Potent Inhibitors of SARS-CoV‑2 Omicron BA.1 and BA.5 Infections of Human Lung Cells
Blagojevic, Polina, Perez-Vargas, Jimena, Jian, Kunzhong, Williams, David E., Villanueva, Ivan, Thompson, Connor A. H., Ennis, Siobhan, Niikura, Masahiro, Tietjen, Ian, Jean, François, Andersen, Raymond J.
Published in Organic letters (07.07.2023)
Published in Organic letters (07.07.2023)
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MP79-04 THE PRECLINICAL CHARACTERIZATION AND DEVELOPMENT OF EPI-7386, AN N-TERMINAL DOMAIN ANDROGEN RECEPTOR INHIBITOR, FOR THE TREATMENT OF PROSTATE CANCER
Moigne, Ronan Le, Banuelos, C. Adriana, Mawji, Nasrin R., Tam, Teresa, Wang, Jun, Jian, Kunzhong, Andersen, Raymond J., Cesano, Alessandra, Sadar, Marianne D., Zhou, Han-Jie, Virsik, Peter
Published in The Journal of urology (01.04.2020)
Published in The Journal of urology (01.04.2020)
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Journal Article
IND candidate EPI-7386 as an N-terminal domain androgen receptor inhibitor in development for the treatment of prostate cancer
Le Moigne, Ronan, Banuelos, C. Adriana, Mawji, Nasrin R., Tam, Teresa, Wang, Jun, Jian, Kunzhong, Andersen, Raymond J., Cesano, Alessandra, Sadar, Marianne, Zhou, Han-Jie, Virsik, Peter
Published in Journal of clinical oncology (20.02.2020)
Published in Journal of clinical oncology (20.02.2020)
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Abstract 1292: A new generation of N-terminal domain androgen receptor inhibitors, with improved pharmaceutical properties, in castration-resistant prostate cancer models
Moigne, Ronan Le, Mawji, Nasrin R., Banuelos, C. Adriana, Wang, Jun, Jian, Kunzhong, Andersen, Raymond J., Sadar, Marianne D., Zhou, Han-Jie, Virsik, Peter
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Abstract B117: Treatment of castrated resistant prostate cancer with EPI-7386, a second generation N-terminal domain androgen receptor inhibitor
Moigne, Ronan Le, Banuelos, C. Adriana, Mawji, Nasrin R, Tam, Teresa, Wang, Jun, Jian, Kunzhong, Andersen, Raymond J, Cesano, Alessandra, Sadar, Marianne D, Zhou, Han-Jie, Virsik, Peter
Published in Molecular cancer therapeutics (01.12.2019)
Published in Molecular cancer therapeutics (01.12.2019)
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Journal Article
MP34-04 A NEW GENERATION OF N-TERMINAL DOMAIN ANDROGEN RECEPTOR INHIBITORS IN CASTRATION-RESISTANT PROSTATE CANCER MODELS
Moigne, Ronan Le, Zhou, Han-Jie, Mawji, Nasrin R., Banuelos, C. Adriana, Wang, Jun, Jian, Kunzhong, Virsik, Peter, Andersen, Raymond J., Sadar, Marianne D.
Published in The Journal of urology (01.04.2019)
Published in The Journal of urology (01.04.2019)
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Journal Article
Next generation N-terminal domain androgen receptor inhibitors with improved potency and metabolic stability in castration-resistant prostate cancer models
Le Moigne, Ronan, Zhou, Han-Jie, Mawji, Nasrin R, Banuelos, C. Adriana, Wang, Jun, Jian, Kunzhong, Virsik, Peter, Andersen, Raymond J, Sadar, Marianne
Published in Journal of clinical oncology (01.03.2019)
Published in Journal of clinical oncology (01.03.2019)
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Revealing Metabolic Liabilities of Ralaniten To Enhance Novel Androgen Receptor Targeted Therapies
Obst, Jon K, Wang, Jun, Jian, Kunzhong, Williams, David E, Tien, Amy H, Mawji, Nasrin, Tam, Teresa, Yang, Yu Chi, Andersen, Raymond J, Chi, Kim N, Montgomery, Bruce, Sadar, Marianne D
Published in ACS pharmacology & translational science (13.12.2019)
Published in ACS pharmacology & translational science (13.12.2019)
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비스페놀 유도체 및 안드로겐 수용체 활성도 조절제로서의 이의 용도
MAWJI NASRIN R, JIAN KUNZHONG, WANG JUN, ANDERSEN RAYMOND, BANUELOS CARMEN ADRIANA, YANG YU CHI, SADAR MARIANNE DOROTHY
Year of Publication 01.02.2019
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Year of Publication 01.02.2019
Patent
An imaging agent to detect androgen receptor and its active splice variants in prostate cancer
Imamura, Yusuke, Tien, Amy H, Pan, Jinhe, Leung, Jacky K, Banuelos, Carmen A, Jian, Kunzhong, Wang, Jun, Mawji, Nasrin R, Fernandez, Javier Garcia, Lin, Kuo-Shyan, Andersen, Raymond J, Sadar, Marianne D
Published in JCI insight (21.07.2016)
Published in JCI insight (21.07.2016)
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