Search Results - "JEFFREY P. WHITTEN" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Anticancer Activity of CX-3543: A Direct Inhibitor of rRNA Biogenesis

Anticancer Activity of CX-3543: A Direct Inhibitor of rRNA Biogenesis

by DRYGIN, Denis, SIDDIQUI-JAIN, Adam, LIM, John K. C, VON HOFF, Daniel, ANDERES, Kenna, RICE, William G, O'BRIEN, Sean, SCHWAEBE, Michael, LIN, Amy, BLIESATH, Josh, HO, Caroline B, PROFFITT, Chris, TRENT, Katy, WHITTEN, Jeffrey P
Published in Cancer research (Chicago, Ill.) (01.10.2009)

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Journal Article

Discovery and SAR of 5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-8-carboxylic Acid (CX-4945), the First Clinical Stage Inhibitor of Protein Kinase CK2 for the Treatment of Cancer

Discovery and SAR of 5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-8-carboxylic Acid (CX-4945), the First Clinical Stage Inhibitor of Protein Kinase CK2 for the Treatment of Cancer

by Pierre, Fabrice, Chua, Peter C, O’Brien, Sean E, Siddiqui-Jain, Adam, Bourbon, Pauline, Haddach, Mustapha, Michaux, Jerome, Nagasawa, Johnny, Schwaebe, Michael K, Stefan, Eric, Vialettes, Anne, Whitten, Jeffrey P, Chen, Ta Kung, Darjania, Levan, Stansfield, Ryan, Anderes, Kenna, Bliesath, Josh, Drygin, Denis, Ho, Caroline, Omori, May, Proffitt, Chris, Streiner, Nicole, Trent, Katy, Rice, William G, Ryckman, David M
Published in Journal of medicinal chemistry (27.01.2011)

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Pre-clinical characterization of CX-4945, a potent and selective small molecule inhibitor of CK2 for the treatment of cancer

Pre-clinical characterization of CX-4945, a potent and selective small molecule inhibitor of CK2 for the treatment of cancer

by Pierre, Fabrice, Chua, Peter C., O’Brien, Sean E., Siddiqui-Jain, Adam, Bourbon, Pauline, Haddach, Mustapha, Michaux, Jerome, Nagasawa, Johnny, Schwaebe, Michael K., Stefan, Eric, Vialettes, Anne, Whitten, Jeffrey P., Chen, Ta Kung, Darjania, Levan, Stansfield, Ryan, Bliesath, Joshua, Drygin, Denis, Ho, Caroline, Omori, May, Proffitt, Chris, Streiner, Nicole, Rice, William G., Ryckman, David M., Anderes, Kenna
Published in Molecular and cellular biochemistry (01.10.2011)

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Discovery of CX-5461, the First Direct and Selective Inhibitor of RNA Polymerase I, for Cancer Therapeutics

Discovery of CX-5461, the First Direct and Selective Inhibitor of RNA Polymerase I, for Cancer Therapeutics

by Haddach, Mustapha, Schwaebe, Michael K, Michaux, Jerome, Nagasawa, Johnny, O'Brien, Sean E, Whitten, Jeffrey P, Pierre, Fabrice, Kerdoncuff, Pauline, Darjania, Levan, Stansfield, Ryan, Drygin, Denis, Anderes, Kenna, Proffitt, Chris, Bliesath, Josh, Siddiqui-Jain, Adam, Omori, May, Huser, Nanni, Rice, William G, Ryckman, David M
Published in ACS medicinal chemistry letters (12.07.2012)

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Discovery of CX-6258. A Potent, Selective, and Orally Efficacious pan-Pim Kinases Inhibitor

Discovery of CX-6258. A Potent, Selective, and Orally Efficacious pan-Pim Kinases Inhibitor

by Haddach, Mustapha, Michaux, Jerome, Schwaebe, Michael K, Pierre, Fabrice, O’Brien, Sean E, Borsan, Cosmin, Tran, Joe, Raffaele, Nicholas, Ravula, Suchitra, Drygin, Denis, Siddiqui-Jain, Adam, Darjania, Levan, Stansfield, Ryan, Proffitt, Chris, Macalino, Diwata, Streiner, Nicole, Bliesath, Joshua, Omori, May, Whitten, Jeffrey P, Anderes, Kenna, Rice, William G, Ryckman, David M
Published in ACS medicinal chemistry letters (09.02.2012)

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Determination of the importance of the stereochemistry of psorospermin in topoisomerase II–induced alkylation of DNA and in vitro and in vivo biological activity

Determination of the importance of the stereochemistry of psorospermin in topoisomerase II–induced alkylation of DNA and in vitro and in vivo biological activity

by Fellows, Ingrid M, Schwaebe, Michael, Dexheimer, Thomas S, Vankayalapati, Hariprasad, Gleason-Guzman, Mary, Whitten, Jeffrey P, Hurley, Laurence H
Published in Molecular cancer therapeutics (01.11.2005)

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Design and Synthesis of a Series of Non-Peptide High-Affinity Human Corticotropin-Releasing Factor1 Receptor Antagonists

Design and Synthesis of a Series of Non-Peptide High-Affinity Human Corticotropin-Releasing Factor1 Receptor Antagonists

by Chen, Dagnino, Raymond, De Souza, Errol B, Grigoriadis, Dimitri E, Huang, Charles Q, Kim, Kyung-Il, Liu, Zhengyu, Moran, Terry, Webb, Thomas R, Whitten, Jeffrey P, Xie, Yun Feng, McCarthy, James R
Published in Journal of medicinal chemistry (25.10.1996)

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Journal Article

COMPOUND REGULATING INTRACELLULAR CALCIUM

COMPOUND REGULATING INTRACELLULAR CALCIUM

by WANG ZHIJUN, BRIAN DYCK, JEFFREY P WHITTEN, CAO JIANGUO, JONATHAN GREY, EVAN ROGERS, PEI YAZHONG
Year of Publication 30.07.2020

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Patent

Nickel(0)-catalyzed coupling of vinylzirconiums to α-bromo-α,α-difluoro esters. Convenient generation of a functionalized allyldifluoro moiety

Nickel(0)-catalyzed coupling of vinylzirconiums to α-bromo-α,α-difluoro esters. Convenient generation of a functionalized allyldifluoro moiety

by Schwaebe, Michael K, McCarthy, James R, Whitten, Jeffrey P
Published in Tetrahedron letters (05.02.2000)

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Journal Article

COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM

COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM

by WANG ZHIJUN, BRIAN DYCK, JEFFREY P WHITTEN, CAO JIANGUO, JONATHAN GREY, EVAN ROGERS, PEI YAZHONG
Year of Publication 11.04.2019

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Patent

COMPOUNDS FOR MODULATING INTRACELLULAR CALCIUM

COMPOUNDS FOR MODULATING INTRACELLULAR CALCIUM

by WANG ZHIJUN, BRIAN DYCK, JEFFREY P WHITTEN, CAO JIANGUO, JONATHAN GREY, EVAN ROGERS, PEI YAZHONG
Year of Publication 07.12.2017

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Patent

Modeling of competitive phosphono amino acid NMDA receptor antagonists

Modeling of competitive phosphono amino acid NMDA receptor antagonists

by Whitten, Jeffrey P, Harrison, Boyd L, Weintraub, Herschel J. R, McDonald, Ian A
Published in Journal of medicinal chemistry (01.05.1992)

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Journal Article

COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM

COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM

by WANG ZHIJUN, BRIAN DYCK, JEFFREY P WHITTEN, CAO JIANGUO, JONATHAN GREY, EVAN ROGERS, PEI YAZHONG
Year of Publication 08.06.2017

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Patent

Synthesis and cardiotonic activity of novel biimidazoles

Synthesis and cardiotonic activity of novel biimidazoles

by Matthews, Donald P, McCarthy, James R, Whitten, Jeffrey P, Kastner, Philip R, Barney, Charlotte L, Marshall, Franklin N, Ertel, Marcia A, Burkhard, Therese, Shea, Philip J, Kariya, Takashi
Published in Journal of medicinal chemistry (01.01.1990)

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Journal Article

Design, synthesis, and SAR of 2-dialkylamino-4-arylpyrimidines as potent and selective corticotropin-releasing factor1 (CRF1) receptor antagonists

Design, synthesis, and SAR of 2-dialkylamino-4-arylpyrimidines as potent and selective corticotropin-releasing factor1 (CRF1) receptor antagonists

by HUANG, Charles Q, GRIGORIADIS, Dimitri E, ZHENGYU LIU, MCCARTHY, James R, RAMPHAL, John, WEBB, Thomas, WHITTEN, Jeffrey P, XIE, Michael Y, CHEN CHEN
Published in Bioorganic & medicinal chemistry letters (03.05.2004)

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Journal Article

INTERCELLULAR CALCIUM MODULATING COMPOUND

INTERCELLULAR CALCIUM MODULATING COMPOUND

by WANG ZHIJUN, BRIAN DYCK, JEFFREY P WHITTEN, CAO JIANGUO, JONATHAN GREY, EVAN ROGERS, PEI YAZHONG
Year of Publication 14.01.2016

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Patent

Rapid Microscale Synthesis, a New Method for Lead Optimization Using Robotics and Solution Phase Chemistry: Application to the Synthesis and Optimization of Corticotropin-Releasing Factor1 Receptor Antagonists

Rapid Microscale Synthesis, a New Method for Lead Optimization Using Robotics and Solution Phase Chemistry: Application to the Synthesis and Optimization of Corticotropin-Releasing Factor1 Receptor Antagonists

by Whitten, Jeffrey P, Xie, Yun Feng, Erickson, Philip E, Webb, Thomas R, De Souza, Errol B, Grigoriadis, Dimitri E, McCarthy, James R
Published in Journal of medicinal chemistry (25.10.1996)

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Journal Article

Facile synthesis of the four 3-aminocyclopentane-1,2-diol stereoisomers

Facile synthesis of the four 3-aminocyclopentane-1,2-diol stereoisomers

by Whitten, Jeffrey P, McCarthy, James R, Whalon, Michael R
Published in Journal of organic chemistry (01.11.1985)

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Journal Article

[2-(Trimethylsilyl)ethoxy]methyl (SEM) as a novel and effective imidazole and fused aromatic imidazole protecting group

[2-(Trimethylsilyl)ethoxy]methyl (SEM) as a novel and effective imidazole and fused aromatic imidazole protecting group

by Whitten, Jeffrey P, Matthews, Donald P, McCarthy, James R
Published in Journal of organic chemistry (01.05.1986)

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Journal Article

(R)-4-Oxo-5-phosphononorvaline: a new competitive glutamate antagonist at the NMDA receptor complex

(R)-4-Oxo-5-phosphononorvaline: a new competitive glutamate antagonist at the NMDA receptor complex

by Whitten, Jeffrey P, Baron, Bruce M, Muench, Daniel, Miller, Francis, White, H. Steven, McDonald, Ian A
Published in Journal of medicinal chemistry (01.11.1990)

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