Dissociation of Transactivation from Transrepression by a Selective Glucocorticoid Receptor Agonist Leads to Separation of Therapeutic Effects from Side Effects
Schäcke, Heike, Schottelius, Arndt, Döcke, Wolf-Dietrich, Strehlke, Peter, Jaroch, Stefan, Schmees, Norbert, Rehwinkel, Hartmut, Hennekes, Hartwig, Asadullah, Khusru
Published in Proceedings of the National Academy of Sciences - PNAS (06.01.2004)
Published in Proceedings of the National Academy of Sciences - PNAS (06.01.2004)
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Discovery of the potent non-steroidal glucocorticoid receptor modulator BAY 1003803 as clinical candidate
Berger, Markus, May, Ekkehard, Rehwinkel, Hartmut, Schäcke, Heike, Neuhaus, Roland, Rottmann, Antje, Zollner, Thomas M., Jaroch, Stefan
Published in Bioorganic & medicinal chemistry letters (15.08.2020)
Published in Bioorganic & medicinal chemistry letters (15.08.2020)
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Discovery of new selective glucocorticoid receptor agonist leads
Berger, Markus, Rehwinkel, Hartmut, Schmees, Norbert, Schäcke, Heike, Edman, Karl, Wissler, Lisa, Reichel, Andreas, Jaroch, Stefan
Published in Bioorganic & medicinal chemistry letters (01.02.2017)
Published in Bioorganic & medicinal chemistry letters (01.02.2017)
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Correction to “Total Synthesis of (−)-Sarain A”
Becker, Michael H, Chua, Peter, Downham, Robert, Douglas, Christopher J, Garg, Neil K, Hiebert, Sheldon, Jaroch, Stefan, Matsuoka, Richard T, Middleton, Joy A, Ng, Fay W, Overman, Larry E
Published in Journal of the American Chemical Society (18.04.2018)
Published in Journal of the American Chemical Society (18.04.2018)
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Abstract 4332: Discovery of BAY 1163877 - A pan-FGFR inhibitor: De novo structure-based design and lead optimization of benzothiophenyl-pyrrolotriazines
Collin, Marie-Pierre L., Lobell, Mario, Huebsch, Walter, Brohm, Dirk, Héroult, Mélanie, Lustig, Klemens, Gruenewald, Sylvia, Boemer, Ulf, Jautelat, Rolf, Hess-Stump, Holger, Jaroch, Stefan, Brands, Michael, Ziegelbauer, Karl
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Total Synthesis of (−)-Sarain A
Becker, Michael H, Chua, Peter, Downham, Robert, Douglas, Christopher J, Garg, Neil K, Hiebert, Sheldon, Jaroch, Stefan, Matsuoka, Richard T, Middleton, Joy A, Ng, Fay W, Overman, Larry E
Published in Journal of the American Chemical Society (03.10.2007)
Published in Journal of the American Chemical Society (03.10.2007)
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Discovery of quinolines as selective glucocorticoid receptor agonists
Jaroch, Stefan, Berger, Markus, Huwe, Christoph, Krolikiewicz, Konrad, Rehwinkel, Hartmut, Schäcke, Heike, Schmees, Norbert, Skuballa, Werner
Published in Bioorganic & medicinal chemistry letters (01.10.2010)
Published in Bioorganic & medicinal chemistry letters (01.10.2010)
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Journal Article
Role of neuronal nitric oxide synthase in ovine sepsis model
Enkhbaatar, Perenlei, Lange, Matthias, Nakano, Yoshimitsu, Hamahata, Atsumori, Jonkam, Collette, Wang, Jianpu, Jaroch, Stefan, Traber, Lillian, Herndon, David, Traber, Daniel
Published in Shock (Augusta, Ga.) (01.09.2009)
Published in Shock (Augusta, Ga.) (01.09.2009)
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Inhibition of neuronal nitric oxide synthase in ovine model of acute lung injury
Enkhbaatar, Perenlei, Connelly, Rhykka, Wang, Jianpu, Nakano, Yoshimitsu, Lange, Matthias, Hamahata, Atsumori, Horvath, Eszter, Szabo, Csaba, Jaroch, Stefan, Hölscher, Peter, Hillmann, Margrit, Traber, Lillian D, Schmalstieg, Frank C, Herndon, David N, Traber, Daniel L
Published in Critical care medicine (01.01.2009)
Published in Critical care medicine (01.01.2009)
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Journal Article
CCR5 receptor antagonists: Discovery and SAR of novel 4-hydroxypiperidine derivatives
Lu, Shou-Fu, Chen, Binglong, Davey, Dave, Dunning, Laura, Jaroch, Stefan, May, Karen, Onuffer, James, Phillips, Gary, Subramanyam, Babu, Tseng, Jih-Lie, Wei, Robert G., Wei, Ming, Ye, Bin
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
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Journal Article
P117. Role of nitric oxide in sepsis following smoke inhalation and pneumonia
Enkhbaatar, Perenlei, Traber, Lillian D., Jaroch, Stefan, Cox, Robert, Hawkins, Hal, Schmalstieg, Frank, Herndon, David, Traber, Daniel L.
Published in Nitric oxide (01.06.2006)
Published in Nitric oxide (01.06.2006)
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Dihydroquinolines with amine-containing side chains as potent n-NOS inhibitors
Jaroch, Stefan, Hölscher, Peter, Rehwinkel, Hartmut, Sülzle, Detlev, Burton, Gerardine, Hillmann, Margrit, McDonald, Fiona M.
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
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Journal Article
Dihydroquinolines as Novel n-NOS Inhibitors
Jaroch, Stefan, Hölscher, Peter, Rehwinkel, Hartmut, Sülzle, Detlev, Burton, Gerardine, Hillmann, Margrit, McDonald, Fiona M.
Published in Bioorganic & medicinal chemistry letters (16.09.2002)
Published in Bioorganic & medicinal chemistry letters (16.09.2002)
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Journal Article
Alkylidene-tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents
BAEURLE STEFAN,BERGER MARKUS,JAROCH STEFAN,KROLIKIEWICZ KONRAD,NGUYEN DUY,REHWINKEL HARTMUT,SCHAECKE HEIKE,SCHMEES NORBERT,SKUBALLA WERNER
Year of Publication 31.10.2007
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Year of Publication 31.10.2007
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