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Published in Cell host & microbe (08.10.2014)
Published in Cell host & microbe (08.10.2014)
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Gremlin regulates renal inflammation via the vascular endothelial growth factor receptor 2 pathway
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Published in The Journal of pathology (01.08.2015)
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Identification of aminopyrimidine‐sulfonamides as potent modulators of Wag31‐mediated cell elongation in mycobacteria
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Published in Molecular microbiology (01.01.2017)
Published in Molecular microbiology (01.01.2017)
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Lead selection and characterization of antitubercular compounds using the Nested Chemical Library
Sipos, Anna, Pató, János, Székely, Rita, Hartkoorn, Ruben C, Kékesi, László, Őrfi, László, Szántai-Kis, Csaba, Mikušová, Katarína, Svetlíková, Zuzana, Korduláková, Jana, Nagaraja, Valakunja, Godbole, Adwait Anand, Bush, Natassja, Collin, Frédéric, Maxwell, Anthony, Cole, Stewart T, Kéri, György
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Published in Tuberculosis (Edinburgh, Scotland) (01.06.2015)
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Development of a Cell-Selective and Intrinsically Active Multikinase Inhibitor Bioconjugate
Harmsen, Stefan, Dolman, M. Emmy M, Nemes, Zoltan, Lacombe, Marie, Szokol, Bálint, Pató, János, Kéri, György, Őrfi, László, Storm, Gert, Hennink, Wim E, Kok, Robbert J
Published in Bioconjugate chemistry (20.04.2011)
Published in Bioconjugate chemistry (20.04.2011)
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Connective tissue growth factor is a new ligand of epidermal growth factor receptor
Rayego-Mateos, Sandra, Rodrigues-Díez, Raquel, Morgado-Pascual, Jose Luis, Rodrigues Díez, Raul R, Mas, Sebastian, Lavoz, Carolina, Alique, Matilde, Pato, Janos, Keri, Gyorgy, Ortiz, Alberto, Egido, Jesus, Ruiz-Ortega, Marta
Published in Journal of molecular cell biology (01.10.2013)
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A novel drug discovery concept for tuberculosis: Inhibition of bacterial and host cell signalling
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Published in Immunology letters (15.03.2008)
Published in Immunology letters (15.03.2008)
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Improved, High Yield Synthesis of 3H-Quinazolin-4-ones, the Key Intermediates of Recently Developed Drugs
Orfi, Laszlo, Waczek, Frigyes, Pato, Janos, Varga, Istvan, Hegymegi-Barakonyi, Balint, Houghten, Richard A., Ker, Gyorgy
Published in Current medicinal chemistry (01.10.2004)
Published in Current medicinal chemistry (01.10.2004)
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Székelyhidi, Zsolt, Pató, János, Wáczek, Frigyes, Bánhegyi, Péter, Hegymegi-Barakonyi, Bálint, Ero˝s, Dániel, Mészáros, György, Hollósy, Ferenc, Hafenbradl, Doris, Obert, Sabine, Klebl, Bert, Kéri, György, O˝rfi, László
Published in Bioorganic & medicinal chemistry letters (01.07.2005)
Published in Bioorganic & medicinal chemistry letters (01.07.2005)
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Machine learning and docking models for Mycobacterium tuberculosis topoisomerase I
Ekins, Sean, Godbole, Adwait Anand, Kéri, György, Orfi, Lászlo, Pato, János, Bhat, Rajeshwari Subray, Verma, Rinkee, Bradley, Erin K, Nagaraja, Valakunja
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Synthesis and characterization of novel quinazoline type inhibitors for mutant and wild-type EGFR and RICK kinases
Breza, Nora, Pato, Janos, Orfi, Laszlo, Hegymegi-Barakonyi, Balint, Banhegyi, Peter, Varkondi, Edit, Borbely, Gabor, Petak, Istvan, Keri, Gyorgy
Published in Journal of receptors and signal transduction (01.01.2008)
Published in Journal of receptors and signal transduction (01.01.2008)
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Synthesis and Structure–Activity relationship of 1-(5-isoquinolinesulfonyl)piperazine analogues as inhibitors of Mycobacterium tuberculosis IMPDH
Singh, Vinayak, Pacitto, Angela, Donini, Stefano, Ferraris, Davide M., Boros, Sándor, Illyés, Eszter, Szokol, Bálint, Rizzi, Menico, Blundell, Tom L., Ascher, David B., Pato, Janos, Mizrahi, Valerie
Published in European journal of medicinal chemistry (15.07.2019)
Published in European journal of medicinal chemistry (15.07.2019)
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TWEAK transactivation of the epidermal growth factor receptor mediates renal inflammation
Rayego-Mateos, Sandra, Morgado-Pascual, Jose Luis, Sanz, Ana Belen, Ramos, Adrian Mario, Eguchi, Satoru, Batlle, Daniel, Pato, Janos, Keri, Gyorgy, Egido, Jesus, Ortiz, Alberto, Ruiz-Ortega, Marta
Published in The Journal of pathology (01.12.2013)
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The Inosine Monophosphate Dehydrogenase, GuaB2, Is a Vulnerable New Bactericidal Drug Target for Tuberculosis
Singh, Vinayak, Donini, Stefano, Pacitto, Angela, Sala, Claudia, Hartkoorn, Ruben C, Dhar, Neeraj, Keri, Gyorgy, Ascher, David B, Mondésert, Guillaume, Vocat, Anthony, Lupien, Andréanne, Sommer, Raphael, Vermet, Hélène, Lagrange, Sophie, Buechler, Joe, Warner, Digby F, McKinney, John D, Pato, Janos, Cole, Stewart T, Blundell, Tom L, Rizzi, Menico, Mizrahi, Valerie
Published in ACS infectious diseases (13.01.2017)
Published in ACS infectious diseases (13.01.2017)
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The C-terminal module IV of connective tissue growth factor, through EGFR/Nox1 signaling, activates the NF-κB pathway and proinflammatory factors in vascular smooth muscle cells
Rodrigues-Diez, Raúl R, Garcia-Redondo, Ana Belen, Orejudo, Macarena, Rodrigues-Diez, Raquel, Briones, Ana Maria, Bosch-Panadero, Enrique, Kery, Gyorgy, Pato, Janos, Ortiz, Alberto, Salaices, Mercedes, Egido, Jesus, Ruiz-Ortega, Marta
Published in Antioxidants & redox signaling (01.01.2015)
Published in Antioxidants & redox signaling (01.01.2015)
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Keri, Gyorgy, Orfi, Laszlo, Greff, Zoltan, Pato, Janos, Szokol, Balint, Kekesi, Laszlo, Sipos, Anna, Garamvolgyi, Rita
Published in Current opinion in biotechnology (01.07.2013)
Published in Current opinion in biotechnology (01.07.2013)
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Leads for antitubercular compounds from kinase inhibitor library screens
Magnet, Sophie, Hartkoorn, Ruben C, Székely, Rita, Pató, János, Triccas, James A, Schneider, Patricia, Szántai-Kis, Csaba, Őrfi, László, Chambon, Marc, Banfi, Damiano, Bueno, Manuel, Turcatti, Gerardo, Kéri, György, Cole, Stewart T
Published in Tuberculosis (Edinburgh, Scotland) (01.11.2010)
Published in Tuberculosis (Edinburgh, Scotland) (01.11.2010)
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Intervention in growth factor activated signaling pathways by renally targeted kinase inhibitors
Fretz, Marjan M., Dolman, M.E. (Emmy) M., Lacombe, Marie, Prakash, Jai, Nguyen, Tri Q., Goldschmeding, Roel, Pato, Janos, Storm, Gert, Hennink, Wim E., Kok, Robbert J.
Published in Journal of controlled release (18.12.2008)
Published in Journal of controlled release (18.12.2008)
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Conference Proceeding
Synthesis and biological evaluation of novel pyrido[2,3-b]pyrazines inhibiting both erlotinib-sensitive and erlotinib-resistant cell lines
Kékesi, László, Sipos, Anna, Németh, Gábor, Pató, János, Breza, Nóra, Baska, Ferenc, Őrfi, László, Kéri, György
Published in Bioorganic & medicinal chemistry letters (15.11.2013)
Published in Bioorganic & medicinal chemistry letters (15.11.2013)
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