Natural Products in Medicine: Transformational Outcome of Synthetic Chemistry
Szychowski, Janek, Truchon, Jean-François, Bennani, Youssef L
Published in Journal of medicinal chemistry (26.11.2014)
Published in Journal of medicinal chemistry (26.11.2014)
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Journal Article
Identification of secreted bacterial proteins by noncanonical amino acid tagging
Mahdavi, Alborz, Szychowski, Janek, Ngo, John T., Sweredoski, Michael J., Graham, Robert L. J., Hess, Sonja, Schneewind, Olaf, Mazmanian, Sarkis K., Tirrell, David A.
Published in Proceedings of the National Academy of Sciences - PNAS (07.01.2014)
Published in Proceedings of the National Academy of Sciences - PNAS (07.01.2014)
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Journal Article
Live-Cell Imaging of Cellular Proteins by a Strain-Promoted Azide-Alkyne Cycloaddition
Beatty, Kimberly E, Fisk, John D, Smart, Brian P, Lu, Ying Ying, Szychowski, Janek, Hangauer, Matthew J, Baskin, Jeremy M, Bertozzi, Carolyn R, Tirrell, David A
Published in Chembiochem : a European journal of chemical biology (18.10.2010)
Published in Chembiochem : a European journal of chemical biology (18.10.2010)
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Journal Article
Cleavable Biotin Probes for Labeling of Biomolecules via Azide−Alkyne Cycloaddition
Szychowski, Janek, Mahdavi, Alborz, Hodas, Jennifer J. L, Bagert, John D, Ngo, John T, Landgraf, Peter, Dieterich, Daniela C, Schuman, Erin M, Tirrell, David A
Published in Journal of the American Chemical Society (29.12.2010)
Published in Journal of the American Chemical Society (29.12.2010)
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Journal Article
Discovery of an Orally Bioavailable and Selective PKMYT1 Inhibitor, RP-6306
Szychowski, Janek, Papp, Robert, Dietrich, Evelyne, Liu, Bingcan, Vallée, Frédéric, Leclaire, Marie-Eve, Fourtounis, Jimmy, Martino, Giovanni, Perryman, Alexander L., Pau, Victor, Yin, Shou Yun, Mader, Pavel, Roulston, Anne, Truchon, Jean-Francois, Marshall, C. Gary, Diallo, Mohamed, Duffy, Nicole M., Stocco, Rino, Godbout, Claude, Bonneau-Fortin, Alexanne, Kryczka, Rosie, Bhaskaran, Vivek, Mao, Daniel, Orlicky, Stephen, Beaulieu, Patrick, Turcotte, Pascal, Kurinov, Igor, Sicheri, Frank, Mamane, Yael, Gallant, Michel, Black, W. Cameron
Published in Journal of medicinal chemistry (11.08.2022)
Published in Journal of medicinal chemistry (11.08.2022)
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Journal Article
A BODIPY-Cyclooctyne for Protein Imaging in Live Cells
Beatty, Kimberly E., Szychowski, Janek, Fisk, John D., Tirrell, David A.
Published in Chembiochem : a European journal of chemical biology (19.09.2011)
Published in Chembiochem : a European journal of chemical biology (19.09.2011)
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Journal Article
Abstract 5650: RP-6306, a novel PKMYT1 inhibitor, demonstrates synthetic lethality as monotherapy and in combination with gemcitabine in CCNE1 amplified cancer cells
Fourtounis, Jimmy, Martino, John, Stocco, Rino, Baruah, Prasamit, Duffy, Nicole, Gallo, David, Fournier, Sarah, Li, JingJing, Li, Li, Aguado, Elia, Petrone, Adam, Roulston, Anne, Mamane, Yael, Morris, Stephen, Szychowski, Janek, Papp, Robert, Zinda, Mike, Marshall, C. Gary
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Journal Article
Inhibition of Aminoglycoside-Deactivating Enzymes APH(3′)-IIIa and AAC(6′)-Ii by Amphiphilic Paromomycin O2′′-Ether Analogues
Szychowski, Janek, Kondo, Jiro, Zahr, Omar, Auclair, Karine, Westhof, Eric, Hanessian, Stephen, Keillor, Jeffrey W.
Published in ChemMedChem (04.11.2011)
Published in ChemMedChem (04.11.2011)
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Journal Article
Structure-based design, synthesis and A-site rRNA co-crystal complexes of novel amphiphilic aminoglycoside antibiotics with new binding modes: A synergistic hydrophobic effect against resistant bacteria
Hanessian, Stephen, Pachamuthu, Kandasamy, Szychowski, Janek, Giguère, Alexandre, Swayze, Eric E., Migawa, Michael T., François, Boris, Kondo, Jiro, Westhof, Eric
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
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Journal Article
Robust polymeric nanoparticles for the delivery of aminoglycoside antibiotics using carboxymethyldextran-b-poly(ethyleneglycols) lightly grafted with n-dodecyl groups
Soliman, Ghareb M., Szychowski, Janek, Hanessian, Stephen, Winnik, Françoise M.
Published in Soft matter (01.01.2010)
Published in Soft matter (01.01.2010)
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Journal Article
Robust polymeric nanoparticles for the delivery of aminoglycoside antibiotics using carboxymethyldextran-b-poly(ethyleneglycols) lightly grafted with n-dodecyl groupsElectronic supplementary information (ESI) available: Further information. See DOI: 10.1039/c0sm00316f
Soliman, Ghareb M, Szychowski, Janek, Hanessian, Stephen, Winnik, Françoise M
Year of Publication 02.09.2010
Year of Publication 02.09.2010
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Journal Article
Antibacterial Aminoglycosides with a Modified Mode of Binding to the Ribosomal-RNA Decoding Site
François, Boris, Szychowski, Janek, Adhikari, Susanta Sekhar, Pachamuthu, Kandasamy, Swayze, Eric E., Griffey, Richard H., Migawa, Michael T., Westhof, Eric, Hanessian, Stephen
Published in Angewandte Chemie (International ed.) (10.12.2004)
Published in Angewandte Chemie (International ed.) (10.12.2004)
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Journal Article
Crystal Structure of the Bacterial Ribosomal Decoding Site Complexed with a Synthetic Doubly Functionalized Paromomycin Derivative: a New Specific Binding Mode to an A-Minor Motif Enhances in vitro Antibacterial Activity
Kondo, Jiro, Pachamuthu, Kandasamy, François, Boris, Szychowski, Janek, Hanessian, Stephen, Westhof, Eric
Published in ChemMedChem (12.11.2007)
Published in ChemMedChem (12.11.2007)
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Journal Article
Structure-Based Design, Synthesis, and A-Site rRNA Cocrystal Complexes of Functionally Novel Aminoglycoside Antibiotics: C2‘ ‘ Ether Analogues of Paromomycin
Hanessian, Stephen, Szychowski, Janek, Adhikari, Susanta Sekhar, Vasquez, Guillermo, Kandasamy, Pachamuthu, Swayze, Eric E, Migawa, Michael T, Ranken, Ray, François, Boris, Wirmer-Bartoschek, Julia, Kondo, Jiro, Westhof, Eric
Published in Journal of medicinal chemistry (17.05.2007)
Published in Journal of medicinal chemistry (17.05.2007)
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Journal Article
Inside Cover: Inhibition of Aminoglycoside-Deactivating Enzymes APH(3′)-IIIa and AAC(6′)-Ii by Amphiphilic Paromomycin O2′′-Ether Analogues (ChemMedChem 11/2011)
Szychowski, Janek, Kondo, Jiro, Zahr, Omar, Auclair, Karine, Westhof, Eric, Hanessian, Stephen, Keillor, Jeffrey W.
Published in ChemMedChem (04.11.2011)
Published in ChemMedChem (04.11.2011)
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Journal Article
Probing the ribosomal RNA A-site with functionally diverse analogues of paromomycin—synthesis of ring I mimetics
Hanessian, Stephen, Adhikari, Susanta, Szychowski, Janek, Pachamuthu, Kandasmy, Wang, Xiaojing, Migawa, Michael T., Griffey, Richard H., Swayze, Eric E.
Published in Tetrahedron (22.01.2007)
Published in Tetrahedron (22.01.2007)
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Journal Article
6-Hydroxy to 6‴-amino tethered ring-to-ring macrocyclic aminoglycosides as probes for APH(3′)-IIIa kinase
Hanessian, Stephen, Szychowski, Janek, Campos-Reales Pineda, Natalhie B., Furtos, Alexandra, Keillor, Jeffrey W.
Published in Bioorganic & medicinal chemistry letters (01.06.2007)
Published in Bioorganic & medicinal chemistry letters (01.06.2007)
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Journal Article
Corrigendum to “Probing the ribosomal RNA A-site with functionally diverse analogues of paromomycin—synthesis of ring I mimetics”: [Tetrahedron 63 (2007) 827–846]
Hanessian, Stephen, Adhikari, Susanta, Szychowski, Janek, Pachamuthu, Kandasmy, Wang, Xiaojing, Migawa, Michael T., Griffey, Richard H., Swayze, Eric E.
Published in Tetrahedron (11.06.2007)
Published in Tetrahedron (11.06.2007)
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Journal Article