Mode of Action for Linear Peptide Inhibitors of HIV-1 gp120 Interactions
Biorn, Alyssa C, Cocklin, Simon, Madani, Navid, Si, Zhihai, Ivanovic, Tijana, Samanen, James, Van Ryk, Donald I, Pantophlet, Ralph, Burton, Dennis R, Freire, Ernesto, Sodroski, Joseph, Chaiken, Irwin M
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Phenylbutyrates as potent, orally bioavailable vitronectin receptor (integrin αvβ3) antagonists
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Discovery of Orally Active Nonpeptide Vitronectin Receptor Antagonists Based on a 2-Benzazepine Gly-Asp Mimetic
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Modulation of vitronectin receptor-mediated osteoclast adhesion by Arg-Gly-Asp peptide analogs: a structure-function analysis
Horton, M A, Dorey, E L, Nesbitt, S A, Samanen, J, Ali, F E, Stadel, J M, Nichols, A, Greig, R, Helfrich, M H
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Potent nonpeptide angiotensin II receptor antagonists. 2. 1-(Carboxybenzyl)imidazole-5-acrylic acids
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Potent, Selective, Orally Active 3-Oxo-1,4-benzodiazepine GPIIb/IIIa Integrin Antagonists
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Enantioselective routes to protected syn- and anti-.beta.-phenylcysteines
Lago, M. Amparo, Samanen, James, Elliott, John D
Published in Journal of organic chemistry (01.06.1992)
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Chemical approaches to improve the oral bioavailability of peptidergic molecules
Samanen, J, Wilson, G, Smith, P L, Lee, C P, Bondinell, W, Ku, T, Rhodes, G, Nichols, A
Published in Journal of pharmacy and pharmacology (01.02.1996)
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Potent non-peptide fibrinogen receptor antagonists which present an alternative pharmacophore
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Discovery of Potent Nonpeptide Vitronectin Receptor (αVβ3) Antagonists
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Samanen, James M., Lee, Chao-Pin, Smith, Philip L., Bondinell, William E., Calvo, Raul R., Jakas, Dalia R., Newlander, Kenneth A., Parker, Michael, Uzinskas, Irene, Yellin, Tobias O., Nichols, Andrew J.
Published in Advanced drug delivery reviews (15.01.1997)
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Published in Tetrahedron letters (25.12.1995)
Published in Tetrahedron letters (25.12.1995)
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SAMANEN JAMES MARTIN SAMANEN JAMES MARTIN, MILLER WILLIAM H. MILLER WILLIAM H, HEERDING DIRK HEERDING DIRK, BONDINELL WILLIAM E. BONDINELL WILLIAM E
Year of Publication 28.03.2001
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Year of Publication 28.03.2001
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The antithrombotic efficacy of lotrafiban (SB 214857) in canine models of acute coronary thrombosis
Toomey, John R, Samanen, James, Valocik, Richard E, Koster, Paul F, Barone, Frank C, Willette, Robert N
Published in Current drug targets. Cardiovascular & hematological disorders (01.06.2002)
Published in Current drug targets. Cardiovascular & hematological disorders (01.06.2002)
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The in vitro pharmacological profile of SK&F 106760, a novel GPIIB/IIIA antagonist
Nichols, Andrew J., Vasko, Janice A., Valocik, Richard E., Kopaciewicz, Linda J., Storer, Barbara L., Ali, Fadia E., Romoff, Todd, Calvo, Raul, Samanen, James M.
Published in Thrombosis research (15.07.1994)
Published in Thrombosis research (15.07.1994)
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