Solid-state characterization of the new antiparasitic drug 5-((5-bromo-1H-indol-3-yl)methylene)-3-(2,6-difluorobenzyl)thiazolidine-2,4-dione (GQ-238)
de Andrade, Fabrício Havy Dantas, de Oliveira, Jamerson Ferreira, da Silva, Paulo César Dantas, da Rocha Pitta, Ivan, Silva, Isabella Nayara Santos, de Oliveira Macedo, Rui, De Lima, Maria do Carmo Alves, Rolim-Neto, Pedro Jose, da Silva, Rosali Maria Ferreira, de Souza, Fábio Santos
Published in Journal of thermal analysis and calorimetry (01.08.2020)
Published in Journal of thermal analysis and calorimetry (01.08.2020)
Get full text
Journal Article
Novel 4-quinoline-thiosemicarbazone derivatives: Synthesis, antiproliferative activity, in vitro and in silico biomacromolecule interaction studies and topoisomerase inhibition
Ribeiro, Amélia Galdino, Almeida, Sinara Mônica Vitalino de, de Oliveira, Jamerson Ferreira, Souza, Tulio Ricardo Couto de Lima, Santos, Keriolaine Lima dos, Albuquerque, Amanda Pinheiro de Barros, Nogueira, Mariane Cajuba de Britto Lira, Carvalho Junior, Luiz Bezerra de, Moura, Ricardo Olímpio de, da Silva, Aline Caroline, Pereira, Valéria Rêgo Alves, Castro, Maria Carolina Accioly Brelaz de, Lima, Maria do Carmo Alves de
Published in European journal of medicinal chemistry (15.11.2019)
Published in European journal of medicinal chemistry (15.11.2019)
Get full text
Journal Article
Synthesis, in vitro and in vivo biological evaluation, COX-1/2 inhibition and molecular docking study of indole-N-acylhydrazone derivatives
Moraes, Ana Daura Travassos de Oliveira, Miranda, Mirelly Dianne Santos de, Jacob, Íris Trindade Tenório, Amorim, Cézar Augusto da Cruz, Moura, Ricardo Olímpio de, Silva, Simone Ângela Soares da, Soares, Milena Botelho Pereira, Almeida, Sinara Mônica Vitalino de, Souza, Túlio Ricardo Couto de Lima, Oliveira, Jamerson Ferreira de, Silva, Teresinha Gonçalves da, Melo, Cristiane Moutinho Lagos de, Moreira, Diogo Rodrigo Magalhães, Lima, Maria do Carmo Alves de
Published in Bioorganic & medicinal chemistry (01.11.2018)
Published in Bioorganic & medicinal chemistry (01.11.2018)
Get full text
Journal Article
Development and evaluation of the in vitro schistosomicidal activity of solid dispersions based on 2-(-5-bromo-1-H-indole-3-yl-methylene)-N-(naphthalene-1-ylhydrazine-carbothiamide
de Luna Rocha, Thâmara Carollyne, Dos Santos Lima, Maria Joanellys, Nunes do Nascimento, Jéfferson Luan, Ferreira de Oliveira, Jamerson, de Oliveira Silva, Emerson, Barbosa Dos Santos, Victor Hugo, de Lima Aires, André, de Albuquerque Wanderley Sales, Victor, Atanazio Rosa, Talita, Rolim Neto, Pedro José, Camelo Pessôa de Azevedo Albuquerque, Mônica, Alves de Lima, Maria do Carmo, Ferreira da Silva, Rosali Maria
Published in Experimental parasitology (01.01.2024)
Published in Experimental parasitology (01.01.2024)
Get full text
Journal Article
Thiazolidinedione and thiazole derivatives potentiate norfloxacin activity against NorA efflux pump over expression in Staphylococcus aureus 1199B strains
Pereira, Pedro Silvino, Lima, Maria do Carmo Alves de, Neto, Pedro Paulo Marcelino, Oliveira-Tintino, Cícera Datiane de Morais, Tintino, Saulo Relison, Menezes, Irwin Rose de Alencar, de Oliveira, Jamerson Ferreira, Marchand, Pascal, Coutinho, Henrique Douglas Melo, Rodrigues, Maria do Desterro, da Silva, Teresinha Gonçalves
Published in Bioorganic & medicinal chemistry (01.09.2019)
Published in Bioorganic & medicinal chemistry (01.09.2019)
Get full text
Journal Article
Synthesis, thermal behavior and biological evaluation of benzodioxole derivatives as potential cytotoxic and antiparasitic agents
Silva, Willams Leal, de Andrade, Fabricio Havy Dantas, Lins, Taynara Batista, da Silva, Anekécia Lauro, da Cruz Amorim, Cezar Augusto, dos Santos Lima, Maria Joanellys, da Silva, Paulo César Dantas, Vilela, Williana Tôrres, Nascimento, Pedro Henrique do Bomfim, de Oliveira, Jamerson Ferreira, de Souza, Fábio Santos, Alves de Lima, Maria do Carmo, da Silva, Rosali Maria Ferreira
Published in Medicinal chemistry research (01.05.2023)
Published in Medicinal chemistry research (01.05.2023)
Get full text
Journal Article
Neurolocomotor Behavior and Oxidative Stress Markers of Thiazole and Thiazolidinedione Derivatives against Nauphoeta cinerea
Pereira, Pedro Silvino, Costa, Adrielle Rodrigues, de Oliveira, Thalyta Julyanne Silva, Oliveira, Carlos Vinícius Barros, de Lima, Maria do Carmo Alves, de Oliveira, Jamerson Ferreira, Kim, Bonglee, Coutinho, Henrique D M, Duarte, Antonia Eliene, Kamdem, Jean Paul, da Silva, Teresinha Gonçalves
Published in Antioxidants (18.02.2022)
Published in Antioxidants (18.02.2022)
Get full text
Journal Article
New Oxazolidines Inhibit the Secretion of IFN-γ and IL-17 by PBMCS from Moderate to Severe Asthmatic Patients
Santos, Renata Virgínia Cavalcanti, Cunha, Eudes Gustavo Constantino, de Mello, Gabriela Souto Vieira, Rizzo, José Ângelo, de Oliveira, Jamerson Ferreira, do Carmo Alves de Lima, Maria, da Rocha Pitta, Ivan, da Rocha Pitta, Maira Galdino, de Melo Rêgo, Moacyr Jesus Barreto
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2021)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2021)
Get more information
Journal Article
Synthesis and biological evaluation of novel imidazolidine derivatives as candidates to schistosomicidal agents
Matos-Rocha, Thiago José, Lima, Maria do Carmo Alves de, Silva, Anekécia Lauro da, Oliveira, Jamerson Ferreira de, Gouveia, Allana Lemos Andrade, Silva, Vinícius Barros Ribeiro da, Almeida, Júnior, Antônio Sérgio Alves de, Brayner, Fábio André, Cardoso, Pablo Ramon Gualberto, Pitta-Galdino, Marina da Rocha, Pitta, Ivan da Rocha, Rêgo, Moacyr Jesus Barreto de Melo, Alves, Luiz Carlos, Pitta, Maira Galdino da Rocha
Published in Revista do Instituto de Medicina Tropical de São Paulo (01.01.2017)
Published in Revista do Instituto de Medicina Tropical de São Paulo (01.01.2017)
Get full text
Journal Article
Medicinal chemistry of antischistosomal drugs: Praziquantel and oxamniquine
da Silva, Vinícius Barros Ribeiro, Campos, Bruna Rafaella Koresch Leiva, de Oliveira, Jamerson Ferreira, Decout, Jean-Luc, do Carmo Alves de Lima, Maria
Published in Bioorganic & medicinal chemistry (01.07.2017)
Published in Bioorganic & medicinal chemistry (01.07.2017)
Get full text
Journal Article
Novel indole-thiazole and indole-thiazolidinone derivatives as DNA groove binders
Alves, Josival Emanuel Ferreira, de Oliveira, Jamerson Ferreira, de Lima Souza, Tulio Ricardo Couto, de Moura, Ricardo Olímpio, de Carvalho Júnior, Luiz Bezerra, Alves de Lima, Maria do Carmo, de Almeida, Sinara Mônica Vitalino
Published in International journal of biological macromolecules (15.02.2021)
Published in International journal of biological macromolecules (15.02.2021)
Get full text
Journal Article
Synthesis, DNA and protein interactions and human topoisomerase inhibition of novel Spiroacridine derivatives
Gouveia, Rawny Galdino, Ribeiro, Amélia Galdino, Segundo, Miguel Ângelo Santos Pinheiro, de Oliveira, Jamerson Ferreira, de Lima, Maria do Carmo Alves, de Lima Souza, Túlio Ricardo Couto, de Almeida, Sinara Mônica Vitalino, de Moura, Ricardo Olímpio
Published in Bioorganic & medicinal chemistry (01.12.2018)
Published in Bioorganic & medicinal chemistry (01.12.2018)
Get full text
Journal Article
Thiosemicarbazones and 4-thiazolidinones indole-based derivatives: Synthesis, evaluation of antiproliferative activity, cell death mechanisms and topoisomerase inhibition assay
de Oliveira, Jamerson Ferreira, Lima, Talitha Santos, Vendramini-Costa, Débora Barbosa, de Lacerda Pedrosa, Sybelle Christianne Batista, Lafayette, Elizabeth Almeida, da Silva, Rosali Maria Ferreira, de Almeida, Sinara Monica Vitalino, de Moura, Ricardo Olímpio, Ruiz, Ana Lúcia Tasca Gois, de Carvalho, João Ernesto, de Lima, Maria do Carmo Alves
Published in European journal of medicinal chemistry (18.08.2017)
Published in European journal of medicinal chemistry (18.08.2017)
Get full text
Journal Article
COVID-19 therapy: What weapons do we bring into battle?
de Almeida, Sinara Mônica Vitalino, Santos Soares, José Cleberson, dos Santos, Keriolaine Lima, Alves, Josival Emanuel Ferreira, Ribeiro, Amélia Galdino, Jacob, Íris Trindade Tenório, da Silva Ferreira, Cindy Juliane, dos Santos, Jéssica Celerino, de Oliveira, Jamerson Ferreira, de Carvalho Junior, Luiz Bezerra, de Lima, Maria do Carmo Alves
Published in Bioorganic & medicinal chemistry (01.12.2020)
Published in Bioorganic & medicinal chemistry (01.12.2020)
Get full text
Journal Article
Synthesis of thiophene-thiosemicarbazone derivatives and evaluation of their in vitro and in vivo antitumor activities
de Oliveira, Jamerson Ferreira, da Silva, Anekécia Lauro, Vendramini-Costa, Débora Barbosa, da Cruz Amorim, Cezar Augusto, Campos, Júlia Furtado, Ribeiro, Amélia Galdino, Olímpio de Moura, Ricardo, Neves, Jorge Luiz, Ruiz, Ana Lúcia Tasca Gois, Ernesto de Carvalho, João, Alves de Lima, Maria do Carmo
Published in European journal of medicinal chemistry (02.11.2015)
Published in European journal of medicinal chemistry (02.11.2015)
Get full text
Journal Article
Study of nitrogen heterocycles as DNA/HSA binder, topoisomerase inhibitors and toxicological safety
Dos Santos, Jéssica Celerino, Alves, Josival Emanuel Ferreira, de Azevedo, Rafael David Souto, de Lima, Maksuelly Libanio, de Oliveira Silva, Maria Regina, da Silva, Josefa Gerlane, da Silva, Jamire Muriel, de Carvalho Correia, Ana Carolina, do Carmo Alves de Lima, Maria, de Oliveira, Jamerson Ferreira, de Moura, Ricardo Olímpio, de Almeida, Sinara Mônica Vitalino
Published in International journal of biological macromolecules (01.01.2024)
Published in International journal of biological macromolecules (01.01.2024)
Get full text
Journal Article
Synthesis, cytotoxicity and antifungal activity of 5-nitro-thiophene-thiosemicarbazones derivatives
de Araújo Neto, Luiz Nascimento, do Carmo Alves de Lima, Maria, de Oliveira, Jamerson Ferreira, de Souza, Edson Rubhens, Buonafina, Maria Daniela Silva, Vitor Anjos, Mayara Nunes, Brayner, Fábio André, Alves, Luiz Carlos, Neves, Rejane Pereira, Mendonça-Junior, Francisco Jaime Bezerra
Published in Chemico-biological interactions (25.06.2017)
Published in Chemico-biological interactions (25.06.2017)
Get full text
Journal Article
Synthesis, in vitro schistosomicidal activity and ultrastructural alterations caused by thiosemicarbazones and thiazolidinones against juvenile and adult Schistosoma mansoni worms (Sambon, 1907)
Tavares da Rocha, Rubens Emanoel, de Almeida Júnior, Antônio Sérgio Alves, Júnior, Nairomberg Cavalcanti Portela, do Nascimento, Amanda Vasconcelos, Leite, Nayara Maria Siqueira, de Oliveira, Jamerson Ferreira, Alves de Lima, Maria do Carmo, Feitosa, Ana Paula Sampaio, Bezerra de Mélo, Maria Eliane, Brayner, Fábio André, Alves, Luiz Carlos
Published in Molecular and biochemical parasitology (01.11.2022)
Published in Molecular and biochemical parasitology (01.11.2022)
Get full text
Journal Article
DNA binding and Topoisomerase inhibition: How can these mechanisms be explored to design more specific anticancer agents?
de Almeida, Sinara Mônica Vitalino, Ribeiro, Amélia Galdino, de Lima Silva, Geilza Carla, Ferreira Alves, Josival Emanuel, Beltrão, Eduardo Isidoro Carneiro, de Oliveira, Jamerson Ferreira, de Carvalho, Luiz Bezerra, Alves de Lima, Maria do Carmo
Published in Biomedicine & pharmacotherapy (01.12.2017)
Published in Biomedicine & pharmacotherapy (01.12.2017)
Get full text
Journal Article
Synthesis of novel indole derivatives as promising DNA-binding agents and evaluation of antitumor and antitopoisomerase I activities
Lafayette, Elizabeth Almeida, de Almeida, Sinara Mônica Vitalino, Cavalcanti Santos, Renata Virginia, de Oliveira, Jamerson Ferreira, Amorim, Cezar Augusto da Cruz, da Silva, Rosali Maria Ferreira, Pitta, Maira Galdino da Rocha, Pitta, Ivan da Rocha, de Moura, Ricardo Olimpio, de Carvalho Júnior, Luiz Bezerra, de Melo Rêgo, Moacyr Jesus Barreto, de Lima, Maria do Carmo Alves
Published in European journal of medicinal chemistry (18.08.2017)
Published in European journal of medicinal chemistry (18.08.2017)
Get full text
Journal Article