Recent Developments in the Field of Tumor-Inhibiting Metal Complexes
Galanski, M S, Arion, V B, Jakupec, M A, Keppler, B K
Published in Current pharmaceutical design (01.10.2003)
Published in Current pharmaceutical design (01.10.2003)
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Multi-scale imaging of anticancer platinum() compounds in murine tumor and kidney
Legin, A. A, Theiner, S, Schintlmeister, A, Reipert, S, Heffeter, P, Jakupec, M. A, Mayr, J, Varbanov, H. P, Kowol, C. R, Galanski, M. S, Berger, W, Wagner, M, Keppler, B. K
Published in Chemical science (Cambridge) (01.01.2016)
Published in Chemical science (Cambridge) (01.01.2016)
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Improved reaction conditions for the synthesis of new NKP-1339 derivatives and preliminary investigations on their anticancer potential
Kuhn, P-S, Pichler, V, Roller, A, Hejl, M, Jakupec, M A, Kandioller, W, Keppler, B K
Published in Dalton transactions : an international journal of inorganic chemistry (14.01.2015)
Published in Dalton transactions : an international journal of inorganic chemistry (14.01.2015)
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Heterocyclic complexes of ruthenium(III) induce apoptosis in colorectal carcinoma cells
KAPITZA, S, PONGRATZ, M, JAKUPEC, M. A, HEFFETER, P, BERGER, W, LACKINGER, L, KEPPLER, B. K, MARIAN, B
Published in Journal of cancer research and clinical oncology (01.02.2005)
Published in Journal of cancer research and clinical oncology (01.02.2005)
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Multidrug-resistant cancer cells are preferential targets of the new antineoplastic lanthanum compound KP772 (FFC24)
Heffeter, P., Jakupec, M.A., Körner, W., Chiba, P., Pirker, C., Dornetshuber, R., Elbling, L., Sutterlüty, H., Micksche, M., Keppler, B.K., Berger, W.
Published in Biochemical pharmacology (15.06.2007)
Published in Biochemical pharmacology (15.06.2007)
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Tumour-inhibiting platinum complexes--state of the art and future perspectives
Jakupec, M A, Galanski, M, Keppler, B K
Published in Reviews of physiology, biochemistry and pharmacology (01.01.2003)
Published in Reviews of physiology, biochemistry and pharmacology (01.01.2003)
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Pharmacological properties of cerium compounds
Jakupec, M A, Unfried, P, Keppler, B K
Published in Reviews of physiology, biochemistry and pharmacology (01.01.2005)
Published in Reviews of physiology, biochemistry and pharmacology (01.01.2005)
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Intrinsic and Acquired Forms of Resistance against the Anticancer Ruthenium Compound KP1019 [Indazolium trans-[tetrachlorobis(1H-indazole)ruthenate (III)] (FFC14A)
Heffeter, P, Pongratz, M, Steiner, E, Chiba, P, Jakupec, M A, Elbling, L, Marian, B, Körner, W, Sevelda, F, Micksche, M, Keppler, B K, Berger, W
Published in The Journal of pharmacology and experimental therapeutics (01.01.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2005)
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KP1019 (FFC14A) from bench to bedside: preclinical and early clinical development--an overview
Jakupec, M A, Arion, V B, Kapitza, S, Reisner, E, Eichinger, A, Pongratz, M, Marian, B, Graf von Keyserlingk, N, Keppler, B K
Published in International journal of clinical pharmacology and therapeutics (01.12.2005)
Published in International journal of clinical pharmacology and therapeutics (01.12.2005)
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Early results from a phase I study on orally administered tris(8-quinolinolato)gallium(III) (FFC11, KP46) in patients with solid tumors--a CESAR study (Central European Society for Anticancer Drug Research--EWIV)
Hofheinz, R D, Dittrich, C, Jakupec, M A, Drescher, A, Jaehde, U, Gneist, M, Graf von Keyserlingk, N, Keppler, B K, Hochhaus, A
Published in International journal of clinical pharmacology and therapeutics (01.12.2005)
Published in International journal of clinical pharmacology and therapeutics (01.12.2005)
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Ribonucleotide reductase as one important target of [Tris(1,10-phenanthroline)lanthanum(III)] trithiocyanate (KP772)
Heffeter, P, Popovic-Bijelic, A, Saiko, P, Dornetshuber, R, Jungwirth, U, Voevodskaya, N, Biglino, D, Jakupec, M A, Elbling, L, Micksche, M, Szekeres, T, Keppler, B K, Gräslund, A, Berger, W
Published in Current cancer drug targets (01.08.2009)
Published in Current cancer drug targets (01.08.2009)
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Rational development of oxaliplatin analogues --synthesis and preliminary structure-activity relationships
Galanski, M, Habala, L, Nazarov, A A, Jakupec, M A, Yasemi, A, Slaby, S, Graf von Keyserlingk, N, Keppler, B K
Published in International journal of clinical pharmacology and therapeutics (01.12.2005)
Published in International journal of clinical pharmacology and therapeutics (01.12.2005)
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Improved reaction conditions for the synthesis of new NKP-1339 derivatives and preliminary investigations on their anticancer potentialElectronic supplementary information (ESI) available: 1H-NMR spectra, cyclovoltammograms, UV-vis data and concentration-effect curves of the synthesised compounds. CCDC 1006143-1006145. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c4dt01645a
Kuhn, P.-S, Pichler, V, Roller, A, Hejl, M, Jakupec, M. A, Kandioller, W, Keppler, B. K
Year of Publication 09.12.2014
Year of Publication 09.12.2014
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Journal Article
Redox behavior of tumor-inhibiting ruthenium(III) complexes and effects of physiological reductants on their binding to GMP
Schluga, Petra, Hartinger, Christian G, Egger, Alexander, Reisner, Erwin, Galanski, Markus, Jakupec, Michael A, Keppler, Bernhard K
Published in Dalton transactions : an international journal of inorganic chemistry (14.04.2006)
Published in Dalton transactions : an international journal of inorganic chemistry (14.04.2006)
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Gallium(III) and Iron(III) Complexes of α-N-Heterocyclic Thiosemicarbazones: Synthesis, Characterization, Cytotoxicity, and Interaction with Ribonucleotide Reductase
Kowol, Christian R, Berger, Roland, Eichinger, Rene, Roller, Alexander, Jakupec, Michael A, Schmidt, Peter P, Arion, Vladimir B, Keppler, Bernhard K
Published in Journal of medicinal chemistry (22.03.2007)
Published in Journal of medicinal chemistry (22.03.2007)
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Redox-Active Antineoplastic Ruthenium Complexes with Indazole: Correlation of in Vitro Potency and Reduction Potential
JAKUPEC, Michael A., REISNER, Erwin, EICHINGER, Anna, PONGRATZ, Martina, ARION, Vladimir B., GALANSKI, Markus, HARTINGER, Christian G., KEPPLER, Bernhard K.
Published in Journal of medicinal chemistry (21.04.2005)
Published in Journal of medicinal chemistry (21.04.2005)
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Journal Article
Gallium in cancer treatment
Jakupec, Michael A, Keppler, Bernhard K
Published in Current topics in medicinal chemistry (01.01.2004)
Published in Current topics in medicinal chemistry (01.01.2004)
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