Comparison of a novel potentiator of CFTR channel activity to ivacaftor in ameliorating mucostasis caused by cigarette smoke in primary human bronchial airway epithelial cells
Tanjala, Adrian Constantin, Jiang, Jia Xin, Eckford, Paul D. W, Ramjeesingh, Mohabir, Li, Canhui, Huan, Ling Jun, Langeveld, Gabrielle, Townsend, Claire, Paone, Daniel V, Busch-Petersen, Jakob, Pekhletski, Roman, Tang, LiPing, Raju, Vamsee, Rowe, Steven M, Bear, Christine E
Published in Respiratory research (10.07.2024)
Published in Respiratory research (10.07.2024)
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Comparison of N, N′-diarylsquaramides and N, N′-diarylureas as antagonists of the CXCR2 chemokine receptor
McCleland, Brent W., Davis, Roderick S., Palovich, Michael R., Widdowson, Katherine L., Werner, Michelle L., Burman, Miriam, Foley, James J., Schmidt, Dulcie B., Sarau, Henry M., Rogers, Martin, Salyers, Kevin L., Gorycki, Peter D., Roethke, Theresa J., Stelman, Gary J., Azzarano, Leonard M., Ward, Keith W., Busch-Petersen, Jakob
Published in Bioorganic & medicinal chemistry letters (15.03.2007)
Published in Bioorganic & medicinal chemistry letters (15.03.2007)
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Journal Article
Comparison of a novel potentiator of CFTR channel activity to ivacaftor in ameliorating mucostasis caused by cigarette smoke in primary human bronchial airway epithelial cells
Tanjala, Adrian Constantin, Jiang, Jia Xin, Eckford, Paul D W, Ramjeesingh, Mohabir, Li, Canhui, Huan, Ling Jun, Langeveld, Gabrielle, Townsend, Claire, Paone, Daniel V, Busch-Petersen, Jakob, Pekhletski, Roman, Tang, LiPing, Raju, Vamsee, Rowe, Steven M, Bear, Christine E
Published in bioRxiv (04.03.2024)
Published in bioRxiv (04.03.2024)
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Journal Article
Anti‐tumor Promoting Activity of Canventol and Its Synthetic Analogs through Inhibition of Protein Isoprenylation
Komori, Atsumasa, Okabe, Sachiko, Suganuma, Masami, Kerr, Michael A., Busch‐Petersen, Jakob, Oh, Lynette M., Zhuo, Jincong, Kamali Kannangara, G. S., Zou, Xianglong, Tius, Marcus A., Fujiki, Hirota
Published in Cancer science (01.09.1996)
Published in Cancer science (01.09.1996)
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Journal Article
Danirixin: A Reversible and Selective Antagonist of the CXC Chemokine Receptor 2
Busch-Petersen, Jakob, Carpenter, Donald C, Burman, Miriam, Foley, James, Hunsberger, Gerald E, Kilian, David J, Salmon, Michael, Mayer, Ruth J, Yonchuk, John G, Tal-Singer, Ruth
Published in The Journal of pharmacology and experimental therapeutics (01.08.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2017)
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Journal Article
Inhibitors of cathepsin C (dipeptidyl peptidase I)
Laine, Dramane I, Busch-Petersen, Jakob
Published in Expert opinion on therapeutic patents (01.04.2010)
Published in Expert opinion on therapeutic patents (01.04.2010)
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Journal Article
3,5-Disubstituted-indole-7-carboxamides as IKKβ Inhibitors: Optimization of Oral Activity via the C3 Substituent
Kerns, Jeffrey K, Busch-Petersen, Jakob, Fu, Wei, Boehm, Jeffrey C, Nie, Hong, Muratore, Michael, Bullion, Ann, Lin, Guoliang, Li, Huijie, Davis, Roderick, Lin, Xichen, Lakdawala, Ami S, Cousins, Rick, Field, Rita, Payne, Jeremy, Miller, David D, Bamborough, Paul, Christopher, John A, Baldwin, Ian, Osborn, Ruth R, Yonchuk, John, Webb, Edward, Rumsey, William L
Published in ACS medicinal chemistry letters (13.12.2018)
Published in ACS medicinal chemistry letters (13.12.2018)
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Journal Article
Efficient and Scalable Synthesis of 3,5,7-Trisubstituted 1H-Indazoles as Potent IKK2 Inhibitors
Lin, Xichen, Busch-Petersen, Jakob, Deng, Jianghe, Edwards, Christine, Zhang, Zhaoguo, Kerns, Jeffrey K.
Published in Synlett (16.12.2008)
Published in Synlett (16.12.2008)
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Journal Article
Camphor sulfonamide derivatives as novel, potent and selective CXCR3 antagonists
Wang, Yonghui, Busch-Petersen, Jakob, Wang, Feng, Kiesow, Terence J., Graybill, Todd L., Jin, Jian, Yang, Zheng, Foley, James J., Hunsberger, Gerald E., Schmidt, Dulcie B., Sarau, Henry M., Capper-Spudich, Elizabeth A., Wu, Zining, Fisher, Laura S., McQueney, Michael S., Rivero, Ralph A., Widdowson, Katherine L.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Journal Article
Tyrosine urea muscarinic acetylcholine receptor antagonists: Achiral quaternary ammonium groups
Jin, Qi, Davis, Roderick S., Bullion, Ann M., Jin, Jian, Wang, Yonghui, Widdowson, Katherine L., Palovich, Michael R., Foley, James J., Schmidt, Dulcie B., Buckley, Peter T., Webb, Edward F., Salmon, Michael, Belmonte, Kristen E., Sarau, Henry M., Busch-Petersen, Jakob
Published in Bioorganic & medicinal chemistry letters (01.12.2012)
Published in Bioorganic & medicinal chemistry letters (01.12.2012)
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Journal Article
Design, synthesis and structure–activity relationship of N-substituted tropane muscarinic acetylcholine receptor antagonists
Lainé, Dramane I., Yan, Hongxing, Xie, Haibo, Davis, Roderick S., Dufour, Jeremy, Widdowson, Katherine L., Palovich, Michael R., Wan, Zehong, Foley, James J., Schmidt, Dulcie B., Hunsberger, Gerald E., Burman, Miriam, Bacon, Alicia M., Webb, Edward F., Luttmann, Mark A., Salmon, Michael, Sarau, Henry M., Umbrecht, Sandra T., Landis, Philip S., Peck, Brian J., Busch-Petersen, Jakob
Published in Bioorganic & medicinal chemistry letters (01.05.2012)
Published in Bioorganic & medicinal chemistry letters (01.05.2012)
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Journal Article
Design, Synthesis, and Structure−Activity Relationship of Tropane Muscarinic Acetylcholine Receptor Antagonists
Lainé, Dramane I, Wan, Zehong, Yan, Hongxing, Zhu, Chongjie, Xie, Haibo, Fu, Wei, Busch-Petersen, Jakob, Neipp, Christopher, Davis, Roderick, Widdowson, Katherine L, Blaney, Frank E, Foley, James, Bacon, Alicia M, Webb, Edward F, Luttmann, Mark A, Burman, Miriam, Sarau, Henry M, Salmon, Michael, Palovich, Michael R, Belmonte, Kristen
Published in Journal of medicinal chemistry (27.08.2009)
Published in Journal of medicinal chemistry (27.08.2009)
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Journal Article
3-Arylamino-2H-1,2,4-benzothiadiazin-5-ol 1,1-dioxides as novel and selective CXCR2 antagonists
Wang, Yonghui, Busch-Petersen, Jakob, Wang, Feng, Ma, Lanping, Fu, Wei, Kerns, Jeffrey K, Jin, Jian, Palovich, Michael R, Shen, Jing-Kang, Burman, Miriam, Foley, James J, Schmidt, Dulcie B, Hunsberger, Gerald E, Sarau, Henry M, Widdowson, Katherine L
Published in Bioorganic & medicinal chemistry letters (15.07.2007)
Published in Bioorganic & medicinal chemistry letters (15.07.2007)
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