Influence of steric parameters on the synthesis of tetramates from alpha-amino-beta-alkoxy-esters and Ph3PCCO
Loke, Inga, Park, Natja, Kempf, Karl, Jagusch, Carsten, Schobert, Rainer, Laschat, Sabine
Published in Tetrahedron (14.01.2012)
Published in Tetrahedron (14.01.2012)
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Synthesis, biological evaluation and molecular modelling studies of methyleneimidazole substituted biaryls as inhibitors of human 17α-hydroxylase-17,20-lyase (CYP17). Part I: Heterocyclic modifications of the core structure
Jagusch, Carsten, Negri, Matthias, Hille, Ulrike E., Hu, Qingzhong, Bartels, Marc, Jahn-Hoffmann, Kerstin, Mendieta, Mariano A.E. Pinto-Bazurco, Rodenwaldt, Barbara, Müller-Vieira, Ursula, Schmidt, Dirk, Lauterbach, Thomas, Recanatini, Maurizio, Cavalli, Andrea, Hartmann, Rolf W.
Published in Bioorganic & medicinal chemistry (15.02.2008)
Published in Bioorganic & medicinal chemistry (15.02.2008)
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Journal Article
Synthesis, Biological Evaluation, and Molecular Modeling of Abiraterone Analogues: Novel CYP17 Inhibitors for the Treatment of Prostate Cancer
Pinto-Bazurco Mendieta, Mariano A. E, Negri, Matthias, Jagusch, Carsten, Müller-Vieira, Ursula, Lauterbach, Thomas, Hartmann, Rolf W
Published in Journal of medicinal chemistry (28.08.2008)
Published in Journal of medicinal chemistry (28.08.2008)
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Replacement of Imidazolyl by Pyridyl in Biphenylmethylenes Results in Selective CYP17 and Dual CYP17/CYP11B1 Inhibitors for the Treatment of Prostate Cancer
Hu, Qingzhong, Jagusch, Carsten, Hille, Ulrike E, Haupenthal, Jörg, Hartmann, Rolf W
Published in Journal of medicinal chemistry (12.08.2010)
Published in Journal of medicinal chemistry (12.08.2010)
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2S3S- 7--2-4--3-1--1H-124--5--4--1234--5- COFORMER SALTS OF 2S3S-METHYL 7-FLUORO-2-4-FLUOROPHENYL-3-1-METHYL-1H-124-TRIAZOL-5-YL-4-OXO-1234-TETRAHYDROQUINOLINE-5-CARBOXYLATE AND METHODS OF PREPARING THEM
CAMPBELL COLM, HERZ CHRISTIAN KLAUS, HENDERSON MARK, JAGUSCH CARSTEN, BAUER NICO, BONNAUD THIERRY, LAMBERT OLIVIER
Year of Publication 07.04.2017
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Year of Publication 07.04.2017
Patent
Synthesis, biological evaluation and molecular modelling studies of novel ACD- and ABD-ring steroidomimetics as inhibitors of CYP17
Pinto-Bazurco Mendieta, Mariano A.E., Negri, Matthias, Jagusch, Carsten, Hille, Ulrike E., Müller-Vieira, Ursula, Schmidt, Dirk, Hansen, Klaus, Hartmann, Rolf W.
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
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CYP17 Inhibitors. Annulations of Additional Rings in Methylene Imidazole Substituted Biphenyls: Synthesis, Biological Evaluation and Molecular Modelling
Pinto-Bazurco Mendieta, Mariano A. E., Negri, Matthias, Hu, Qingzhong, Hille, Ulrike E., Jagusch, Carsten, Jahn-Hoffmann, Kerstin, Müller-Vieira, Ursula, Schmidt, Dirk, Lauterbach, Thomas, Hartmann, Rolf W.
Published in Archiv der Pharmazie (Weinheim) (01.10.2008)
Published in Archiv der Pharmazie (Weinheim) (01.10.2008)
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