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Published in Journal of the American Society of Nephrology (01.02.2014)
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The novel chemokine receptor CXCR7 regulates trans-endothelial migration of cancer cells
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Elucidation of CXCR7-Mediated Signaling Events and Inhibition of CXCR4-Mediated Tumor Cell Transendothelial Migration by CXCR7 Ligands
Zabel, Brian A, Wang, Yu, Lewen, Susanna, Berahovich, Robert D, Penfold, Mark E. T, Zhang, Penglie, Powers, Jay, Summers, Bretton C, Miao, Zhenhua, Zhao, Bin, Jalili, Ali, Janowska-Wieczorek, Anna, Jaen, Juan C, Schall, Thomas J
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CCR2 antagonist CCX140-B provides renal and glycemic benefits in diabetic transgenic human CCR2 knockin mice
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Published in American journal of physiology. Renal physiology (01.11.2013)
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Characterization of CCX282-B, an orally bioavailable antagonist of the CCR9 chemokine receptor, for treatment of inflammatory bowel disease
Walters, Matthew J, Wang, Yu, Lai, Nu, Baumgart, Trageen, Zhao, Bin N, Dairaghi, Daniel J, Bekker, Pirow, Ertl, Linda S, Penfold, Mark E T, Jaen, Juan C, Keshav, Satish, Wendt, Emily, Pennell, Andrew, Ungashe, Solomon, Wei, Zheng, Wright, J J Kim, Schall, Thomas J
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Synthesis and optimization of substituted furo[2,3-d]-pyrimidin-4-amines and 7H-pyrrolo[2,3-d]pyrimidin-4-amines as ACK1 inhibitors
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Published in Bioorganic & medicinal chemistry letters (01.10.2012)
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CCR1 blockade reduces tumor burden and osteolysis in vivo in a mouse model of myeloma bone disease
Dairaghi, Daniel J., Oyajobi, Babatunde O., Gupta, Anjana, McCluskey, Brandon, Miao, Shichang, Powers, Jay P., Seitz, Lisa C., Wang, Yu, Zeng, Yibin, Zhang, Penglie, Schall, Thomas J., Jaen, Juan C.
Published in Blood (16.08.2012)
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Experimental evidence for the use of CCR2 antagonists in the treatment of type 2 diabetes
Sullivan, Timothy J, Miao, Zhenhua, Zhao, Bin N, Ertl, Linda S, Wang, Yu, Krasinski, Antoni, Walters, Matthew J, Powers, Jay P, Dairaghi, Daniel J, Baumgart, Trageen, Seitz, Lisa C, Berahovich, Robert D, Schall, Thomas J, Jaen, Juan C
Published in Metabolism, clinical and experimental (01.11.2013)
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Tissue proteases convert CCL23 into potent monocyte chemoattractants in patients with chronic rhinosinusitis
Poposki, Julie A., MS, Keswani, Anjeni, MD, Kim, Julie K., MD, Klingler, Aiko I., PhD, Suh, Lydia A., BS, Norton, James, MS, Carter, Roderick G., BS, Peters, Anju T., MD, Hulse, Kathryn E., PhD, Grammer, Leslie C., MD, Tan, Bruce K., MD, Conley, David B., MD, Jaen, Juan C., PhD, Schall, Thomas J., PhD, Kern, Robert C., MD, Kato, Atsushi, PhD
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CCR9 Antagonists in the Treatment of Ulcerative Colitis
Sullivan, Timothy J., Jaen, Juan C., Schall, Thomas J., Powers, Jay P., Punna, Sreenivas, Charvat, Trevor T., Ertl, Linda S., Berahovich, Robert D., Walters, Matthew J., Ebsworth, Karen, Bekker, Pirow, Campbell, James J.
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CXCR7 protein is not expressed on human or mouse leukocytes
Berahovich, Robert D, Zabel, Brian A, Penfold, Mark E T, Lewén, Susanna, Wang, Yu, Miao, Zhenhua, Gan, Lin, Pereda, Jaime, Dias, Jessica, Slukvin, Igor I, McGrath, Kathleen E, Jaen, Juan C, Schall, Thomas J
Published in The Journal of immunology (1950) (01.11.2010)
Published in The Journal of immunology (1950) (01.11.2010)
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CXCR7 protein expression correlates with elevated mmp-3 secretion in breast cancer cells
ZABEL, BRIAN A, MIAO, ZHENHUA, LAI, NU L, WANG, YU, LEWÉN, SUSANNA, BERAHOVICH, ROBERT D, JAÉN, JUAN C, SCHALL, THOMAS J
Published in Oncology letters (01.09.2010)
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SAR and Mode of Action of Novel Non-Nucleoside Inhibitors of Hepatitis C NS5b RNA Polymerase
Powers, Jay P, Piper, Derek E, Li, Yang, Mayorga, Veronica, Anzola, John, Chen, James M, Jaen, Juan C, Lee, Gary, Liu, Jinqian, Peterson, M. Greg, Tonn, George R, Ye, Qiuping, Walker, Nigel P. C, Wang, Zhulun
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Published in Journal of medicinal chemistry (09.02.2006)
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Discovery of potent, selective, and orally bioavailable inhibitors of interleukin-1 receptor-associate kinase-4
Wang, Zhulun, Sun, Daqing, Johnstone, Sheree, Cao, Zhaodan, Gao, Xiong, Jaen, Juan C., Liu, Jingqian, Lively, Sarah, Miao, Shichang, Sudom, Athena, Tomooka, Craig, Walker, Nigel P.C., Wright, Matthew, Yan, Xuelei, Ye, Qiuping, Powers, Jay P.
Published in Bioorganic & medicinal chemistry letters (01.12.2015)
Published in Bioorganic & medicinal chemistry letters (01.12.2015)
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ITOC2 – 011. Identification of second-generation potent and selective inhibitors of indoleamine-2,3-dioxygenase-1 (IDO1) for the treatment of cancer
Juan, Jaen C, Pia, Bjorck, Jordan, Fridman S, Lisa, Marshall, Jan, Melom, Rajkumar, Noubade, Max, Osipov, Matthew, Walters J, Mikhail, Zibinsky, Jay, Powers P
Published in European journal of cancer (1990) (01.03.2015)
Published in European journal of cancer (1990) (01.03.2015)
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Discovery and optimization of benzenesulfonanilide derivatives as a novel class of 11β-HSD1 inhibitors
Rew, Yosup, DeGraffenreid, Michael, He, Xiao, Jaen, Juan C., McMinn, Dustin L., Sun, Daqing, Tu, Hua, Ursu, Stefania, Powers, Jay P.
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
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Discovery of Novel, Potent Benzamide Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1) Exhibiting Oral Activity in an Enzyme Inhibition ex Vivo Model
Julian, Lisa D, Wang, Zhulun, Bostick, Tracy, Caille, Seb, Choi, Rebekah, DeGraffenreid, Michael, Di, Yongmei, He, Xiao, Hungate, Randall W, Jaen, Juan C, Liu, Jinsong, Monshouwer, Mario, McMinn, Dustin, Rew, Yosup, Sudom, Athena, Sun, Daqing, Tu, Hua, Ursu, Stefania, Walker, Nigel, Yan, Xuelei, Ye, Qiuping, Powers, Jay P
Published in Journal of medicinal chemistry (10.07.2008)
Published in Journal of medicinal chemistry (10.07.2008)
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Distinctive molecular inhibition mechanisms for selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1
Tu, Hua, Powers, Jay P., Liu, Jinsong, Ursu, Stefania, Sudom, Athena, Yan, Xuelei, Xu, Haoda, Meininger, David, DeGraffenreid, Michael, He, Xiao, Jaen, Juan C., Sun, Daqing, Labelle, Marc, Yamamoto, Hiroshi, Shan, Bei, Walker, Nigel P.C., Wang, Zhulun
Published in Bioorganic & medicinal chemistry (01.10.2008)
Published in Bioorganic & medicinal chemistry (01.10.2008)
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