Selective estrogen receptor degraders with novel structural motifs induce regression in a tamoxifen-resistant breast cancer xenograft
Govek, Steven P., Bonnefous, Celine, Julien, Jackaline D., Nagasawa, Johnny Y., Kahraman, Mehmet, Lai, Andiliy G., Douglas, Karensa L., Aparicio, Anna M., Darimont, Beatrice D., Grillot, Katherine L., Joseph, James D., Kaufman, Joshua A., Lee, Kyoung-Jin, Lu, Nhin, Moon, Michael J., Prudente, Rene Y., Sensintaffar, John, Rix, Peter J., Hager, Jeffrey H., Smith, Nicholas D.
Published in Bioorganic & medicinal chemistry letters (01.02.2019)
Published in Bioorganic & medicinal chemistry letters (01.02.2019)
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Journal Article
ESTROGEN RECEPTOR MODULATOR AND USE THEREOF
GOVEK STEVEN P, JOHNNY Y NAGASAWA, CELINE BONNEFOUS, NICHOLAS D SMITH, MARK R HERBERT, ANDILIY G LAI, MEHMET KAHRAMAN, JACKALINE D JULIEN, KARENSA L DOUGLAS
Year of Publication 01.09.2016
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Year of Publication 01.09.2016
Patent
The selective estrogen receptor downregulator GDC-0810 is efficacious in diverse models of ER+ breast cancer
Joseph, James D, Darimont, Beatrice, Zhou, Wei, Arrazate, Alfonso, Young, Amy, Ingalla, Ellen, Walter, Kimberly, Blake, Robert A, Nonomiya, Jim, Guan, Zhengyu, Kategaya, Lorna, Govek, Steven P, Lai, Andiliy G, Kahraman, Mehmet, Brigham, Dan, Sensintaffar, John, Lu, Nhin, Shao, Gang, Qian, Jing, Grillot, Kate, Moon, Michael, Prudente, Rene, Bischoff, Eric, Lee, Kyoung-Jin, Bonnefous, Celine, Douglas, Karensa L, Julien, Jackaline D, Nagasawa, Johnny Y, Aparicio, Anna, Kaufman, Josh, Haley, Benjamin, Giltnane, Jennifer M, Wertz, Ingrid E, Lackner, Mark R, Nannini, Michelle A, Sampath, Deepak, Schwarz, Luis, Manning, Henry Charles, Tantawy, Mohammed Noor, Arteaga, Carlos L, Heyman, Richard A, Rix, Peter J, Friedman, Lori, Smith, Nicholas D, Metcalfe, Ciara, Hager, Jeffrey H
Published in eLife (13.07.2016)
Published in eLife (13.07.2016)
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Journal Article
Estrogen receptor modulators and uses thereof
Julien, Jackaline, D, Govek, Steven, P, Bonnefous, Celine, Douglas, Karensa L, Lai, Andiliy, G, Smith, Nicholas, D, Nagasawa, Johnny, Y, Kahraman, Mehmet, Herbert, Mark R
Year of Publication 15.11.2023
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Year of Publication 15.11.2023
Patent