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Biochemical characterization of tirabrutinib and other irreversible inhibitors of Bruton's tyrosine kinase reveals differences in on - and off - target inhibition
Liclican, Albert, Serafini, Loredana, Xing, Weimei, Czerwieniec, Gregg, Steiner, Bart, Wang, Ting, Brendza, Katherine M., Lutz, Justin D., Keegan, Kathleen S., Ray, Adrian S., Schultz, Brian E., Sakowicz, Roman, Feng, Joy Y.
Published in Biochimica et biophysica acta. General subjects (01.04.2020)
Published in Biochimica et biophysica acta. General subjects (01.04.2020)
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Green tea ingestion greatly reduces plasma concentrations of nadolol in healthy subjects
Misaka, S, Yatabe, J, Müller, F, Takano, K, Kawabe, K, Glaeser, H, Yatabe, M S, Onoue, S, Werba, J P, Watanabe, H, Yamada, S, Fromm, M F, Kimura, J
Published in Clinical pharmacology and therapeutics (01.04.2014)
Published in Clinical pharmacology and therapeutics (01.04.2014)
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Clinical Outcomes and Plasma Concentrations of Baloxavir Marboxil and Favipiravir in COVID-19 Patients: An Exploratory Randomized, Controlled Trial
Lou, Yan, Liu, Lin, Yao, Hangping, Hu, Xingjiang, Su, Junwei, Xu, Kaijin, Luo, Rui, Yang, Xi, He, Lingjuan, Lu, Xiaoyang, Zhao, Qingwei, Liang, Tingbo, Qiu, Yunqing
Published in European journal of pharmaceutical sciences (01.02.2021)
Published in European journal of pharmaceutical sciences (01.02.2021)
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Tucatinib Inhibits Renal Transporters OCT2 and MATE Without Impacting Renal Function in Healthy Subjects
Topletz‐Erickson, Ariel R., Lee, Anthony J., Mayor, JoAl G., Rustia, Evelyn L., Abdulrasool, Layth I., Wise, Amanda L., Dailey, Ben, DeChenne, Sharon, Walker, Luke N., Alley, Stephen C., Endres, Christopher J.
Published in Journal of clinical pharmacology (01.04.2021)
Published in Journal of clinical pharmacology (01.04.2021)
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Phase I Clinical Trial Results of Auranofin, a Novel Antiparasitic Agent
Capparelli, Edmund V., Bricker-Ford, Robin, Rogers, M. John, McKerrow, James H., Reed, Sharon L.
Published in Antimicrobial agents and chemotherapy (01.01.2017)
Published in Antimicrobial agents and chemotherapy (01.01.2017)
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Characterisation of the potential of β-lactoglobulin and α-lactalbumin as sources of bioactive peptides affecting incretin function: In silico and in vitro comparative studies
Tulipano, Giovanni, Faggi, Lara, Nardone, Alessandro, Cocchi, Daniela, Caroli, Anna Maria
Published in International dairy journal (01.09.2015)
Published in International dairy journal (01.09.2015)
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Phenotypic heterogeneity is a selected trait in natural yeast populations subject to environmental stress
Holland, Sara L, Reader, Tom, Dyer, Paul S, Avery, Simon V
Published in Environmental microbiology (01.06.2014)
Published in Environmental microbiology (01.06.2014)
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Rhamnetin induces sensitization of hepatocellular carcinoma cells to a small molecular kinase inhibitor or chemotherapeutic agents
Jia, Hui, Yang, Qian, Wang, Tao, Cao, Yu, Jiang, Qi-yu, Ma, Hong-da, Sun, Hui-wei, Hou, Ming-xiao, Yang, Yong-ping, Feng, Fan
Published in Biochimica et biophysica acta (01.07.2016)
Published in Biochimica et biophysica acta (01.07.2016)
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BMY 7378, a selective α 1D -adrenoceptor antagonist, is a new angiotensin converting enzyme inhibitor: In silico, in vitro and in vivo approach
Rodríguez, Jessica E, Andrade-Jorge, Erik, Barquet-Nieto, Alina, Estrada-Soto, Samuel E, Gallardo-Ortíz, Itzell A, Villalobos-Molina, Rafael
Published in Biochimica et biophysica acta. General subjects (01.01.2025)
Published in Biochimica et biophysica acta. General subjects (01.01.2025)
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The chemotherapeutic potential of PEG-b-PLGA copolymer micelles that combine chloroquine as autophagy inhibitor and docetaxel as an anti-cancer drug
Zhang, Xudong, Zeng, Xiaowei, Liang, Xin, Yang, Ying, Li, Xiaoming, Chen, Hongbo, Huang, Laiqiang, Mei, Lin, Feng, Si-Shen
Published in Biomaterials (01.11.2014)
Published in Biomaterials (01.11.2014)
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Chemical genetics strategy identifies an HCV NS5A inhibitor with a potent clinical effect
Gao, Min, Nettles, Richard E., Belema, Makonen, Snyder, Lawrence B., Nguyen, Van N., Fridell, Robert A., Serrano-Wu, Michael H., Langley, David R., Sun, Jin-Hua, O’Boyle II, Donald R., Lemm, Julie A., Wang, Chunfu, Knipe, Jay O., Chien, Caly, Colonno, Richard J., Grasela, Dennis M., Meanwell, Nicholas A., Hamann, Lawrence G.
Published in Nature (London) (06.05.2010)
Published in Nature (London) (06.05.2010)
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Pharmacodynamics, Safety, and Pharmacokinetics of BMS-663068, an Oral HIV-1 Attachment Inhibitor in HIV-1-Infected Subjects
Nettles, Richard E., Schürmann, Dirk, Zhu, Li, Stonier, Michele, Huang, Shu-Pang, Chang, Ih, Chien, Caly, Krystal, Mark, Wind-Rotolo, Megan, Ray, Neelanjana, Hanna, George J., Bertz, Richard, Grasela, Dennis
Published in The Journal of infectious diseases (01.10.2012)
Published in The Journal of infectious diseases (01.10.2012)
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Mitochondrial dysfunction, autophagy stimulation and non-apoptotic cell death caused by nitric oxide-inducing Pt-coated Au nanoparticle in human lung carcinoma cells
Akhtar, Mohd Javed, Ahamed, Maqusood, Alhadlaq, Hisham A., Kumar, Sudhir, Alrokayan, Salman A.
Published in Biochimica et biophysica acta. General subjects (01.01.2020)
Published in Biochimica et biophysica acta. General subjects (01.01.2020)
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Gold nanorod embedded reduction responsive block copolymer micelle-triggered drug delivery combined with photothermal ablation for targeted cancer therapy
Parida, Sheetal, Maiti, Chiranjit, Rajesh, Y, Dey, Kaushik K, Pal, Ipsita, Parekh, Aditya, Patra, Rusha, Dhara, Dibakar, Dutta, Pranab Kumar, Mandal, Mahitosh
Published in Biochimica et biophysica acta. General subjects (01.01.2017)
Published in Biochimica et biophysica acta. General subjects (01.01.2017)
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Eugenol disrupts Plasmodium falciparum intracellular development during the erythrocytic cycle and protects against cerebral malaria
Pontes, Kesley A.O., Silva, Leandro S., Santos, Edgleyson C., Pinheiro, Alessandro S., Teixeira, Douglas E., Peruchetti, Diogo B., Silva-Aguiar, Rodrigo P., Wendt, Camila H.C., Miranda, Kildare R., Coelho-de-Souza, Andrelina N., Leal-Cardoso, José Henrique, Caruso-Neves, Celso, Pinheiro, Ana Acacia S.
Published in Biochimica et biophysica acta. General subjects (01.03.2021)
Published in Biochimica et biophysica acta. General subjects (01.03.2021)
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Ebselen and analogs as inhibitors of Bacillus anthracis thioredoxin reductase and bactericidal antibacterials targeting Bacillus species, Staphylococcus aureus and Mycobacterium tuberculosis
Gustafsson, Tomas N., Osman, Harer, Werngren, Jim, Hoffner, Sven, Engman, Lars, Holmgren, Arne
Published in Biochimica et biophysica acta (01.06.2016)
Published in Biochimica et biophysica acta (01.06.2016)
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Detection of Weak Organic Anion–Transporting Polypeptide 1B Inhibition by Probenecid with Plasma-Based Coproporphyrin in Humans
Zhang, Yueping, Holenarsipur, Vinay K., Kandoussi, Hamza, Zeng, Jianing, Mariappan, T. Thanga, Sinz, Michael, Shen, Hong
Published in Drug metabolism and disposition (01.10.2020)
Published in Drug metabolism and disposition (01.10.2020)
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Relative resistance of HIV-1 founder viruses to control by interferon-alpha
Fenton-May, Angharad E, Dibben, Oliver, Emmerich, Tanja, Ding, Haitao, Pfafferott, Katja, Aasa-Chapman, Marlen M, Pellegrino, Pierre, Williams, Ian, Cohen, Myron S, Gao, Feng, Shaw, George M, Hahn, Beatrice H, Ochsenbauer, Christina, Kappes, John C, Borrow, Persephone
Published in Retrovirology (03.12.2013)
Published in Retrovirology (03.12.2013)
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