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Novel Synthesis of 3,4-Diarylisoxazole Analogues of Valdecoxib: Reversal Cyclooxygenase-2 Selectivity by Sulfonamide Group Removal
Di Nunno, Leonardo, Vitale, Paola, Scilimati, Antonio, Tacconelli, Stefania, Patrignani, Paola
Published in Journal of medicinal chemistry (23.09.2004)
Published in Journal of medicinal chemistry (23.09.2004)
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Therapeutic Amprenavir Concentrations in Cerebrospinal Fluid
Croteau, David, Letendre, Scott, Best, Brookie M., Rossi, Steven S., Ellis, Ronald J., Clifford, David B., Collier, Ann C., Gelman, Benjamin B., Marra, Christina M., McArthur, Justin, McCutchan, J. Allen, Morgello, Susan, Simpson, David M., Way, Lauren, Capparelli, Edmund, Grant, Igor
Published in Antimicrobial Agents and Chemotherapy (01.04.2012)
Published in Antimicrobial Agents and Chemotherapy (01.04.2012)
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Synthesis and evaluation of debromohymenialdisine-derived Chk2 inhibitors
Saleem, Rahman Shah Zaib, Lansdell, Theresa A., Tepe, Jetze J.
Published in Bioorganic & medicinal chemistry (15.02.2012)
Published in Bioorganic & medicinal chemistry (15.02.2012)
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Pharmacokinetics, pharmacodynamics and safety of CKD-519, a CETP inhibitor, in healthy subjects
Kim, Choon Ok, Oh, Eun Sil, Choi, Chungam, Kim, Yeonjoo, Lee, Sera, Kim, Semi, Park, Min Soo
Published in Drug design, development and therapy (01.01.2016)
Published in Drug design, development and therapy (01.01.2016)
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A High Level of Cyclooxygenase-2 Inhibitor Selectivity is Associated with a Reduced Interference of Platelet Cyclooxygenase-1 Inactivation by Aspirin
Ouellet, Marc, Riendeau, Denis, Percival, M. David
Published in Proceedings of the National Academy of Sciences - PNAS (04.12.2001)
Published in Proceedings of the National Academy of Sciences - PNAS (04.12.2001)
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Anti-Inflammatory Effect of Fluvastatin on IL-8 Production Induced by Pseudomonas aeruginosa and Aspergillus fumigatus Antigens in Cystic Fibrosis
Jouneau, Stéphane, Bonizec, Mélanie, Belleguic, Chantal, Desrues, Benoit, Brinchault, Graziella, Galaine, Jeanne, Gangneux, Jean-Pierre, Martin-Chouly, Corinne
Published in PloS one (03.08.2011)
Published in PloS one (03.08.2011)
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Ex vivo drug sensitivity profiles of Plasmodium falciparum field isolates from Cambodia and Thailand, 2005 to 2010, determined by a histidine-rich protein-2 assay
Tyner, Stuart D, Lon, Chanthap, Se, Youry, Bethell, Delia, Socheat, Doung, Noedl, Harald, Sea, Darapiseth, Satimai, Wichai, Schaecher, Kurt, Rutvisuttinunt, Wiriya, Fukuda, Mark M, Chaorattanakawee, Suwanna, Yingyuen, Kritsanai, Sundrakes, Siratchana, Chaichana, Panjaporn, Saingam, Piyaporn, Buathong, Nillawan, Sriwichai, Sabaithip, Chann, Soklyda, Timmermans, Ans, Saunders, David L, Walsh, Douglas S
Published in Malaria journal (13.06.2012)
Published in Malaria journal (13.06.2012)
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Developing a list of reference chemicals for testing alternatives to whole fish toxicity tests
Schirmer, Kristin, Tanneberger, Katrin, Kramer, Nynke I., Völker, Doris, Scholz, Stefan, Hafner, Christoph, Lee, Lucy E.J., Bols, Niels C., Hermens, Joop L.M.
Published in Aquatic toxicology (11.11.2008)
Published in Aquatic toxicology (11.11.2008)
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Specific, Irreversible Inactivation of the Epidermal Growth Factor Receptor and erbB2, by a New Class of Tyrosine Kinase Inhibitor
Fry, David W., Bridges, Alexander J., Denny, William A., Doherty, Annette, Greis, Kenneth D., Hicks, James L., Hook, Kenneth E., Keller, Paul R., Leopold, Wilbur R., Loo, Joseph A., McNamara, Dennis J., Nelson, James M., Sherwood, Veronika, Smaill, Jeff B., Trumpp-Kallmeyer, Susanne, Dobrusin, Ellen M.
Published in Proceedings of the National Academy of Sciences - PNAS (29.09.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (29.09.1998)
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Resistance Profile of the Human Immunodeficiency Virus Type 1 Reverse Transcriptase Inhibitor Abacavir (1592U89) after Monotherapy and Combination Therapy
Harrigan, P. Richard, Stone, Chris, Griffin, Phillip, Nájera, Isabel, Bloor, Stuart, Kemp, Sharon, Tisdale, Margaret, Larder, Brendan
Published in The Journal of infectious diseases (01.03.2000)
Published in The Journal of infectious diseases (01.03.2000)
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Identification of angiotensin I-converting enzyme inhibitory peptides derived from salmon muscle and their antihypertensive effect
Enari, H.(Nichiro Corp., Kawasaki, Kanagawa (Japan). Central Research Lab.), Takahashi, Y, Kawarasaki, M, Tada, M, Tatsuta, K
Published in Fisheries science (01.08.2008)
Published in Fisheries science (01.08.2008)
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Discovery of a novel proteasome inhibitor selective for cancer cells over non-transformed cells
Kazi, Aslamuzzaman, Lawrence, Harshani, Guida, Wayne C., McLaughlin, Mark L., Springett, Gregory M., Berndt, Norbert, Yip, Richard M., Sebti, Said M.
Published in Cell cycle (Georgetown, Tex.) (15.06.2009)
Published in Cell cycle (Georgetown, Tex.) (15.06.2009)
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A novel glycine transporter-1 (GlyT1) inhibitor, ASP2535 (4-[3-isopropyl-5-(6-phenyl-3-pyridyl)-4H-1,2,4-triazol-4-yl]-2,1,3-benzoxadiazole), improves cognition in animal models of cognitive impairment in schizophrenia and Alzheimer's disease
Harada, Katsuya, Nakato, Kazuhiro, Yarimizu, Junko, Yamazaki, Mayako, Morita, Masahiko, Takahashi, Shinji, Aota, Masaki, Saita, Kyoko, Doihara, Hitoshi, Sato, Yuichiro, Yamaji, Takayuki, Ni, Keni, Matsuoka, Nobuya
Published in European journal of pharmacology (15.06.2012)
Published in European journal of pharmacology (15.06.2012)
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Reversible, Time-Dependent Inhibition of CYP3A-Mediated Metabolism of Midazolam and Tacrolimus by Telaprevir in Human Liver Microsomes
Chapron, Brian, Risler, Linda, Phillips, Brian, Collins, Carol, Thummel, Kenneth, Shen, Danny
Published in Journal of pharmacy & pharmaceutical sciences (01.01.2015)
Published in Journal of pharmacy & pharmaceutical sciences (01.01.2015)
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Age and gender dependent heart rate circadian model development and performance verification on the proarrhythmic drug case study
Fijorek, Kamil, Patel, Nikunjkumar, Klima, Łukasz, Stolarz-Skrzypek, Katarzyna, Kawecka-Jaszcz, Kalina, Polak, Sebastian
Published in Theoretical biology and medical modelling (09.02.2013)
Published in Theoretical biology and medical modelling (09.02.2013)
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Purification and characterization of a galactose-specific lectin with mitogenic activity from pinto beans
Wong, Jack H., Wong, Clarence C.T., Ng, T.B.
Published in Biochimica et biophysica acta (01.05.2006)
Published in Biochimica et biophysica acta (01.05.2006)
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Antimalarial Activity of Tigecycline, a Novel Glycylcycline Antibiotic
Starzengruber, P., Thriemer, K., Haque, R., Khan, W. A., Fuehrer, H. P., Siedl, A., Hofecker, V., Ley, B., Wernsdorfer, W. H., Noedl, H.
Published in Antimicrobial Agents and Chemotherapy (01.09.2009)
Published in Antimicrobial Agents and Chemotherapy (01.09.2009)
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