5-MEMBERED HETEROARYLAMINOSULFONAMIDES FOR TREATING CONDITIONS MEDIATED BY DEFICIENT CFTR ACTIVITY
BALTZER, Sylvie, WIRE, William, MA, Nina, HARTUNG, Ryan, GAO, Zhongli, LIAO, Junkai, YEOMAN, Helen, NESTLER, Hans, Peter, HURLBUT, Gregory, MECHIN, Ingrid, THURAIRATNAM, Sukanthini, VIVET, Bertrand, FREED, Brian, MUNSON, Mark, SMRCINA, Martin, LEBRETON, Sylvain
Year of Publication 21.09.2022
Get full text
Year of Publication 21.09.2022
Patent
NOVEL HETEROARYL-UREA COMPOUNDS AS KV7.2 INHIBITORS
SMRCINA, MARTIN, LI, RONGHUA, NAGARAJAN, KARTHIGEYAN, GRAHAM, CHRISTOPHER JOHN, SAFAROVA, ALENA, GERLACH, AARON, CHAPMAN, MARK, MOWREY, DAVID, REDONDO PENA, ROGER LLUIS, DAVIDSON, JAMES, DAVIES, NICHOLAS GARETH MORSE, LEBRETON, SYLVAIN, NORCROSS, ROGER DAVID, MECHIN, INGRID, NAIR, ANIL, MA, NINA
Year of Publication 25.05.2023
Get full text
Year of Publication 25.05.2023
Patent
5-membered heteroarylaminosulfonamides for treating conditions mediated by deficient CFTR activity
BALTZER, Sylvie, NESTLER, Hans Peter, WIRE, William, MA, Nina, HARTUNG, Ryan, GAO, Zhongli, LIAO, Junkai, YEOMAN, Helen, HURLBUT, Gregory, MECHIN, Ingrid, THURAIRATNAM, Sukanthini, VIVET, Bertrand, FREED, Brian, MUNSON, Mark, SMRCINA, Martin, LEBRETON, Sylvain
Year of Publication 26.05.2022
Get full text
Year of Publication 26.05.2022
Patent
ARYLAMIDES AND METHODS OF USE THEREOF
NESTLER, Hans, MECHIN, Ingrid, SCHOLTE, Andrew, BOCK, William, VIVET, Bertrand, MUNSON, Mark, HARTUNG, Ryan, GAO, Zhongli, LIAO, Junkai, SMRCINA, Martin, LI, Ronghua, HURLBUT, Gregory
Year of Publication 10.06.2021
Get full text
Year of Publication 10.06.2021
Patent
CFTR-MODULATING ARYLAMIDES
NESTLER, Hans, KIM, Joseph, MA, Nina, HARTUNG, Ryan, GAO, Zhongli, LIAO, Junkai, LI, Ronghua, HURLBUT, Gregory, MECHIN, Ingrid, BOCK, William, MUNSON, Mark, SMRCINA, Martin, VIVET, Bertand
Year of Publication 10.06.2021
Get full text
Year of Publication 10.06.2021
Patent
5-MEMBERED HETEROARYLAMINOSULFONAMIDES FOR TREATING CONDITIONS MEDIATED BY DEFICIENT CFTR ACTIVITY
BALTZER, Sylvie, NESTLER, Hans, WIRE, William, MA, Nina, HARTUNG, Ryan, GAO, Zhongli, LIAO, Junkai, YEOMAN, Helen, HURLBUT, Gregory, MECHIN, Ingrid, THURAIRATNAM, Sukanthini, VIVET, Bertrand, FREED, Brian, MUNSON, Mark, SMRCINA, Martin, LEBRETON, Sylvain
Year of Publication 20.05.2021
Get full text
Year of Publication 20.05.2021
Patent
5-MEMBERED HETEROARYLAMINOSULFONAMIDES FOR TREATING CONDITIONS MEDIATED BY DEFICIENT CFTR ACTIVITY
VIVET, BERTRAND, GAO, ZHONGLI, SMRCINA, MARTIN, HARTUNG, RYAN, HURLBUT, GREGORY, BALTZER, SYLVIE, FREED, BRIAN, YEOMAN, HELEN, MUNSON, MARK, LEBRETON, SYLVAIN, THURAIRATNAM, SUKANTHINI, LIAO, JUNKAI, NESTLER, HANS PETER, MECHIN, INGRID, MA, NINA, WIRE, WILLIAM
Year of Publication 20.05.2021
Get full text
Year of Publication 20.05.2021
Patent
The ΔF508 CFTR defect: molecular mechanism of suppressor mutation V510D and the contribution of transmembrane helix unraveling
Simon, Kailene S, Nagarajan, Karthi, Mechin, Ingrid, Duffy, Caroline, Manavalan, Partha, Altmann, Steve, Majewski, Aliza, Foley, Joseph, Kaczmarek, J Stefan, Bercury, Scott, Maderia, Matthew, Hilbert, Brendan J, Batchelor, Joseph D, Ziegler, Robin, Bajko, Jeffrey, Kothe, Michael, Scheule, Ronald K, Nair, Anil, Hurlbut, Gregory D
Published in bioRxiv (20.04.2020)
Published in bioRxiv (20.04.2020)
Get full text
Paper
Compuestos de heteroaril-urea novedosos como inhibidores de kv7.2
MOWREY, David, DAVIES, Nicholas Gareth Morse, REDONDO PENA, Roger Lluis, NAIR, Anil, NAGARAJAN, Karthigeyan, MA, Nina, LI, Ronghua, MECHIN, Ingrid, NORCROSS, Roger David, GRAHAM, Christopher John, CHAPMAN, Mark, DAVIDSON, James, SMRCINA, Martin, LEBRETON, Sylvain, SAFAROVA, Alena, GERLACH, Aaron
Year of Publication 17.06.2024
Get full text
Year of Publication 17.06.2024
Patent
CRYSTALLOGRAPHIC MODEL OF THE BINDING SITE AND A MODULATOR REGULATING THE CATALYTIC ACTIVITY OF PHOSPHOFRUCTOKINASE (PFK), A METHOD OF DESIGNING, SELECTING AND PRODUCING THE PFK MODULATOR, A COMPUTER-BASED METHOD FOR THE ANALYSIS OF THE INTERACTIONS BETWEEN THE MODULATOR AND PFK
Get full text
Patent
Heteroarilaminosulfonamidas de 5 miembros para tratar afecciones mediadas por una actividad deficiente de cftr
William Wire, Zhongli Gao, Mark Munson, Bertrand Vivet, Sylvain Lebreton, Hans Peter Nestler, Sylvie Baltzer, Brian Freed, Gregory Hurlbut, Helen Yeoman, Martin Smrcina, Ryan Hartung, Junkai Liao, Ingrid Mechin, Nina Ma, Sukanthini Thurairatnam
Year of Publication 10.03.2023
Get full text
Year of Publication 10.03.2023
Patent
5-MEMBERED HETEROARYLAMINOSULFONAMIDES FOR TREATING CONDITIONS MEDIATED BY DEFICIENT CFTR ACTIVITY
BALTZER, Sylvie, WIRE, William, MA, Nina, HARTUNG, Ryan, GAO, Zhongli, LIAO, Junkai, YEOMAN, Helen, NESTLER, Hans, Peter, HURLBUT, Gregory, MECHIN, Ingrid, THURAIRATNAM, Sukanthini, VIVET, Bertrand, FREED, Brian, MUNSON, Mark, SMRCINA, Martin, LEBRETON, Sylvain
Year of Publication 30.01.2023
Get full text
Year of Publication 30.01.2023
Patent
HETEROARILAMINOSULFONAMIDAS DE 5 MIEMBROS PARA TRATAR AFECCIONES MEDIADAS POR UNA ACTIVIDAD DEFICIENTE DE CFTR
BALTZER, Sylvie, NESTLER, Hans Peter, WIRE, William, MA, Nina, HARTUNG, Ryan, GAO, Zhongli, LIAO, Junkai, YEOMAN, Helen, HURLBUT, Gregory, MECHIN, Ingrid, THURAIRATNAM, Sukanthini, VIVET, Bertrand, FREED, Brian, MUNSON, Mark, SMRCINA, Martin, LEBRETON, Sylvain
Year of Publication 21.09.2022
Get full text
Year of Publication 21.09.2022
Patent
Heteroarilaminosulfonamidas de 5 miembros para tratar afecciones mediadas por una actividad deficiente de cftr
BALTZER, Sylvie, NESTLER, Hans Peter, WIRE, William, MA, Nina, HARTUNG, Ryan, GAO, Zhongli, LIAO, Junkai, YEOMAN, Helen, HURLBUT, Gregory, MECHIN, Ingrid, THURAIRATNAM, Sukanthini, VIVET, Bertrand, FREED, Brian, MUNSON, Mark, SMRCINA, Martin, LEBRETON, Sylvain
Year of Publication 09.09.2022
Get full text
Year of Publication 09.09.2022
Patent
HETEROARILAMINOSULFONAMIDAS DE 5 MIEMBROS PARA TRATAR AFECCIONES MEDIADAS POR UNA ACTIVIDAD DEFICIENTE DE CFTR
BALTZER, Sylvie, NESTLER, Hans, WIRE, William, MA, Nina, HARTUNG, Ryan, GAO, Zhongli, YEOMAN, Helen, LIAO, Junkai, HURLBUT, Gregory, MECHIN, Ingrid, THURAIRATNAM, Sukanthini, VIVET, Bertrand, FREED, Brian, MUNSON, Mark, SMRCINA, Martin, LEBRETON, Sylvain
Year of Publication 31.08.2022
Get full text
Year of Publication 31.08.2022
Patent
HETEROARILAMINOSSULFONAMIDAS DE 5 MEMBROS PARA TRATAR AFECÇÕES MEDIADAS POR ATIVIDADE DE CFTR DEFICIENTE
BRIAN FREED, NINA MA, HANS PETER NESTLER, MARK MUNSON, GREGORY HURLBUT, RYAN HARTUNG, JUNKAI LIAO, INGRID MECHIN, SYLVIE BALTZER, ZHONGLI GAO, HELEN YEOMAN, WILLIAM WIRE, MARTIN SMRCINA, SUKANTHINI THURAIRATNAM, SYLVAIN LEBRETON, BERTRAND VIVET
Year of Publication 26.07.2022
Get full text
Year of Publication 26.07.2022
Patent