Intermolecular Rhodium-Catalyzed [3+2+2] Carbocyclization of Alkenylidenecyclopropanes with Activated Alkynes: Regio- and Diastereoselective Construction of cis-Fused Bicycloheptadienes
Evans, P. Andrew, Inglesby, Phillip A
Published in Journal of the American Chemical Society (01.10.2008)
Published in Journal of the American Chemical Society (01.10.2008)
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Synthesis of 2‑Oxopropanethioamide for the Manufacture of Lanabecestat: A New Route for Control, Robustness, and Operational Improvements
Taylor, Brian, Fernandez Barrat, Cristina, Woodward, Robert L, Inglesby, Phillip A
Published in Organic process research & development (15.09.2017)
Published in Organic process research & development (15.09.2017)
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Process Development of a Suzuki Reaction Used in the Manufacture of Lanabecestat
Ashworth, Ian W, Campbell, Andrew D, Cherryman, Janette H, Clark, Jemma, Crampton, Alex, Eden-Rump, Edward G. B, Evans, Matthew, Jones, Martin F, McKeever-Abbas, Sahar, Meadows, Rebecca E, Skilling, Kathryn, Whittaker, David T. E, Woodward, Robert L, Inglesby, Phillip A
Published in Organic process research & development (21.12.2018)
Published in Organic process research & development (21.12.2018)
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Process Development, Manufacture, and Understanding of the Atropisomerism and Polymorphism of Verinurad
Ring, Oliver T, Hayter, Barry R, Ronson, Thomas O, Agnew, Lauren R, Ashworth, Ian W, Cherryman, Janette, Gall, Malcolm A. Y, Hamilton, Peter R, Inglesby, Phillip A, Jones, Martin F, Lamacraft, Alex L, Leahy, Adam J, McKinney, David, Miller-Potucka, Lucie, Powell, Lyn, Putra, Okky D, Robbins, Andrew J, Tomasi, Simone, Wordsworth, Rosemary A
Published in Organic process research & development (18.03.2022)
Published in Organic process research & development (18.03.2022)
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Route Design to Manufacture: Synthesis of the Heterocyclic Fragment of AZD5718 Using a Non-cryogenic Lithiation-Alkoxycarbonylation Reaction
Burns, Matthew, Perkins, Dave, Chan, Lai C, Pilling, Michael J, Jawor-Baczynska, Anna, Mullen, Alexander K, Steven, Alan, Wimsey, Chris, Elmekawy, Ahmed, Lamacraft, Alex, Dobson, Benjamin C, McMillan, Angus E, Hose, David R. J, Inglesby, Phillip A, Raw, Steven A, Jones, Martin F
Published in Organic process research & development (16.04.2021)
Published in Organic process research & development (16.04.2021)
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Chemospecific Cyclizations of α‐Carbonyl Sulfoxonium Ylides on Aryls and Heteroaryls
Clare, Daniel, Dobson, Benjamin C., Inglesby, Phillip A., Aïssa, Christophe
Published in Angewandte Chemie (04.11.2019)
Published in Angewandte Chemie (04.11.2019)
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Diastereoselective Rhodium-Catalyzed [(3+2+2)] Carbocyclization Reactions with Tethered Alkynylidenecyclopropanes: Synthesis of the Tremulane Sesquiterpene Natural Products
Evans, P. Andrew, Dushnicky, Molly J., Cho, Dasol, Majhi, Jadab, Choi, Seulhui, Pipaliya, Bhavin, Inglesby, Phillip A., Baik, Mu-Hyun
Published in Asian journal of organic chemistry (01.08.2021)
Published in Asian journal of organic chemistry (01.08.2021)
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Exploiting the Physical Properties of Diethanolamine Boronic Esters for Process Improvements in AZD5718
Henry, Jean-Marc, Milne, David, Perkins, Dave, Hicks, William, Hose, David R. J., Campbell, Andrew D., Mullen, Alexander K., Inglesby, Phillip A., Raw, Steven A., Jones, Martin F.
Published in Organic process research & development (17.03.2023)
Published in Organic process research & development (17.03.2023)
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