Structure-activity relationship studies for inhibitors for vancomycin-resistant Enterococcus and human carbonic anhydrases
An, Weiwei, Holly, Katrina J., Nocentini, Alessio, Imhoff, Ryan D., Hewitt, Chad. S., Abutaleb, Nader S., Cao, Xufeng, Seleem, Mohamed N., Supuran, Claudiu T., Flaherty, Daniel P.
Published in Journal of enzyme inhibition and medicinal chemistry (31.12.2022)
Published in Journal of enzyme inhibition and medicinal chemistry (31.12.2022)
Get full text
Journal Article
Optimization and Anti-Cancer Properties of Fluoromethylketones as Covalent Inhibitors for Ubiquitin C-Terminal Hydrolase L1
Krabill, Aaron D, Chen, Hao, Hussain, Sajjad, Hewitt, Chad S, Imhoff, Ryan D, Muli, Christine S, Das, Chittaranjan, Galardy, Paul J, Wendt, Michael K, Flaherty, Daniel P
Published in Molecules (Basel, Switzerland) (25.02.2021)
Published in Molecules (Basel, Switzerland) (25.02.2021)
Get full text
Journal Article
Identification of covalent fragment inhibitors for Plasmodium falciparum UCHL3 with anti-malarial efficacy
Imhoff, Ryan D., Rosenthal, Melissa R., Ashraf, Kutub, Bhanot, Purnima, Ng, Caroline L., Flaherty, Daniel P.
Published in Bioorganic & medicinal chemistry letters (01.10.2023)
Published in Bioorganic & medicinal chemistry letters (01.10.2023)
Get full text
Journal Article
Covalent Fragment Screening and Optimization Identifies the Chloroacetohydrazide Scaffold as Inhibitors for Ubiquitin C‑terminal Hydrolase L1
Imhoff, Ryan D., Patel, Rishi, Safdar, Muhammad Hassan, Jones, Hannah B. L., Pinto-Fernandez, Adan, Vendrell, Iolanda, Chen, Hao, Muli, Christine S., Krabill, Aaron D., Kessler, Benedikt M., Wendt, Michael K., Das, Chittaranjan, Flaherty, Daniel P.
Published in Journal of medicinal chemistry (28.03.2024)
Published in Journal of medicinal chemistry (28.03.2024)
Get full text
Journal Article