Discovery of Gemilukast (ONO-6950), a Dual CysLT1 and CysLT2 Antagonist As a Therapeutic Agent for Asthma
Itadani, Satoshi, Yashiro, Kentaro, Aratani, Yoshiyuki, Sekiguchi, Tetsuya, Kinoshita, Atsushi, Moriguchi, Hideki, Ohta, Nobukazu, Takahashi, Shinya, Ishida, Akiharu, Tajima, Yohei, Hisaichi, Katsuya, Ima, Masaki, Ueda, Junya, Egashira, Hiromu, Sekioka, Tomohiko, Kadode, Michiaki, Yonetomi, Yasuo, Nakao, Takafumi, Inoue, Atsuto, Nomura, Hiroaki, Kitamine, Tetsuya, Fujita, Manabu, Nabe, Takeshi, Yamaura, Yoshiyuki, Matsumura, Naoya, Imagawa, Akira, Nakayama, Yoshisuke, Takeuchi, Jun, Ohmoto, Kazuyuki
Published in Journal of medicinal chemistry (13.08.2015)
Published in Journal of medicinal chemistry (13.08.2015)
Get full text
Journal Article
Discovery of Highly Potent Dual CysLT1 and CysLT2 Antagonist
Itadani, Satoshi, Takahashi, Shinya, Ima, Masaki, Sekiguchi, Tetsuya, Fujita, Manabu, Nakayama, Yoshisuke, Takeuchi, Jun
Published in ACS medicinal chemistry letters (13.11.2014)
Published in ACS medicinal chemistry letters (13.11.2014)
Get full text
Journal Article
Discovery of Gemilukast (ONO-6950), a Dual CysLT(1) and CysLT(2) Antagonist As a Therapeutic Agent for Asthma
Itadani, Satoshi, Yashiro, Kentaro, Aratani, Yoshiyuki, Sekiguchi, Tetsuya, Kinoshita, Atsushi, Moriguchi, Hideki, Ohta, Nobukazu, Takahashi, Shinya, Ishida, Akiharu, Tajima, Yohei, Hisaichi, Katsuya, Ima, Masaki, Ueda, Junya, Egashira, Hiromu, Sekioka, Tomohiko, Kadode, Michiaki, Yonetomi, Yasuo, Nakao, Takafumi, Inoue, Atsuto, Nomura, Hiroaki, Kitamine, Tetsuya, Fujita, Manabu, Nabe, Takeshi, Yamaura, Yoshiyuki, Matsumura, Naoya, Imagawa, Akira, Nakayama, Yoshisuke, Takeuchi, Jun, Ohmoto, Kazuyuki
Published in Journal of medicinal chemistry (13.08.2015)
Published in Journal of medicinal chemistry (13.08.2015)
Get full text
Journal Article
Discovery of a potent, orally available dual CysLT(1) and CysLT(2) antagonist with dicarboxylic acid
Itadani, Satoshi, Takahashi, Shinya, Ima, Masaki, Sekiguchi, Tetsuya, Aratani, Yoshiyuki, Egashira, Hiromu, Matsumura, Naoya, Inoue, Atsuto, Yonetomi, Yasuo, Fujita, Manabu, Nakayama, Yoshisuke, Takeuchi, Jun
Published in Bioorganic & medicinal chemistry (01.05.2015)
Published in Bioorganic & medicinal chemistry (01.05.2015)
Get full text
Journal Article
Discovery of a potent, orally available dual CysLT1 and CysLT2 antagonist with dicarboxylic acid
Itadani, Satoshi, Takahashi, Shinya, Ima, Masaki, Sekiguchi, Tetsuya, Aratani, Yoshiyuki, Egashira, Hiromu, Matsumura, Naoya, Inoue, Atsuto, Yonetomi, Yasuo, Fujita, Manabu, Nakayama, Yoshisuke, Takeuchi, Jun
Published in Bioorganic & medicinal chemistry (01.05.2015)
Published in Bioorganic & medicinal chemistry (01.05.2015)
Get full text
Journal Article
Discovery of Highly Potent Dual CysLT(1) and CysLT(2) Antagonist
Itadani, Satoshi, Takahashi, Shinya, Ima, Masaki, Sekiguchi, Tetsuya, Fujita, Manabu, Nakayama, Yoshisuke, Takeuchi, Jun
Published in ACS medicinal chemistry letters (01.11.2014)
Published in ACS medicinal chemistry letters (01.11.2014)
Get full text
Journal Article
Discovery of Gemilukast (ONO-6950), a Dual CysLT 1 and CysLT 2 Antagonist As a Therapeutic Agent for Asthma
Itadani, Satoshi, Yashiro, Kentaro, Aratani, Yoshiyuki, Sekiguchi, Tetsuya, Kinoshita, Atsushi, Moriguchi, Hideki, Ohta, Nobukazu, Takahashi, Shinya, Ishida, Akiharu, Tajima, Yohei, Hisaichi, Katsuya, Ima, Masaki, Ueda, Junya, Egashira, Hiromu, Sekioka, Tomohiko, Kadode, Michiaki, Yonetomi, Yasuo, Nakao, Takafumi, Inoue, Atsuto, Nomura, Hiroaki, Kitamine, Tetsuya, Fujita, Manabu, Nabe, Takeshi, Yamaura, Yoshiyuki, Matsumura, Naoya, Imagawa, Akira, Nakayama, Yoshisuke, Takeuchi, Jun, Ohmoto, Kazuyuki
Published in Journal of medicinal chemistry (13.08.2015)
Published in Journal of medicinal chemistry (13.08.2015)
Get full text
Journal Article
Discovery of Highly Potent Dual CysLT 1 and CysLT 2 Antagonist
Itadani, Satoshi, Takahashi, Shinya, Ima, Masaki, Sekiguchi, Tetsuya, Fujita, Manabu, Nakayama, Yoshisuke, Takeuchi, Jun
Published in ACS medicinal chemistry letters (13.11.2014)
Published in ACS medicinal chemistry letters (13.11.2014)
Get full text
Journal Article
Further optimization of sulfonamide analogs as EP1 receptor antagonists: Synthesis and evaluation of bioisosteres for the carboxylic acid group
Naganawa, Atsushi, Matsui, Toshiaki, Ima, Masaki, Saito, Tetsuji, Murota, Masayuki, Aratani, Yoshiyuki, Kijima, Hideomi, Yamamoto, Hiroshi, Maruyama, Takayuki, Ohuchida, Shuichi, Nakai, Hisao, Toda, Masaaki
Published in Bioorganic & medicinal chemistry (01.11.2006)
Published in Bioorganic & medicinal chemistry (01.11.2006)
Get full text
Journal Article
Optimization of sulfonamide derivatives as highly selective EP1 receptor antagonists
Naganawa, Atsushi, Matsui, Toshiaki, Ima, Masaki, Yoshida, Koji, Tsuruta, Hiroshi, Yamamoto, Shingo, Yamamoto, Hiroshi, Okada, Hiroki, Maruyama, Takayuki, Nakai, Hisao, Kondo, Kigen, Toda, Masaaki
Published in Bioorganic & medicinal chemistry (01.12.2006)
Published in Bioorganic & medicinal chemistry (01.12.2006)
Get full text
Journal Article
Discovery of heteroaryl sulfonamides as new EP1 receptor selective antagonists
Naganawa, Atsushi, Matsui, Toshiaki, Saito, Tetsuji, Ima, Masaki, Tatsumi, Tadashi, Yamamoto, Shingo, Murota, Masayuki, Yamamoto, Hiroshi, Maruyama, Takayuki, Ohuchida, Shuichi, Nakai, Hisao, Kondo, Kigen, Toda, Masaaki
Published in Bioorganic & medicinal chemistry (01.10.2006)
Published in Bioorganic & medicinal chemistry (01.10.2006)
Get full text
Journal Article
DIPHENYL ETHER COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE
NAKAYAMA, YOSHISUKE, TAJIMA, HISAO, KUSUDA, SHINYA, IMA, MASAKI, KATO, SACHIKO
Year of Publication 10.02.2005
Get full text
Year of Publication 10.02.2005
Patent
Diphenyl ether compound, process for producing the same, and use
KUSUDA SHINYA, TAJIMA HISAO, KATO SACHIKO, IMA MASAKI, NAKAYAMA YOSHISUKE
Year of Publication 21.10.2010
Get full text
Year of Publication 21.10.2010
Patent
DIPHENYL ETHER COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE
NAKAYAMA, YOSHISUKE, TAJIMA, HISAO, KUSUDA, SHINYA, IMA, MASAKI, KATO, SACHIKO
Year of Publication 29.11.2006
Get full text
Year of Publication 29.11.2006
Patent
DIPHENYL ETHER COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE
NAKAYAMA, YOSHISUKE, TAJIMA, HISAO, KUSUDA, SHINYA, IMA, MASAKI, KATO, SACHIKO
Year of Publication 31.05.2006
Get full text
Year of Publication 31.05.2006
Patent