Rational design and synthesis of 2-(1H-indazol-6-yl)-1H-benzo[d]imidazole derivatives as inhibitors targeting FMS-like tyrosine kinase 3 (FLT3) and its mutants
Im, Daseul, Jun, Joonhong, Baek, Jihyun, Kim, Haejin, Kang, Dahyun, Bae, Hyunah, Cho, Hyunwook, Hah, Jung-Mi
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2022)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2022)
Get full text
Journal Article
Discovery of 1-Pyrimidinyl-2-Aryl-4,6-Dihydropyrrolo [3,4-d]Imidazole-5(1 H )-Carboxamide as a Novel JNK Inhibitor
Jang, Miyoung, Oh, Youri, Cho, Hyunwook, Yang, Songyi, Moon, Hyungwoo, Im, Daseul, Hah, Jung-Mi
Published in International journal of molecular sciences (02.03.2020)
Published in International journal of molecular sciences (02.03.2020)
Get full text
Journal Article
Discovery of 4-arylamido 3-methyl isoxazole derivatives as novel FMS kinase inhibitors
Im, Daseul, Jung, Kyungjin, Yang, Songyi, Aman, Waqar, Hah, Jung-Mi
Published in European journal of medicinal chemistry (18.09.2015)
Published in European journal of medicinal chemistry (18.09.2015)
Get full text
Journal Article
Design and Synthesis of a Novel PLK1 Inhibitor Scaffold Using a Hybridized 3D-QSAR Model
Oh, Youri, Jung, Hoyong, Kim, Hyejin, Baek, Jihyun, Jun, Joonhong, Cho, Hyunwook, Im, Daseul, Hah, Jung-Mi
Published in International journal of molecular sciences (08.04.2021)
Published in International journal of molecular sciences (08.04.2021)
Get full text
Journal Article
Discovery of 3-alkyl-5-aryl-1-pyrimidyl-1H-pyrazole derivatives as a novel selective inhibitor scaffold of JNK3
Oh, Youri, Jang, Miyoung, Cho, Hyunwook, Yang, Songyi, Im, Daseul, Moon, Hyungwoo, Hah, Jung-Mi
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Get full text
Journal Article
Computer-aided design and synthesis of 3-carbonyl-5-phenyl-1H-pyrazole as highly selective and potent BRAFV600E and CRAF inhibitor
Kim, Jinwoong, Choi, Byeongha, Im, Daseul, Jung, Hoyong, Moon, Hyungwoo, Aman, Waqar, Hah, Jung-Mi
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Get full text
Journal Article
Discovery of 5-methyl-N-(2-arylquinazolin-7-yl)isoxazole-4-carboxamide analogues as highly selective FLT3 inhibitors
Im, Daseul, Moon, Hyungwoo, Kim, Jinwoong, Oh, Youri, Jang, Miyoung, Hah, Jung-Mi
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Get full text
Journal Article
Conformational restriction of a type II FMS inhibitor leading to discovery of 5-methyl-N-(2-aryl-1H-benzo[d]imidazo-5-yl)isoxazole-4-carboxamide analogues as selective FLT3 inhibitors
Im, Daseul, Moon, Hyungwoo, Kim, Jingwoong, Oh, Youri, Jang, Miyoung, Hah, Jung-Mi
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2019)
Get full text
Journal Article
New potential application of hydroxypropyl-β-cyclodextrin in solid self-nanoemulsifying drug delivery system and solid dispersion
Kim, Jung Suk, Choi, Yoo Jin, Woo, Mi Ran, Cheon, Seunghyun, Ji, Sang Hun, Im, Daseul, ud Din, Fakhar, Kim, Jong Oh, Youn, Yu Seok, Oh, Kyung Taek, Lim, Soo-Jeong, Jin, Sung Giu, Choi, Han-Gon
Published in Carbohydrate polymers (01.11.2021)
Published in Carbohydrate polymers (01.11.2021)
Get full text
Journal Article
Rational design and synthesis of 2-(1 H -indazol-6-yl)-1 H -benzo[d]imidazole derivatives as inhibitors targeting FMS-like tyrosine kinase 3 (FLT3) and its mutants
Im, Daseul, Jun, Joonhong, Baek, Jihyun, Kim, Haejin, Kang, Dahyun, Bae, Hyunah, Cho, Hyunwook, Hah, Jung-Mi
Published in Journal of enzyme inhibition and medicinal chemistry (31.12.2022)
Published in Journal of enzyme inhibition and medicinal chemistry (31.12.2022)
Get full text
Journal Article
Discovery of novel imidazole chemotypes as isoform-selective JNK3 inhibitors for the treatment of Alzheimer's disease
Jun, Joonhong, Yang, Songyi, Lee, Junghun, Moon, Hyungwoo, Kim, Jinwoong, Jung, Hoyong, Im, Daseul, Oh, Youri, Jang, Miyoung, Cho, Hyunwook, Baek, Jihyun, Kim, Hyejin, Kang, Dahyun, Bae, Hyunah, Tak, Chanwool, Hwang, Kyungrim, Kwon, Hoseok, Kim, HyunTae, Hah, Jung-Mi
Published in European journal of medicinal chemistry (05.01.2023)
Published in European journal of medicinal chemistry (05.01.2023)
Get full text
Journal Article
Discovery of 3-alkyl-5-aryl-1-pyrimidyl-1 H- pyrazole derivatives as a novel selective inhibitor scaffold of JNK3
Oh, Youri, Jang, Miyoung, Cho, Hyunwook, Yang, Songyi, Im, Daseul, Moon, Hyungwoo, Hah, Jung-Mi
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2020)
Get full text
Journal Article
Crystal structure of the YoeBSa1-YefMSa1 complex from Staphylococcus aureus
Eun, Hyun-Jong, Lee, Ki-Young, Kim, Dong-Gyun, Im, Daseul, Lee, Bong-Jin
Published in Biochemical and biophysical research communications (18.06.2020)
Published in Biochemical and biophysical research communications (18.06.2020)
Get full text
Journal Article
Computer-aided design and synthesis of 3-carbonyl-5-phenyl-1 H -pyrazole as highly selective and potent BRAFV600E and CRAF inhibitor
Kim, Jinwoong, Choi, Byeongha, Im, Daseul, Jung, Hoyong, Moon, Hyungwoo, Aman, Waqar, Hah, Jung-Mi
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2019)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2019)
Get full text
Journal Article
Discovery of novel 4-aryl-thieno[1,4]diazepin-2-one derivatives targeting multiple protein kinases as anticancer agents
Lee, Junghun, Jung, Hoyong, Kim, Minjung, Lee, Eunkyu, Im, Daseul, Aman, Waqar, Hah, Jung-Mi
Published in Bioorganic & medicinal chemistry (01.05.2018)
Published in Bioorganic & medicinal chemistry (01.05.2018)
Get full text
Journal Article
Crystal structure of the YoeB Sa1 -YefM Sa1 complex from Staphylococcus aureus
Eun, Hyun-Jong, Lee, Ki-Young, Kim, Dong-Gyun, Im, Daseul, Lee, Bong-Jin
Published in Biochemical and biophysical research communications (18.06.2020)
Get full text
Published in Biochemical and biophysical research communications (18.06.2020)
Journal Article