Bioassay protocol metadata annotation: Proposed standards adoption
Balakrishnan, Rama, Berg, Ellen L., Butler, Christopher C., Clark, Alex M., Denker, Sheryl P., Feierberg, Isabella, Harris, Jason, Ikeda, Timothy P., Jeschonek, Samantha, Makarov, Vladimir A., Southan, Christopher, Vanderwall, Dana, Winstanley, Peter
Published in SLAS discovery (01.12.2024)
Published in SLAS discovery (01.12.2024)
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Optimization of a series of potent, selective and orally bioavailable SYK inhibitors
Grimster, Neil P., Gingipalli, Lakshmaiah, Barlaam, Bernard, Su, Qibin, Zheng, XiaoLan, Watson, David, Wang, Haixia, Simpson, Iain, Pike, Andy, Balazs, Amber, Boiko, Scott, Ikeda, Timothy P., Impastato, Anna C., Jones, Natalie H., Kawatkar, Sameer, Kemmitt, Paul, Lamont, Scott, Patel, Joe, Read, Jon, Sarkar, Ujjal, Sha, Li, Tomlinson, Ronald C., Wang, Haiyun, Wilson, David M., Zehnder, Troy E., Wang, Lianghe, Wang, Peng, Goldberg, Frederick W., Shao, Wenlin, Fawell, Stephen, Dry, Hannah, Dowling, James E., Edmondson, Scott D.
Published in Bioorganic & medicinal chemistry letters (01.10.2020)
Published in Bioorganic & medicinal chemistry letters (01.10.2020)
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High-throughput mechanistic screening of non-equilibrium inhibitors by a fully automated data analysis pipeline in early drug-discovery
Srinivasan, Bharath, Flórez Weidinger, Juan Daniel, Zhai, Xiang, Lemercier, Guillaume, Ikeda, Timothy, Brewer, Mark, Zhang, Bairu, Heyse, Stephan, Wingfield, Jonathan, Steigele, Stephan
Published in SLAS discovery (01.12.2022)
Published in SLAS discovery (01.12.2022)
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Novel potent and selective pyrazolylpyrimidine-based SYK inhibitors
Barlaam, Bernard, Boiko, Scott, Boyd, Scott, Dry, Hannah, Gingipalli, Lakshmaiah, Ikeda, Timothy, Johnson, Tony, Kawatkar, Sameer, Lorthioir, Olivier, Pike, Andy, Pollard, Hannah, Read, Jon, Su, Qibin, Wang, Haiyun, Wang, Huimin, Wang, Lianghe, Wang, Peng, Edmondson, Scott D.
Published in Bioorganic & medicinal chemistry letters (15.11.2020)
Published in Bioorganic & medicinal chemistry letters (15.11.2020)
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Identification of a novel series of azabenzimidazole-derived inhibitors of spleen tyrosine kinase
Kawatkar, Sameer P., Barlaam, Bernard, Kemmitt, Paul, Simpson, Iain, Watson, David, Wang, Peng, Lamont, Scott, Su, Qibin, Boiko, Scott, Ikeda, Timothy, Patel, Joe, Pike, Andy, Pollard, Hannah, Read, Jon, Sarkar, Ujjal, Wang, Haiyun, Wen, Quanshan, Yan, Zhiyuan, Dowling, James E., Dry, Hannah, Edmondson, Scott D.
Published in Bioorganic & medicinal chemistry letters (15.09.2020)
Published in Bioorganic & medicinal chemistry letters (15.09.2020)
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Isocitrate Dehydrogenase Kinase/Phosphatase
Miller, Stephen P., Karschnia, Elizabeth J., Ikeda, Timothy P., LaPorte, David C.
Published in The Journal of biological chemistry (09.08.1996)
Published in The Journal of biological chemistry (09.08.1996)
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