Crystal Structures of Rat Vitamin D Receptor Bound to Adamantyl Vitamin D Analogs: Structural Basis for Vitamin D Receptor Antagonism and Partial Agonism
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Identification of a highly potent vitamin D receptor antagonist: (25S)-26-Adamantyl-25-hydroxy-2-methylene-22,23-didehydro-19,27-dinor-20-epi-vitamin D3 (ADMI3)
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Year of Publication 24.07.2023
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Methods of Using 4-Amino-N-[4-(Methoxymethyl)Phenyl]-7-(1-Methylcyclopropyl)-6-(3-Morpholinoprop-1-YN-1-YL)-7H-Pyrrolo[2,3-D]Pyrimidine-5-Carboxamide for the Treatment of Tumors
Giuliano, Claudio, Kato, Masanori, Bonifacio, Annalisa, Miyazaki, Isao, Lovati, Emanuela, Igarashi, Miharu, Bernareggi, Alberto, Giorgino, Ruben, Doria, Simona
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Year of Publication 04.01.2024
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METHODS OF USING 4-AMINO-N-[4-(METHOXYMETHYL)PHENYL]-7-(1-METHYLCYCLOPROPYL)-6-(3-MORPHOLINOPROP-1-YN-1-YL)-7H-PYRROLO[2,3-D]PYRIMIDINE-5-CARBOXAMIDE FOR THE TREATMENT OF TUMORS
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Year of Publication 27.09.2023
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Year of Publication 27.09.2023
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Methods of using 4-amino-n-[4-(methoxymethyl)phenyl]-7-(1-methylcyclopropyl)-6-(3-morpholinoprop-1-yn-1-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carboxamide for the treatment of tumors
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Year of Publication 01.06.2023
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METHODS OF USING 4-AMINO-N-[4-(METHOXYMETHYL)PHENYL]-7-(1-METHYLCYCLOPROPYL)-6-(3-MORPHOLINOPROP-1-YN-1-YL)-7H-PYRROLO[2,3-D]PYRIMIDINE-5-CARBOXAMIDE FOR THE TREATMENT OF TUMORS
DORIA, Simona, BONIFACIO, Annalisa, KATO, Masanori, MIYAZAKI, Isao, GIULIANO, Claudio, GIORGINO, Ruben, IGARASHI, Miharu, BERNAREGGI, Alberto, LOVATI, Emanuela
Year of Publication 25.05.2023
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Year of Publication 25.05.2023
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METHODS OF USING 4-AMINO-N-[4-(METHOXYMETHYL)PHENYL]-7-(1-METHYLCYCLOPROPYL)-6-(3-MORPHOLINOPROP-1-YN-1-YL)-7H-PYRROLO[2,3-D]PYRIMIDINE-5-CARBOXAMIDE FOR THE TREATMENT OF TUMORS
DORIA, Simona, BONIFACIO, Annalisa, KATO, Masanori, MIYAZAKI, Isao, GIULIANO, Claudio, GIORGINO, Ruben, IGARASHI, Miharu, BERNAREGGI, Alberto, LOVATI, Emanuela
Year of Publication 27.05.2022
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Year of Publication 27.05.2022
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METHODS OF USING 4-AMINO-N-[4-(METHOXYMETHYL)PHENYL]-7-(1-METHYLCYCLOPROPYL)-6-(3-MORPHOLINOPROP-1-YN-1-YL)-7H-PYRROLO[2,3-D]PYRIMIDINE-5-CARBOXAMIDE FOR THE TREATMENT OF TUMORS
MIYAZAKI, ISAO, GIULIANO, CLAUDIO, BERNAREGGI, ALBERTO, BONIFACIO, ANNALISA, KATO, MASANORI, LOVATI, EMANUELA, DORIA, SIMONA, IGARASHI, MIHARU, GIORGINO, RUBEN
Year of Publication 27.05.2022
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Year of Publication 27.05.2022
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METHODS OF USING 4-AMINO-N-[4-(METHOXYMETHYL)PHENYL]-7-(1-METHYLC YCLOPROPYL)-6-(3-MORPHOLINOPROP-1-YN-1-YL)-7H-PYRROLO[2,3-D]PYRI MIDINE-5-CARBOXAMIDE FOR THE TREATMENT OF TUMORS
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Year of Publication 17.07.2023
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Year of Publication 17.07.2023
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Methods of using 4-amino-N-[4-(methoxymethyl)phenyl]-7-(1-methylcyclopropyl)-6-(3-morpholinoprop-1-yn-1-yl)-7H-pyrrolo[2,3-D]pyrimidine-5-carboxamide for the treatment of tumors
MIYAZAKI, ISAO, GIULIANO, CLAUDIO, BERNAREGGI, ALBERTO, BONIFACIO, ANNALISA, KATO, MASANORI, LOVATI, EMANUELA, DORIA, SIMONA, IGARASHI, MIHARU, GIORGINO, RUBEN
Year of Publication 01.10.2022
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Year of Publication 01.10.2022
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