Antagonists of the human adenosine A2A receptor. Part 3 Design and synthesis of pyrazolo[3,4-d]pyrimidines, pyrrolo[2,3-d]pyrimidines and 6-arylpurines
GILLESPIE, Roger J, CLIFFE, Ian A, ROLFEY, Jonathan, STRATTON, Gemma C, UPTON, Rebecca, WEISS, Scott M, WILLIAMSON, Douglas S, DAWSON, Claire E, DOURISH, Colin T, GAUR, Suneel, JORDAN, Allan M, KNIGHT, Antony R, LERPINIERE, Joanne, MISRA, Anil, PRATT, Robert M
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
Get full text
Journal Article
Approaches towards the development of chimeric DPP4/ACE inhibitors for treating metabolic syndrome
Sattigeri, Jitendra A., Sethi, Sachin, Davis, Joseph A., Ahmed, Shahadat, Rayasam, Geeta V., Jadhav, Balasaheb G., Chilla, Satya M., Datta, Dhrubajyoti, Gadhave, A., Tulasi, Vamshi K., Jain, Tarun, Voleti, Sreedhara, Benjamin, Biju, Udupa, Sunitha, Jain, Garima, Singh, Yogender, Srinivas, Kona, Bansal, Vinay S., Ray, Abhijit, Bhatnagar, Pradip K., Cliffe, Ian A.
Published in Bioorganic & medicinal chemistry letters (01.06.2017)
Published in Bioorganic & medicinal chemistry letters (01.06.2017)
Get full text
Journal Article
Efficient and Selective Demethylation of Heteroaryl Methyl Ethers in the Presence of Aryl Methyl Ethers
Soni, Ajay, Dutt, Akhilesh, Sattigeri, Viswajanani, Cliffe, Ian A.
Published in Synthetic communications (04.05.2011)
Published in Synthetic communications (04.05.2011)
Get full text
Journal Article
Synthesis and evaluation of 4,5-dihydro-5-methylisoxazolin-5-carboxamide derivatives as VLA-4 antagonists
Soni, Ajay, Rehman, Abdul, Naik, Keshav, Dastidar, Sunanda, Alam, M.S., Ray, Abhijit, Chaira, Tridib, Shah, Vanya, Palle, Venkata P., Cliffe, Ian A., Sattigeri, Viswajanani J.
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
Get full text
Journal Article
Antagonists of the human adenosine A2A receptor. Part 1 Discovery and synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives
GILLESPIE, Roger J, ADAMS, David R, JORDAN, Allan M, KNIGHT, Antony R, KNUTSEN, Lars J. S, LAWRENCE, Anthony, LERPINIERE, Joanne, MISRA, Anil, PORTER, Richard H. P, PRATT, Robert M, SHEPHERD, Robin, UPTON, Rebecca, BEBBINGTON, David, WARD, Simon E, WEISS, Scott M, WILLIAMSON, Douglas S, BENWELL, Karen, CLIFFE, Ian A, DAWSON, Claire E, DOURISH, Colin T, FLETCHER, Allan, GAUR, Suneel, GILES, Paul R
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
Get full text
Journal Article
Antagonists of the human adenosine A2A receptor. Part 2 Design and synthesis of 4-arylthieno[3,2-d]pyrimidine derivatives
GILLESPIE, Roger J, CLIFFE, Ian A, MISRA, Anil, PRATT, Robert M, TODD, Richard S, UPTON, Rebecca, WEISS, Scott M, WILLIAMSON, Douglas S, DAWSON, Claire E, DOURISH, Colin T, GAUR, Suneel, GILES, Paul R, JORDAN, Allan M, KNIGHT, Antony R, LAWRENCE, Anthony, LERPINIERE, Joanne
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
Get full text
Journal Article
Pharmacodynamic and pharmacokinetic profile of RBx 343E48F0: A novel, long acting muscarinic receptor antagonist
Gupta, Suman, Malhotra, Shivani, Sinha, Sandeep, Singh, Shashi K., Singh, Rakesh K., Krishna, Siddarangaiah, Chhabra, Pooja, Chaira, Tridib, Kannayiram, Janaki, Sharma, Pradeep, Aeron, Shelly, Kaur, Jaskiran, Kumar, Naresh, Sattigeri, Jitendra, Shirumalla, Raj K., Paliwal, Jyoti, Dastidar, Sunanda G., Cliffe, Ian A., Ray, Abhijit, Bhatnagar, Pradip
Published in European journal of pharmacology (11.05.2011)
Published in European journal of pharmacology (11.05.2011)
Get full text
Journal Article
A pharmacological profile of the selective silent 5-HT1A receptor antagonist, WAY-100635
Forster, E A, Cliffe, I A, Bill, D J, Dover, G M, Jones, D, Reilly, Y, Fletcher, A
Published in European journal of pharmacology (25.07.1995)
Published in European journal of pharmacology (25.07.1995)
Get full text
Journal Article
Synthesis and biological activity of N-substituted aminocarbonyl-1,3-dioxolanes as VLA-4 antagonists
Rehman, Abdul, Soni, Ajay, Naik, Keshav, Nair, Sreeji, Palle, Venkata P., Dastidar, Sunanda, Ray, Abhijit, Alam, M.S., Salman, Mohammad, Cliffe, Ian A., Sattigeri, Viswajanani
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
Get full text
Journal Article
A retrospect on the discovery of way-100635 and the prospect for improved 5-HT1A receptor PET radioligands
Get full text
Conference Proceeding
Journal Article
UDP-N-acetylglucosamine enolpyruvyl transferase from Pseudomonas aeruginosa
Dube, Smita, Nanda, Kamna, Rani, Reema, Kaur, Namrata Jit, Nagpal, Jatin Kumar, Upadhyay, Dilip J, Cliffe, Ian A, Saini, Kulvinder Singh, Purnapatre, Kedar P
Published in World journal of microbiology & biotechnology (01.09.2010)
Published in World journal of microbiology & biotechnology (01.09.2010)
Get full text
Journal Article
Synthesis and antibacterial activity of potent heterocyclic oxazolidinones and the identification of RBx 8700
Rudra, Sonali, Yadav, Ajay, Raja Rao, A.V.S., Srinivas, A.S.S.V., Pandya, Manisha, Bhateja, Pragya, Mathur, Tarun, Malhotra, Sunita, Rattan, Ashok, Salman, Mohammed, Mehta, Anita, Cliffe, Ian A., Das, Biswajit
Published in Bioorganic & medicinal chemistry letters (15.12.2007)
Published in Bioorganic & medicinal chemistry letters (15.12.2007)
Get full text
Journal Article
Pyrrolo(iso)quinoline derivatives as 5-HT2C receptor agonists
ADAMS, David R, BENTLEY, Jonathan M, MALCOLM, Craig S, MANSELL, Howard L, MISRA, Anil, QUIRK, Kathleen, ROFFEY, Jonathan R. A, VICKERS, Steven P, BENWELL, Karen R, BICKERDIKE, Michael J, BODKIN, Corinna D, CLIFFE, Ian A, DOURISH, Colin T, GEORGE, Ashley R, KENNETT, Guy A, KNIGHT, Antony R
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Get full text
Journal Article
Silent 5-HT1A receptor antagonists : utility as research tools and therapeutic agents
FLETCHER, A, CLIFFE, I. A, DOURISH, C. T
Published in Trends in pharmacological sciences (Regular ed.) (01.12.1993)
Published in Trends in pharmacological sciences (Regular ed.) (01.12.1993)
Get full text
Journal Article
WAY100135 : a novel, selective antagonist at presynaptic and postsynaptic 5-HT1A receptors
FLETCHER, A, BILL, D. J, BILL, S. J, CLIFFE, I. A, DOVER, G. M, FORSTER, E. A, HASKINS, J. T, JONES, D, MANSELL, H. L, REILLY, Y
Published in European journal of pharmacology (24.06.1993)
Published in European journal of pharmacology (24.06.1993)
Get full text
Journal Article
5-HT2C receptor agonists for the treatment of obesity. Biological and chemical adventures
Adams, D, Benardeau, A, Bickerdike, MJ, Bentley, JM, Bissantz, C, Bourson, A, Cliffe, IA, Hebeisen, P, Kennett, GA, Knight, AR, Malcolm, CS, Mizrahi, J, Plancher, JM, Richter, H, Rover, S, Taylor, S, Vickers, SP
Published in Chimia (01.09.2004)
Published in Chimia (01.09.2004)
Get full text
Journal Article
Oral hypoglycemic agents. Pyrimido[1,2-a]indoles and related compounds
Cliffe, Ian A, Lien, Eric L, Mansell, Howard L, Steiner, Kurt E, Todd, Richard S, White, Alan C, Black, Robin M
Published in Journal of medicinal chemistry (01.04.1992)
Published in Journal of medicinal chemistry (01.04.1992)
Get full text
Journal Article