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AVN-322 is a Safe Orally Bio-Available Potent and Highly Selective Antagonist of 5-HT6R with Demonstrated Ability to Improve Impaired Memory in Animal Models
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Optimization of the dipeptide motifs in the PSMA ligands linker structure: synthesis and in vitro evaluation
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2-Pyrazol-1-yl-thiazole derivatives as novel highly potent antibacterials
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Published in Journal of antibiotics (01.11.2019)
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A Comprehensive Insight into the Chemical Space and ADME Features of Small Molecule NS5A Inhibitors
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Chemistry42: An AI-Driven Platform for Molecular Design and Optimization
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In Silico Approaches to the Design of NS5A Inhibitors
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Identification of Novel Small-Molecule ASGP-R Ligands
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Salihov, Sergei V., Ivanenkov, Yan A., Krechetov, Sergei P., Veselov, Mark S., Sviridenkova, Natalia V., Savchenko, Alexander G., Klyachko, Natalya L., Golovin, Yury I., Chufarova, Nina V., Beloglazkina, Elena K., Majouga, Alexander G.
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Sorting Out Antibiotics' Mechanisms of Action: a Double Fluorescent Protein Reporter for High-Throughput Screening of Ribosome and DNA Biosynthesis Inhibitors
Osterman, Ilya A, Komarova, Ekaterina S, Shiryaev, Dmitry I, Korniltsev, Ilya A, Khven, Irina M, Lukyanov, Dmitry A, Tashlitsky, Vadim N, Serebryakova, Marina V, Efremenkova, Olga V, Ivanenkov, Yan A, Bogdanov, Alexey A, Sergiev, Petr V, Dontsova, Olga A
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Deep learning enables rapid identification of potent DDR1 kinase inhibitors
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Published in Nature biotechnology (01.09.2019)
Published in Nature biotechnology (01.09.2019)
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Resistance profiles for the investigational neuraminidase inhibitor AV5080 in influenza A and B viruses
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Published in Antiviral research (01.09.2023)
Published in Antiviral research (01.09.2023)
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Synthesis and Biological Evaluation of PSMA Ligands with Aromatic Residues and Fluorescent Conjugates Based on Them
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Published in Journal of medicinal chemistry (22.04.2021)
Published in Journal of medicinal chemistry (22.04.2021)
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Synthesis and initial in vitro evaluation of PSMA-targeting ligands with a modified aromatic moiety at the lysine ε-nitrogen atom
Zyk, Nikolai Y., Ber, Anton P., Nimenko, Ekaterina A., Shafikov, Radik R., Evteev, Sergei A., Petrov, Stanislav A., Uspenskaya, Anastasia A., Dashkova, Natalia S., Ivanenkov, Yan A., Skvortsov, Dmitry A., Beloglazkina, Elena K., Majouga, Alexander G., Machulkin, Aleksei E.
Published in Bioorganic & medicinal chemistry letters (01.09.2022)
Published in Bioorganic & medicinal chemistry letters (01.09.2022)
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