First X-ray Cocrystal Structure of a Bacterial FabH Condensing Enzyme and a Small Molecule Inhibitor Achieved Using Rational Design and Homology Modeling
Daines, Robert A, Pendrak, Israil, Sham, Kelvin, Van Aller, Glenn S, Konstantinidis, Alex K, Lonsdale, John T, Janson, Cheryl A, Qiu, Xiayang, Brandt, Martin, Khandekar, Sanjay S, Silverman, Carol, Head, Martha S
Published in Journal of medicinal chemistry (02.01.2003)
Published in Journal of medicinal chemistry (02.01.2003)
Get full text
Journal Article
Synthesis and Anti-HSV Activity of A-Ring-Deleted Mappicine Ketone Analog
Pendrak, Israil, Barney, Shawn, Wittrock, Robert, Lambert, Dennis M, Kingsbury, William D
Published in Journal of organic chemistry (01.05.1994)
Published in Journal of organic chemistry (01.05.1994)
Get full text
Journal Article
Development of GSK's reagent guides ― embedding sustainability into reagent selection
ADAMS, Joseph P, ALDER, Catherine M, REDMAN, Anikó M, SHUSTER, Leanna E, SNEDDON, Helen F, WALKER, Matthew D, ANDREWS, Ian, BULLION, Ann M, CAMPBELL-CRAWFORD, Matthew, DARCY, Michael G, HAYLER, John D, HENDERSON, Richard K, OARE, Catriona A, PENDRAK, Israil
Published in Green chemistry : an international journal and green chemistry resource : GC (01.01.2013)
Published in Green chemistry : an international journal and green chemistry resource : GC (01.01.2013)
Get full text
Journal Article
Design and Optimization of Sulfone Pyrrolidine Sulfonamide Antagonists of Transient Receptor Potential Vanilloid‑4 with in Vivo Activity in a Pulmonary Edema Model
Pero, Joseph E, Matthews, Jay M, Behm, David J, Brnardic, Edward J, Brooks, Carl, Budzik, Brian W, Costell, Melissa H, Donatelli, Carla A, Eisennagel, Stephen H, Erhard, Karl, Fischer, Michael C, Holt, Dennis A, Jolivette, Larry J, Li, Huijie, Li, Peng, McAtee, John J, McCleland, Brent W, Pendrak, Israil, Posobiec, Lorraine M, Rivera, Katrina L.K, Rivero, Ralph A, Roethke, Theresa J, Sender, Matthew R, Shu, Arthur, Terrell, Lamont R, Vaidya, Kalindi, Xu, Xiaoping, Lawhorn, Brian G
Published in Journal of medicinal chemistry (27.12.2018)
Published in Journal of medicinal chemistry (27.12.2018)
Get full text
Journal Article
Synthesis and LTB4 receptor antagonist activities of the naturally occurring LTB4 receptor antagonist leucettamine A and related analogs
Boehm, Jeffrey C, Gleason, John G, Pendrak, Israil, Sarau, Henry M, Schmidt, Dulcie B, Foley, James J, Kingsbury, William D
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
Get full text
Journal Article
Development of GSK's reagent guides embedding sustainability into reagent selectionElectronic supplementary information (ESI) available. See DOI: 10.1039/c3gc40225h
Adams, Joseph P, Alder, Catherine M, Andrews, Ian, Bullion, Ann M, Campbell-Crawford, Matthew, Darcy, Michael G, Hayler, John D, Henderson, Richard K, Oare, Catriona A, Pendrak, Israil, Redman, Anik M, Shuster, Leanna E, Sneddon, Helen F, Walker, Matthew D
Year of Publication 24.05.2013
Year of Publication 24.05.2013
Get full text
Journal Article
Synthesis of structural analogs of leukotriene B4 and their receptor binding activity
Kingsbury, William D, Pendrak, Israil, Leber, Jack D, Boehm, Jeffery C, Mallet, Brenda, Sarau, Henry M, Foley, James J, Schmidt, Dulcie B, Daines, Robert A
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
Get full text
Journal Article
Trisubstituted pyridine leukotriene B4 receptor antagonists: synthesis and structure-activity relationships
Daines, Robert A, Chambers, Pamela A, Pendrak, Israil, Jakas, Dalia R, Sarau, Henry M, Foley, James J, Schmidt, Dulcie B, Kingsbury, William D
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
Get full text
Journal Article
PHARMACEUTICAL COMPOSITION COMPRISING 2-SUBSTITUTED CEPHEM COMPOUND
YAMAWAKI KENJI, REEMA THALGI, SATO ATSUSHI, AOKI TOSHIAKI, YOKOO KATSUMI, ISRAIL PENDRAK, PEARSON NEIL DAVID, KUSANO HIROKI, LIAO XIANGMIN
Year of Publication 10.12.2015
Get full text
Year of Publication 10.12.2015
Patent
Synthesis and Anti-HSV Activity of Methylenedioxy Mappicine Ketone Analogs
Pendrak, Israil, Wittrock, Robert, Kingsbury, William D.
Published in Journal of organic chemistry (01.05.1995)
Published in Journal of organic chemistry (01.05.1995)
Get full text
Journal Article
CRYSTALLINE FORMS OF GEPOTIDACIN
DAVISON, Senthil, DAI, Wenning, WILLIAMS, Glenn Robert, COUCH, Ricky Wayne, PENDRAK, Israil
Year of Publication 01.06.2023
Get full text
Year of Publication 01.06.2023
Patent
CRYSTALLINE FORMS OF GEPOTIDACIN
DAVISON, Senthil, DAI, Wenning, WILLIAMS, Glenn Robert, COUCH, Ricky Wayne, PENDRAK, Israil
Year of Publication 08.03.2023
Get full text
Year of Publication 08.03.2023
Patent
CHEMICAL COMPOUNDS
PERO, Joseph E, EVANS, Karen Anderson, PENDRAK, Israil, DEMARTINO, Michael P
Year of Publication 19.08.2021
Get full text
Year of Publication 19.08.2021
Patent
CHEMICAL COMPOUNDS
PERO, Joseph E, EVANS, Karen Anderson, PENDRAK, Israil, DEMARTINO, Michael P
Year of Publication 19.05.2021
Get full text
Year of Publication 19.05.2021
Patent
CHEMICAL COMPOUNDS
EVANS, KAREN ANDERSON, DEMARTINO, MICHAEL P, PERO, JOSEPH E, PENDRAK, ISRAIL
Year of Publication 16.01.2020
Get full text
Year of Publication 16.01.2020
Patent
CHEMICAL COMPOUNDS
PERO, Joseph E, EVANS, Karen Anderson, PENDRAK, Israil, DEMARTINO, Michael P
Year of Publication 16.01.2020
Get full text
Year of Publication 16.01.2020
Patent
2-SUBSTITUTED CEPHEM COMPOUNDS
THALGI, REEMA, PEARSON, NEIL, DAVID, YAMAWAKI, KENJI, AOKI, TOSHIAKI, KUSANO, HIROKI, YOKOO, KATSUKI, SATO, JUN, LIAO, XIANGMIN, PENDRAK, ISRAIL
Year of Publication 31.08.2020
Get full text
Year of Publication 31.08.2020
Patent