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Harikrishnan, Lalgudi S., Kamau, Muthoni G., Wan, Honghe, Inghrim, Jennifer A., Zimmermann, Kurt, Sang, Xiaopeng, Mastalerz, Harold A., Johnson, Walter L., Zhang, Guifen, Lombardo, Louis J., Poss, Michael A., Trainor, George L., Tokarski, John S., Lorenzi, Matthew V., You, Dan, Gottardis, Marco M., Baldwin, Kathy F., Lippy, Jonathan, Nirschl, David S., Qiu, Ruhui, Miller, Arthur V., Khan, Javed, Sack, John S., Purandare, Ashok V.
Published in Bioorganic & medicinal chemistry letters (01.03.2011)
Published in Bioorganic & medicinal chemistry letters (01.03.2011)
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Silyl-Substituted Spirodiepoxides: Stereoselective Formation and Regioselective Opening
Ghosh, Partha, Cusick, Joseph R, Inghrim, Jennifer, Williams, Lawrence J
Published in Organic letters (15.10.2009)
Published in Organic letters (15.10.2009)
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Discovery of a Highly Selective JAK2 Inhibitor, BMS-911543, for the Treatment of Myeloproliferative Neoplasms
Wan, Honghe, Schroeder, Gretchen M, Hart, Amy C, Inghrim, Jennifer, Grebinski, James, Tokarski, John S, Lorenzi, Matthew V, You, Dan, Mcdevitt, Theresa, Penhallow, Becky, Vuppugalla, Ragini, Zhang, Yueping, Gu, Xiaomei, Iyer, Ramaswamy, Lombardo, Louis J, Trainor, George L, Ruepp, Stefan, Lippy, Jonathan, Blat, Yuval, Sack, John S, Khan, Javed A, Stefanski, Kevin, Sleczka, Bogdan, Mathur, Arvind, Sun, Jung-Hui, Wong, Michael K, Wu, Dauh-Rurng, Li, Peng, Gupta, Anuradha, Arunachalam, P. N, Pragalathan, Bala, Narayanan, Sankara, K.C, Nanjundaswamy, Kuppusamy, Prakasam, Purandare, Ashok V
Published in ACS medicinal chemistry letters (13.08.2015)
Published in ACS medicinal chemistry letters (13.08.2015)
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Spirodiepoxides: Synthesis of Epoxomicinoids
Zhang, Yue, Cusick, Joseph R, Ghosh, Partha, Shangguan, Ning, Katukojvala, Sreenivas, Inghrim, Jennifer, Emge, Thomas J, Williams, Lawrence J
Published in Journal of organic chemistry (16.10.2009)
Published in Journal of organic chemistry (16.10.2009)
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Structure-Based Design of Selective Janus Kinase 2 Imidazo[4,5‑d]pyrrolo[2,3‑b]pyridine Inhibitors
Hart, Amy C, Schroeder, Gretchen M, Wan, Honghe, Grebinski, James, Inghrim, Jennifer, Kempson, James, Guo, Junqing, Pitts, William J, Tokarski, John S, Sack, John S, Khan, Javed A, Lippy, Jonathan, Lorenzi, Matthew V, You, Dan, McDevitt, Theresa, Vuppugalla, Ragini, Zhang, Yueping, Lombardo, Louis J, Trainor, George L, Purandare, Ashok V
Published in ACS medicinal chemistry letters (13.08.2015)
Published in ACS medicinal chemistry letters (13.08.2015)
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Abstract DDT01-03: Discovery of BMS-911543, a highly selective JAK2 inhibitor, as a clinical candidate for the treatment of myeloproliferative disease and other malignancies
Purandare, Ashok V., Wan, Honghe, Schroeder, Gretchen, Hart, Amy, Grebinski, James, Inghrim, Jennifer, Tokarski, John, You, Dan, Penhallow, Becky, McDevitt, Theresa, Vuppugalla, Ragini, Zhang, Yueping, Ruepp, Stefan, Trainor, George, Han, Xia, Lombardo, Louis, Lee, Francis Y., Gottardis, Marco, Hosbach, Jennifer, Fitzpatrick, Elizabeth, Emanuel, Stuart, Pardanani, Animesh, Lasho, Terra L., Tefferi, Ayalew, Lorenzi, Matthew V.
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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Synthesis and Biological Evaluation of Novel Compounds within a Class of 3-Aminochroman Derivatives with Dual 5-HT1A Receptor and Serotonin Transporter Affinity
Hatzenbuhler, Nicole T, Evrard, Deborah A, Harrison, Boyd L, Huryn, Donna, Inghrim, Jennifer, Kraml, Christina, Mattes, James F, Mewshaw, Richard E, Zhou, Dahui, Hornby, Geoffrey, Lin, Qian, Smith, Deborah L, Sullivan, Kelly M, Schechter, Lee E, Beyer, Chad E, Andree, Terrance H
Published in Journal of medicinal chemistry (27.07.2006)
Published in Journal of medicinal chemistry (27.07.2006)
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Pyrrolo[1,2-f]triazines as JAK2 inhibitors: Achieving potency and selectivity for JAK2 over JAK3 Purandare
Harikrishnan, Lalgudi S, Kamau, Muthoni G, Wan, Honghe, Inghrim, Jennifer A, Zimmermann, Kurt, Sang, Xiaopeng, Mastalerz, Harold A, Johnson, Walter L, Zhang, Guifen, Lombardo, Louis J, Poss, Michael A, Trainor, George L, Tokarski, John S, Lorenzi, Matthew V, You, Dan, Gottardis, Marco M, Baldwin, Kathy F, Lippy, Jonathan, Nirschl, David S, Qiu, Ruhui
Published in Bioorganic & medicinal chemistry letters (01.03.2011)
Published in Bioorganic & medicinal chemistry letters (01.03.2011)
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JAK2 INHIBITORS AND THEIR USE FOR THE TREATMENT OF MYELOPROLIFERATIVE DISEASES AND CANCER
HART AMY, SCHROEDER GRETCHEN, INGHRIM JENNIFER, GREBINSKI JAMES W, PURANDARE ASHOK V, WAN HONGHE
Year of Publication 13.06.2012
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Year of Publication 13.06.2012
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IMIDAZOTRIAZINECARBONITRILES USEFUL AS KINASE INHIBITORS
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Year of Publication 01.06.2015
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Year of Publication 01.06.2015
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Synthesis and Biological Evaluation of Novel Compounds within a Class of 3-Aminochroman Derivatives with Dual 5-HT 1A Receptor and Serotonin Transporter Affinity
Hatzenbuhler, Nicole T., Evrard, Deborah A., Harrison, Boyd L., Huryn, Donna, Inghrim, Jennifer, Kraml, Christina, Mattes, James F., Mewshaw, Richard E., Zhou, Dahui, Hornby, Geoffrey, Lin, Qian, Smith, Deborah L., Sullivan, Kelly M., Schechter, Lee E., Beyer, Chad E., Andree, Terrance H.
Published in Journal of medicinal chemistry (01.07.2006)
Published in Journal of medicinal chemistry (01.07.2006)
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JAK2 INHIBITORS AND THEIR USE FOR THE TREATMENT OF MYELOPROLIFERATIVE DISEASES AND CANCER
WAN, HONGHE, INGHRIM, JENNIFER, HART, AMY, GREBINSKI, JAMES W, PURANDARE, ASHOK V, SCHROEDER, GRETCHEN
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Year of Publication 19.09.2017
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JAK2 inhibitors and their use for the treatment of myeloproliferative diseases and cancer
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Year of Publication 14.04.2016
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inibidores de jak2 e seu uso para o tratamento de doenças mieloproliferativas e câncer
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Year of Publication 12.04.2016
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Year of Publication 12.04.2016
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IDO inhibitors
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Year of Publication 19.09.2017
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Inibitori di jak2 e loro uso per il trattamento del cancro e di malattie mieloproliferative
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Year of Publication 15.01.2015
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JAK2 INHIBITORS AND THEIR USE FOR THE TREATMENT OF MYELOPROLIFERATIVE DISEASES AND CANCER
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Year of Publication 28.11.2014
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Year of Publication 28.11.2014
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JAK2 INHIBITORS AND THEIR USE FOR THE TREATMENT OF MYELOPROLIFERATIVE DISEASES AND CANCER
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Year of Publication 30.10.2014
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Year of Publication 30.10.2014
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JAK-2-HÆMMERE OG ANVENDELSE HERAF TIL BEHANDLING AF MYELOPROLIFERATIVESYGDOMME OG CANCER
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Year of Publication 20.10.2014
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Year of Publication 20.10.2014
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