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Published in Bioorganic & medicinal chemistry letters (01.01.2019)
Published in Bioorganic & medicinal chemistry letters (01.01.2019)
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Synthesis and Biological Activity of Various Derivatives of a Novel Class of Potent, Selective, and Orally Active Prostaglandin D2 Receptor Antagonists. 2. 6,6-Dimethylbicyclo[3.1.1]heptane Derivatives
Mitsumori, Susumu, Tsuri, Tatsuo, Honma, Tsunetoshi, Hiramatsu, Yoshiharu, Okada, Toshihiko, Hashizume, Hiroshi, Kida, Shiro, Inagaki, Masanao, Arimura, Akinori, Yasui, Kiyoshi, Asanuma, Fujio, Kishino, Junji, Ohtani, Mitsuaki
Published in Journal of medicinal chemistry (05.06.2003)
Published in Journal of medicinal chemistry (05.06.2003)
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Total synthesis of discorhabdin C: a general aza spiro dienone formation from O-silylated phenol derivatives using a hypervalent iodine reagent
Kita, Yasuyuki, Tohma, Hirofumi, Inagaki, Masanao, Hatanaka, Kenji, Yakura, Takayuki
Published in Journal of the American Chemical Society (01.03.1992)
Published in Journal of the American Chemical Society (01.03.1992)
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Total Synthesis of Terprenin, a Highly Potent and Novel Immunoglobulin E Antibody Suppressant
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Published in Angewandte Chemie (International ed.) (20.04.1998)
Published in Angewandte Chemie (International ed.) (20.04.1998)
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Discovery of S-777469: An orally available CB2 agonist as an antipruritic agent
Odan, Masahide, Ishizuka, Natsuki, Hiramatsu, Yoshiharu, Inagaki, Masanao, Hashizume, Hiroshi, Fujii, Yasuhiko, Mitsumori, Susumu, Morioka, Yasuhide, Soga, Masahiko, Deguchi, Masashi, Yasui, Kiyoshi, Arimura, Akinori
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
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Discovery of S-444823, a potent CB1/CB2 dual agonist as an antipruritic agent
Odan, Masahide, Ishizuka, Natsuki, Hiramatsu, Yoshiharu, Inagaki, Masanao, Hashizume, Hiroshi, Fujii, Yasuhiko, Mitsumori, Susumu, Morioka, Yasuhide, Soga, Masahiko, Deguchi, Masashi, Yasui, Kiyoshi, Arimura, Akinori
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
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CB 1/2 dual agonists with 3-carbamoyl 2-pyridone derivatives as antipruritics: Reduction of CNS side effects by introducing polar functional groups
Odan, Masahide, Ishizuka, Natsuki, Hiramatsu, Yoshiharu, Inagaki, Masanao, Hashizume, Hiroshi, Fujii, Yasuhiko, Mitsumori, Susumu, Morioka, Yasuhide, Soga, Masahiko, Deguchi, Masashi, Yasui, Kiyoshi, Arimura, Akinori
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
Published in Bioorganic & medicinal chemistry letters (15.04.2012)
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HETEROCYCLIC DERIVATIVE HAVING TrkA-INHIBITING ACTIVITY
INAGAKI, Masanao, NAKAMURA, Kenichiroh, FUJIU, Motohiro, YUKIMASA, Akira, YAMAGUCHI, Hiroki, HATA, Kayoko, INOUE, Takatsugu, KANO, Kazuya
Year of Publication 12.01.2017
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Year of Publication 12.01.2017
Patent
Novel Antiarthritic Agents with 1,2-Isothiazolidine-1,1-dioxide (γ-Sultam) Skeleton: Cytokine Suppressive Dual Inhibitors of Cyclooxygenase-2 and 5-Lipoxygenase
Inagaki, Masanao, Tsuri, Tatsuo, Jyoyama, Hirokuni, Ono, Takashi, Yamada, Katsutoshi, Kobayashi, Mika, Hori, Yozo, Arimura, Akinori, Yasui, Kiyoshi, Ohno, Kouji, Kakudo, Shinji, Koizumi, Kenzo, Suzuki, Ryuji, Kato, Miyako, Kawai, Shinichi, Matsumoto, Saichi
Published in Journal of medicinal chemistry (18.05.2000)
Published in Journal of medicinal chemistry (18.05.2000)
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CRYSTAL OF 6,7-UNSATURATED-7-CARBAMOYL MORPHINAN DERIVATIVE, AND METHOD FOR PRODUCING THE SAME
NOGUCHI KOUICHI, INAGAKI MASANAO, TAMURA YOSHINORI, OMURA SOHEI, HAGA NOBUHIRO, MORIMOTO KENJI, ODA SHINICHI
Year of Publication 12.05.2014
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Year of Publication 12.05.2014
Patent
Synthesis and Biological Activity of Various Derivatives of a Novel Class of Potent, Selective, and Orally Active Prostaglandin D2 Receptor Antagonists. 1. Bicyclo[2.2.1]heptane Derivatives
Mitsumori, Susumu, Tsuri, Tatsuo, Honma, Tsunetoshi, Hiramatsu, Yoshiharu, Okada, Toshihiko, Hashizume, Hiroshi, Inagaki, Masanao, Arimura, Akinori, Yasui, Kiyoshi, Asanuma, Fujio, Kishino, Junji, Ohtani, Mitsuaki
Published in Journal of medicinal chemistry (05.06.2003)
Published in Journal of medicinal chemistry (05.06.2003)
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Journal Article
Synthesis and biological activity of various derivatives of a novel class of potent, selective, and orally active prostaglandin D-2 receptor antagonists. 2. 6,6-dimethylbicyclo[3.1.1]heptane derivatives
Mitsumori, S, Tsuri, T, Honma, T, Hiramatsu, Y, Okada, T, Hashizume, H, Kida, S, Inagaki, M, Arimura, A, Yasui, M, Asanuma, F, Kishino, J, Ohtani, M
Published in Journal of medicinal chemistry (05.06.2003)
Published in Journal of medicinal chemistry (05.06.2003)
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Journal Article
CRYSTALLINE 6,7-UNSATURATED-7-CARBAMOYL MORPHINANE DERIVATIVE, AND METHOD FOR PRODUCING SAME
NOGUCHI KOUICHI, INAGAKI MASANAO, TAMURA YOSHINORI, OMURA SOHEI, HAGA NOBUHIRO, MORIMOTO KENJI, ODA SHINICHI
Year of Publication 05.11.2013
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Year of Publication 05.11.2013
Patent