Tetracyclic indole inhibitors of hepatitis C virus NS5B-polymerase
Stansfield, Ian, Ercolani, Caterina, Mackay, Angela, Conte, Immacolata, Pompei, Marco, Koch, Uwe, Gennari, Nadia, Giuliano, Claudio, Rowley, Michael, Narjes, Frank
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
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Journal Article
Unusual Father-to-Daughter Transmission of Incontinentia Pigmenti Due to Mosaicism in IP Males
Fusco, Francesca, Conte, Matilde Immacolata, Diociaiuti, Andrea, Bigoni, Stefania, Branda, Maria Francesca, Ferlini, Alessandra, El Hachem, Maya, Ursini, Matilde Valeria
Published in Pediatrics (Evanston) (01.09.2017)
Published in Pediatrics (Evanston) (01.09.2017)
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Journal Article
Development of carboxylic acid replacements in indole- N-acetamide inhibitors of hepatitis C virus NS5B polymerase
Stansfield, Ian, Pompei, Marco, Conte, Immacolata, Ercolani, Caterina, Migliaccio, Giovanni, Jairaj, Mark, Giuliano, Claudio, Rowley, Michael, Narjes, Frank
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
Published in Bioorganic & medicinal chemistry letters (15.09.2007)
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Journal Article
Identification of thieno[3,2- b]pyrroles as allosteric inhibitors of hepatitis C virus NS5B polymerase
Ontoria, Jesus M., Martìn Hernando, Jose I., Malancona, Savina, Attenni, Barbara, Stansfield, Ian, Conte, Immacolata, Ercolani, Caterina, Habermann, Jörg, Ponzi, Simona, Di Filippo, Marcello, Koch, Uwe, Rowley, Michael, Narjes, Frank
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
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Journal Article
Development of a Scalable Chiral Synthesis of MK-3281, an Inhibitor of the Hepatitis C Virus NS5B Polymerase
Colarusso, Stefania, Conte, Immacolata, Di Filippo, Marcello, Ercolani, Caterina, Mackay, Angela C., Palumbi, Maria Cecilia, Ferreira, Maria del Rosario Rico, Stansfield, Ian, Zaramella, Simone, Narjes, Frank, Habermann, Joerg
Published in Synlett (01.07.2011)
Published in Synlett (01.07.2011)
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Journal Article
The Design and Enzyme-Bound Crystal Structure of Indoline Based Peptidomimetic Inhibitors of Hepatitis C Virus NS3 Protease
Ontoria, Jesus M, Di Marco, Stefania, Conte, Immacolata, Di Francesco, M. Emilia, Gardelli, Cristina, Koch, Uwe, Matassa, Victor G, Poma, Marco, Steinkühler, Christian, Volpari, Cinzia, Harper, Steven
Published in Journal of medicinal chemistry (16.12.2004)
Published in Journal of medicinal chemistry (16.12.2004)
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Journal Article
The aporetic dialogues of Modena on gender differences: Is it all about testosterone? EPISODE I: CRIME
Brigante, Giulia, D'Angelo, Giulia, Caccin, Vanessa, Coluccia, Silvia, Conte, Immacolata, Demichelis, Veronica Maria, Cecchi, Rossana, Simoni, Manuela
Published in Andrology (Oxford) (07.11.2024)
Published in Andrology (Oxford) (07.11.2024)
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Journal Article
SAR evolution towards potent C-terminal carboxamide peptide inhibitors of Zika virus NS2B-NS3 protease
Colarusso, Stefania, Ferrigno, Federica, Ponzi, Simona, Pavone, Francesca, Conte, Immacolata, Abate, Luigi, Beghetto, Elisa, Missineo, Antonino, Amaudrut, Jerome, Bresciani, Alberto, Paonessa, Giacomo, Tomei, Licia, Montalbetti, Christian, Bianchi, Elisabetta, Toniatti, Carlo, Ontoria, Jesus M.
Published in Bioorganic & medicinal chemistry (01.03.2022)
Published in Bioorganic & medicinal chemistry (01.03.2022)
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Journal Article
Discovery of (7 R )-14-Cyclohexyl-7-{[2-(dimethylamino)ethyl](methyl) amino}-7,8-dihydro-6 H -indolo[1,2- e ][1,5]benzoxazocine-11-carboxylic Acid (MK-3281), a Potent and Orally Bioavailable Finger-Loop Inhibitor of the Hepatitis C Virus NS5B Polymerase
Narjes, Frank, Crescenzi, Benedetta, Ferrara, Marco, Habermann, Jörg, Colarusso, Stefania, del Rosario Rico Ferreira, Maria, Stansfield, Ian, Mackay, Angela Claire, Conte, Immacolata, Ercolani, Caterina, Zaramella, Simone, Palumbi, Maria-Cecilia, Meuleman, Philip, Leroux-Roels, Geert, Giuliano, Claudio, Fiore, Fabrizio, Di Marco, Stefania, Baiocco, Paola, Koch, Uwe, Migliaccio, Giovanni, Altamura, Sergio, Laufer, Ralph, De Francesco, Raffaele, Rowley, Michael
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
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Journal Article
Discovery of (7R)-14-Cyclohexyl-7-{[2-(dimethylamino)ethyl](methyl) amino}-7,8-dihydro-6H-indolo[1,2-e][1,5]benzoxazocine-11-carboxylic Acid (MK-3281), a Potent and Orally Bioavailable Finger-Loop Inhibitor of the Hepatitis C Virus NS5B Polymerase
Narjes, Frank, Crescenzi, Benedetta, Ferrara, Marco, Habermann, Jörg, Colarusso, Stefania, del Rosario Rico Ferreira, Maria, Stansfield, Ian, Mackay, Angela Claire, Conte, Immacolata, Ercolani, Caterina, Zaramella, Simone, Palumbi, Maria-Cecilia, Meuleman, Philip, Leroux-Roels, Geert, Giuliano, Claudio, Fiore, Fabrizio, Di Marco, Stefania, Baiocco, Paola, Koch, Uwe, Migliaccio, Giovanni, Altamura, Sergio, Laufer, Ralph, De Francesco, Raffaele, Rowley, Michael
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
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Journal Article
Synthesis and SAR of piperazinyl- N-phenylbenzamides as inhibitors of hepatitis C virus RNA replication in cell culture
Conte, Immacolata, Giuliano, Claudio, Ercolani, Caterina, Narjes, Frank, Koch, Uwe, Rowley, Michael, Altamura, Sergio, Francesco, Raffaele De, Neddermann, Petra, Migliaccio, Giovanni, Stansfield, Ian
Published in Bioorganic & medicinal chemistry letters (15.03.2009)
Published in Bioorganic & medicinal chemistry letters (15.03.2009)
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Journal Article
2-(2-Thienyl)-5,6-dihydroxy-4-carboxypyrimidines as Inhibitors of the Hepatitis C Virus NS5B Polymerase: Discovery, SAR, Modeling, and Mutagenesis
Koch, Uwe, Attenni, Barbara, Malancona, Savina, Colarusso, Stefania, Conte, Immacolata, Di Filippo, Marcello, Harper, Steven, Pacini, Barbara, Giomini, Claudia, Thomas, Steven, Incitti, Ilario, Tomei, Licia, De Francesco, Raffaele, Altamura, Sergio, Matassa, Victor G, Narjes, Frank
Published in Journal of medicinal chemistry (09.03.2006)
Published in Journal of medicinal chemistry (09.03.2006)
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Journal Article
EDA-ID and IP, Two Faces of the Same Coin: How the Same IKBKG/NEMO Mutation Affecting the NF-κB Pathway Can Cause Immunodeficiency and/or Inflammation
Fusco, Francesca, Pescatore, Alessandra, Conte, Matilde Immacolata, Mirabelli, Peppino, Paciolla, Mariateresa, Esposito, Elio, Lioi, Maria Brigida, Ursini, Matilde Valeria
Published in International reviews of immunology (01.01.2015)
Published in International reviews of immunology (01.01.2015)
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Journal Article
Incontinentia pigmenti: report on data from 2000 to 2013
Fusco, Francesca, Paciolla, Mariateresa, Conte, Matilde Immacolata, Pescatore, Alessandra, Esposito, Elio, Mirabelli, Peppino, Lioi, Maria Brigida, Ursini, Matilde Valeria
Published in Orphanet journal of rare diseases (24.06.2014)
Published in Orphanet journal of rare diseases (24.06.2014)
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Journal Article
Insight into IKBKG/NEMO Locus: Report of New Mutations and Complex Genomic Rearrangements Leading to Incontinentia Pigmenti Disease
Conte, Matilde Immacolata, Pescatore, Alessandra, Paciolla, Mariateresa, Esposito, Elio, Miano, Maria Giuseppina, Lioi, Maria Brigida, McAleer, Maeve A., Giardino, Giuliana, Pignata, Claudio, Irvine, Alan D., Scheuerle, Angela E., Royer, Ghislaine, Hadj-Rabia, Smail, Bodemer, Christine, Bonnefont, Jean-Paul, Munnich, Arnold, Smahi, Asma, Steffann, Julie, Fusco, Francesca, Ursini, Matilde Valeria
Published in Human mutation (01.02.2014)
Published in Human mutation (01.02.2014)
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Journal Article
Evolution, synthesis and SAR of tripeptide α-ketoacid Inhibitors of the hepatitis C virus NS3/NS4A serine protease
Colarusso, Stefania, Gerlach, Benjamin, Koch, Uwe, Muraglia, Ester, Conte, Immacolata, Stansfield, Ian, Matassa, Victor G, Narjes, Frank
Published in Bioorganic & medicinal chemistry letters (25.02.2002)
Published in Bioorganic & medicinal chemistry letters (25.02.2002)
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Journal Article
B cells from nuclear factor kB essential modulator deficient patients fail to differentiate to antibody secreting cells in response to TLR9 ligand
Giardino, Giuliana, Cirillo, Emilia, Gallo, Vera, Esposito, Tiziana, Fusco, Francesca, Conte, Matilde Immacolata, Quinti, Isabella, Ursini, Matilde Valeria, Carsetti, Rita, Pignata, Claudio
Published in Clinical immunology (Orlando, Fla.) (01.12.2015)
Published in Clinical immunology (Orlando, Fla.) (01.12.2015)
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Journal Article
Rare Mendelian Primary Immunodeficiency diseases associated to impaired NF-κB signaling
Paciolla, Mariateresa, Pescatore, Alessandra, Conte, Matilde Immacolata, Esposito, Elio, Incoronato, Mariarosaria, Lioi, Maria Brigida, Fusco, Francesca, Ursini, Matilde Valeria
Published in Genes and immunity (12.03.2015)
Published in Genes and immunity (12.03.2015)
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Journal Article
Cyclic polypeptides for PCSK9 inhibition
Costantini, Willy, Tucker, Thomas Joseph, Embrey, Mark W, Boyer, Nicolas Cedric, Ingenito, Raffaele, Conte, Immacolata, Xiong, Yusheng, Santoprete, Alessia, Colarusso, Stefania, Ricardo, Alonso, Kerekes, Angela Dawn, LaPlaca, Derek M, Shahripour, Aurash, Wu, Chengwei, Bianchi, Elisabetta, Branca, Danila, Stringer, Joseph R, Gilbert, Eric J, Costante, Roberto, Ha, Sookhee Nicole, Youm, Hyewon
Year of Publication 18.06.2024
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Year of Publication 18.06.2024
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