Highly Regioselective Nucleophilic Carbon−Carbon Bond Formation on Furans and Thiophenes Initiated by Pummerer-Type Reaction
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Published in Organic letters (14.10.2004)
Published in Organic letters (14.10.2004)
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Regioselective, nucleophilic carbon–carbon bond formation at the C4-position of indoles initiated by the aromatic Pummerer-type reaction
Akai, Shuji, Kawashita, Norihito, Wada, Yasufumi, Satoh, Hideharu, Alinejad, Anahita Hessamian, Kakiguchi, Keisuke, Kuriwaki, Ikumi, Kita, Yasuyuki
Published in Tetrahedron letters (20.03.2006)
Published in Tetrahedron letters (20.03.2006)
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Discovery of ASP5878: Synthesis and structure–activity relationships of pyrimidine derivatives as pan-FGFRs inhibitors with improved metabolic stability and suppressed hERG channel inhibitory activity
Kuriwaki, Ikumi, Kameda, Minoru, Iikubo, Kazuhiko, Hisamichi, Hiroyuki, Kawamoto, Yuichiro, Kikuchi, Shigetoshi, Moritomo, Hiroyuki, Terasaka, Tadashi, Iwai, Yoshinori, Noda, Atsushi, Tomiyama, Hiroshi, Kikuchi, Aya, Hirano, Masaaki
Published in Bioorganic & medicinal chemistry (01.04.2022)
Published in Bioorganic & medicinal chemistry (01.04.2022)
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Structure-based drug design of 1,3,5-triazine and pyrimidine derivatives as novel FGFR3 inhibitors with high selectivity over VEGFR2
Kuriwaki, Ikumi, Kameda, Minoru, Hisamichi, Hiroyuki, Kikuchi, Shigetoshi, Iikubo, Kazuhiko, Kawamoto, Yuichiro, Moritomo, Hiroyuki, Kondoh, Yutaka, Amano, Yasushi, Tateishi, Yukihiro, Echizen, Yuka, Iwai, Yoshinori, Noda, Atsushi, Tomiyama, Hiroshi, Suzuki, Tomoyuki, Hirano, Masaaki
Published in Bioorganic & medicinal chemistry (15.05.2020)
Published in Bioorganic & medicinal chemistry (15.05.2020)
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Synthesis and structure-activity relationships of pyrimidine derivatives as potent and orally active FGFR3 inhibitors with both increased systemic exposure and enhanced in vitro potency
Kuriwaki, Ikumi, Kameda, Minoru, Iikubo, Kazuhiko, Hisamichi, Hiroyuki, Kawamoto, Yuichiro, Kikuchi, Shigetoshi, Moritomo, Hiroyuki, Kondoh, Yutaka, Terasaka, Tadashi, Amano, Yasushi, Tateishi, Yukihiro, Echizen, Yuka, Iwai, Yoshinori, Noda, Atsushi, Tomiyama, Hiroshi, Nakazawa, Taisuke, Hirano, Masaaki
Published in Bioorganic & medicinal chemistry (01.03.2021)
Published in Bioorganic & medicinal chemistry (01.03.2021)
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Journal Article
Total Synthesis of (±)-γ-Rubromycin on the Basis of Two Aromatic Pummerer-Type Reactions
Akai, Shuji, Kakiguchi, Keisuke, Nakamura, Yuka, Kuriwaki, Ikumi, Dohi, Toshifumi, Harada, Shusaku, Kubo, Ozora, Morita, Nobuyoshi, Kita, Yasuyuki
Published in Angewandte Chemie (International ed.) (01.01.2007)
Published in Angewandte Chemie (International ed.) (01.01.2007)
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ARYL ALKYNAMIDE DERIVATIVES
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Year of Publication 18.01.2024
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ARYL ALKYNAMIDE DERIVATIVES
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4-AMINOQUINAZOLINE COMPOUND
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4-AMINOQUINAZOLINE COMPOUND
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Year of Publication 20.12.2023
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BICYCLIC 1,4-DIAZEPANONES AND THERAPEUTIC USES THEREOF
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Year of Publication 07.11.2024
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Year of Publication 07.11.2024
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4-AMINOQUINAZOLINE COMPOUNDS
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Year of Publication 29.05.2024
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Bicyclic 1,4-diazepanones and therapeutic uses thereof
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WASHIO, Takuya, KOIZUMI, Yuka, KURAMOTO, Kazuyuki, YAMAKI, Susumu, TOMIYAMA, Hiroshi, INAGAKI, Yusuke, KOIKE, Takanori, MAEDA, Junko, NAKAMURA, Akihiko, TOYA, Hiroki, KURIWAKI, Ikumi, IWAI, Yoshinori, SABA, Kengo, YAMASHITA, Yumi, KAMIKUBO, Takashi
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Yamaki, Susumu, Iida, Maiko, Kuriwaki, Ikumi, Kamikubo, Takashi, Koizumi, Yuka, Maeda, Junko, Saba, Kengo, Inagaki, Yusuke, Koike, Takanori, Negoro, Kenji, Nigawara, Takahiro, Shishikura, Junichi
Year of Publication 06.04.2023
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Year of Publication 06.04.2023
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Annulated pyridazine compound
KOIZUMI Yuka, YAMASHITA Yumi, IWAI Yoshinori, KURIWAKI Ikumi, MAEDA Junko, KOIKE Takanori, TOMIYAMA Hiroshi, WASHIO Takuya, SABA Kengo, KAMIKUBO Takashi, KURAMOTO Kazuyuki, TOYA Hiroki, INAGAKI Yusuke, NAKAMURA Akihiko, YAMAKI Susumu
Year of Publication 01.03.2024
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Year of Publication 01.03.2024
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