Open Innovation and Drug Discovery Ecosystem
Ikeura, Yoshinori
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
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Journal Article
Axially Chiral 1,7-Naphthyridine-6-carboxamide Derivatives as Orally Active Tachykinin NK1 Receptor Antagonists: Synthesis, Antagonistic Activity, and Effects on Bladder Functions
Natsugari, Hideaki, Ikeura, Yoshinori, Kamo, Izumi, Ishimaru, Takenori, Ishichi, Yuji, Fujishima, Akira, Tanaka, Toshimasa, Kasahara, Fumiko, Kawada, Mitsuru, Doi, Takayuki
Published in Journal of medicinal chemistry (23.09.1999)
Published in Journal of medicinal chemistry (23.09.1999)
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Journal Article
Effects of TAK-637, a Novel Neurokinin-1 Receptor Antagonist, on Colonic Function in Vivo
Okano, S, Nagaya, H, Ikeura, Y, Natsugari, H, Inatomi, N
Published in The Journal of pharmacology and experimental therapeutics (01.08.2001)
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Published in The Journal of pharmacology and experimental therapeutics (01.08.2001)
Journal Article
Synthesis and structure activity relationship studies of benzothieno[3,2-b]furan derivatives as a novel class of IKKbeta inhibitors
Sugiyama, Hideyuki, Yoshida, Masato, Mori, Kouji, Kawamoto, Tomohiro, Sogabe, Satoshi, Takagi, Terufumi, Oki, Hideyuki, Tanaka, Toshimasa, Kimura, Hiroyuki, Ikeura, Yoshinori
Published in Chemical & pharmaceutical bulletin (2007)
Published in Chemical & pharmaceutical bulletin (2007)
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Journal Article
Axially Chiral N-Benzyl-N,7-dimethyl-5-phenyl-1,7-naphthyridine-6-carboxamide Derivatives as Tachykinin NK1 Receptor Antagonists: Determination of the Absolute Stereochemical Requirements
Ikeura, Yoshinori, Ishichi, Yuji, Tanaka, Toshimasa, Fujishima, Akira, Murabayashi, Mika, Kawada, Mitsuru, Ishimaru, Takenori, Kamo, Izumi, Doi, Takayuki, Natsugari, Hideaki
Published in Journal of medicinal chemistry (22.10.1998)
Published in Journal of medicinal chemistry (22.10.1998)
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Journal Article
Enantioselective synthesis of an axially chiral 1,7-naphthyridine-6-carboxamide derivative having potent antagonist activity at the NK1 receptor
Ikeura, Y, Ishimaru, T, Doi, T, Kawada, M, Fujishima, A, Natsugari, H
Published in Chemical communications (Cambridge, England) (1998)
Published in Chemical communications (Cambridge, England) (1998)
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Journal Article
Novel, Potent, and Orally Active Substance P Antagonists: Synthesis and Antagonist Activity of N-Benzylcarboxamide Derivatives of Pyrido[3,4-b]pyridine
Natsugari, Hideaki, Ikeura, Yoshinori, Kiyota, Yutaka, Ishichi, Yuji, Ishimaru, Takenori, Saga, Osamu, Shirafuji, Hideo, Tanaka, Toshimasa, Kamo, Izumi
Published in Journal of medicinal chemistry (01.08.1995)
Published in Journal of medicinal chemistry (01.08.1995)
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Journal Article
Effects of TAK-637, a tachykinin receptor antagonist, on lower urinary tract function in the guinea pig
Doi, Takayuki, Kamo, Izumi, Imai, Shigemitsu, Okanishi, Satoshi, Ishimaru, Takenori, Ikeura, Yoshinori, Natsugari, Hideaki
Published in European journal of pharmacology (03.11.1999)
Published in European journal of pharmacology (03.11.1999)
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Journal Article
Retraction notice to “3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis” [Bioorg. Med. Chem. 19 (2011) 5175–5182]
Shirai, Junya, Nakamura, Minoru, Tarui, Naoki, Hashimoto, Tadatoshi, Ikeura, Yoshinori
Published in Bioorganic & medicinal chemistry (01.01.2015)
Published in Bioorganic & medicinal chemistry (01.01.2015)
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Journal Article
Retraction notice to ‘Corrigendum to “3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis”’ [Bioorg. Med. Chem. 20 (2012) 5668–5668]
Shirai, Junya, Yamaoka, Masayoshi, Imamiya, Eikoh, Nakamura, Minoru, Tarui, Naoki, Hashimoto, Tadatoshi, Ikeura, Yoshinori
Published in Bioorganic & medicinal chemistry (01.12.2014)
Published in Bioorganic & medicinal chemistry (01.12.2014)
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Journal Article
헤테로시클릭 화합물
IKEURA YOSHINORI, YOSHIDA YOSHINORI, NARA HIROSHI, KAIEDA AKIRA, KONDO SHIGERU, MIKI KENJI
Year of Publication 11.12.2020
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Year of Publication 11.12.2020
Patent
Corrigendum to “Design, structure–activity relationship, and highly efficient asymmetric synthesis of 3-phenyl-4-benzylaminopiperidine derivatives as novel neurokinin-1 receptor antagonists” [Bioorg. Med. Chem. 19 (2011) 6430–6446]
Shirai, Junya, Yoshikawa, Takeshi, Yamashita, Masayuki, Yamamoto, Yasuharu, Kawamoto, Makiko, Tarui, Naoki, Kamo, Izumi, Hashimoto, Tadatoshi, Ikeura, Yoshinori
Published in Bioorganic & medicinal chemistry (01.04.2014)
Published in Bioorganic & medicinal chemistry (01.04.2014)
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Journal Article
HETEROCYCLIC COMPOUND
KONDO, Shigeru, IKEURA, Yoshinori, YOSHIDA, Yoshinori, NARA, Hiroshi, MIKI, Kenji, KAIEDA, Akira
Year of Publication 03.10.2019
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Year of Publication 03.10.2019
Patent
RETRACTED: Corrigendum to “3-Benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis” [Bioorg. Med. Chem. 19 (2011) 5175–5182]
Shirai, Junya, Yamaoka, Masayoshi, Imamiya, Eikoh, Nakamura, Minoru, Tarui, Naoki, Hashimoto, Tadatoshi, Ikeura, Yoshinori
Published in Bioorganic & medicinal chemistry (15.09.2012)
Published in Bioorganic & medicinal chemistry (15.09.2012)
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