Novel Protein Kinase Inhibitors: SMART Drug Design Technology
Sawyer, Tomi K, Bohacek, Regine S, III, Chester A. Metcalf, Shakespeare, William C, Wang, Yihan, Sundaramoorthi, Raji, Keenan, Terence, Narula, Surinder, Weigele, Manfred, Dalgarno, David C
Published in BioTechniques (01.06.2003)
Published in BioTechniques (01.06.2003)
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Journal Article
AP24534, a Pan-BCR-ABL Inhibitor for Chronic Myeloid Leukemia, Potently Inhibits the T315I Mutant and Overcomes Mutation-Based Resistance
O'Hare, Thomas, Shakespeare, William C., Zhu, Xiaotian, Eide, Christopher A., Rivera, Victor M., Wang, Frank, Adrian, Lauren T., Zhou, Tianjun, Huang, Wei-Sheng, Xu, Qihong, Metcalf, Chester A., Tyner, Jeffrey W., Loriaux, Marc M., Corbin, Amie S., Wardwell, Scott, Ning, Yaoyu, Keats, Jeffrey A., Wang, Yihan, Sundaramoorthi, Raji, Thomas, Mathew, Zhou, Dong, Snodgrass, Joseph, Commodore, Lois, Sawyer, Tomi K., Dalgarno, David C., Deininger, Michael W.N., Druker, Brian J., Clackson, Tim
Published in Cancer cell (06.11.2009)
Published in Cancer cell (06.11.2009)
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Identification of Src-specific phosphorylation site on focal adhesion kinase: Dissection of the role of Src SH2 and catalytic functions and their consequences for tumor cell behavior
BRUNTON, Valerie G, AVIZIENYTE, Egle, FINCHAM, Valerie J, SERRELS, Bryan, METCALF, Chester A, SAWYER, Tomi K, FRAME, Margaret C
Published in Cancer research (Chicago, Ill.) (15.02.2005)
Published in Cancer research (Chicago, Ill.) (15.02.2005)
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Journal Article
Activity of Dual SRC-ABL Inhibitors Highlights the Role of BCR/ABL Kinase Dynamics in Drug Resistance
Azam, Mohammad, Nardi, Valentina, Shakespeare, William C., Metcalf, Chester A., Bohacek, Regine S., Wang, Yihan, Sundaramoorthi, Raji, Sliz, Piotr, Veach, Darren R., Bornmann, William G., Clarkson, Bayard, Dalgarno, David C., Sawyer, Tomi K., Daley, George Q.
Published in Proceedings of the National Academy of Sciences - PNAS (13.06.2006)
Published in Proceedings of the National Academy of Sciences - PNAS (13.06.2006)
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Journal Article
Antiangiogenic and antitumor effects of src inhibition in ovarian carcinoma
HAN, Liz Y, LANDEN, Charles N, SHAKESPEARE, William C, YIHAN WANG, SUNDARAMOORTH, Raji, METCALF, Chester A, DALGARNO, David C, SAWYER, Tomi K, GALLICK, Gary E, SOOD, Anil K, TREVINO, Jose G, HALDER, Jyotsnabaran, LIN, Yvonne G, KAMAT, Aparna A, KIM, Tae-Jin, MERRITT, William M, COLEMAN, Robert L, GERSHENSON, David M
Published in Cancer research (Chicago, Ill.) (01.09.2006)
Published in Cancer research (Chicago, Ill.) (01.09.2006)
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Journal Article
AP23846, a novel and highly potent Src family kinase inhibitor, reduces vascular endothelial growth factor and interleukin-8 expression in human solid tumor cell lines and abrogates downstream angiogenic processes
Summy, Justin M, Trevino, Jose G, Lesslie, Donald P, Baker, Cheryl H, Shakespeare, William C, Wang, Yihan, Sundaramoorthi, Raji, Metcalf, 3rd, Chester A, Keats, Jeffrey A, Sawyer, Tomi K, Gallick, Gary E
Published in Molecular cancer therapeutics (01.12.2005)
Published in Molecular cancer therapeutics (01.12.2005)
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Journal Article
Src Inhibitors in Metastatic Bone Disease
Boyce, Brendan F, Xing, Lianping, Yao, Zhenqiang, Yamashita, Teruhito, Shakespeare, William C, Wang, Yihan, Metcalf, 3rd, Chester A, Sundaramoorthi, Raji, Dalgarno, David C, Iuliucci, John D, Sawyer, Tomi K
Published in Clinical cancer research (15.10.2006)
Published in Clinical cancer research (15.10.2006)
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Journal Article
Conference Proceeding
Future Anti-Catabolic Therapeutic Targets in Bone Disease
BOYCE, BRENDAN F., XING, LIANPING, YAO, ZHENQIANG, SHAKESPEARE, WILLIAM C., WANG, YIHAN, METCALF III, CHESTER A., SUNDARAMOORTHI, RAJI, DALGARNO, DAVID C., IULIUCCI, JOHN D., SAWYER, TOMI K.
Published in Annals of the New York Academy of Sciences (01.04.2006)
Published in Annals of the New York Academy of Sciences (01.04.2006)
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Journal Article
Structure-based design of novel nonpeptide inhibitors of the Src SH2 domain: Phosphotyrosine mimetics exploiting multifunctional group replacement chemistry
Sundaramoorthi, Raji, Kawahata, Noriyuki, Yang, Michael G., Shakespeare, William C., Metcalf III, Chester A., Wang, Yihan, Merry, Taylor, Eyermann, Charles J., Bohacek, Regine S., Narula, Surinder, Dalgarno, David C., Sawyer, Tomi K.
Published in Biopolymers (2003)
Published in Biopolymers (2003)
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FATTY ACID-BIFUNCTIONAL DEGRADER CONJUGATES AND THEIR METHODS OF USE
Fazal, Tanzina, Hollingworth, Gregory John, Palermo, Mark Gabriel, Metcalf, III, Chester A, Zoller, Thomas, Duvadie, Rohit Kumar, Lorber, Julien, Plummer, Scott Vaughan, Li, Jialiang, Sendzik, Martin, Broennimann, Valerie, Vulpetti, Anna, Adcock, Claire, Grotzfeld, Robert Martin, Gao, Jinhai, Michael, Walter, Zhao, Liang, Usera, Aimee Richardson, Cheng, Jiashun, Guo, Fengfeng, Hebach, Christina, Zecri, Frederic, Karpov, Alexei, Jones, Darryl Brynley, Roache, James Harold, Thomas, Ranny Mathew
Year of Publication 04.07.2024
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Year of Publication 04.07.2024
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FATTY ACID-BIFUNCTIONAL DEGRADER CONJUGATES AND THEIR METHODS OF USE
PLUMMER, Scott, Vaughan, SENDZIK, Martin, GROTZFELD, Robert, Martin, USERA, Aimee, Richardson, FAZAL, Tanzina, ADCOCK, Claire, METCALF III, Chester A, ZECRI, Frederic, ZOLLER, Thomas, THOMAS, Ranny, Mathew, GAO, Jinhai, MICHAEL, Walter, GUO, Fengfeng, DUVADIE, Rohit Kumar, KARPOV, Alexei, LORBER, Julien, ZHAO, Liang, HEBACH, Christina, PALERMO, Mark, Gabriel, JONES, Darryl, Brynley, LI, Jialiang, CHENG, Jiashun, VULPETTI, Anna, ROACHE, James, Harold, BROENNIMANN, Valerie, HOLLINGWORTH, Gregory John
Year of Publication 17.01.2024
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Year of Publication 17.01.2024
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SUBSTITUTED ACETYLENIC PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS KINASE INHIBITORS
Metcalf, III, Chester A, Qi, Jiwei, Thomas, R. Mathew, Dalgarno, David C, Romero, Jan Antoinette C, Zhu, Xiaotian, Sawyer, Tomi K, Zou, Dong, Huang, Wei-Sheng, Wang, Yihan, Shakespeare, William C, Sundaramoorthi, Rajeswari
Year of Publication 17.03.2022
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Year of Publication 17.03.2022
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INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL
LIU, Christopher, LI, Qingyi, JACKSON, Andrew, J, METCALF, Chester, A. III, CHENG, Lily, LIPPA, Blaise, S, WRONA, Iwona
Year of Publication 04.12.2019
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Year of Publication 04.12.2019
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FATTY ACID-BIFUNCTIONAL DEGRADER CONJUGATES AND THEIR METHODS OF USE
SENDZIK, Martin, FAZAL, Tanzina, THOMAS, Ranny, ADCOCK, Claire, PLUMMER, Scott, METCALF III, Chester A, ROACHE, James, ZECRI, Frederic, ZOLLER, Thomas, GROTZFELD, Robert, GAO, Jinhai, MICHAEL, Walter, GUO, Fengfeng, DUVADIE, Rohit Kumar, KARPOV, Alexei, LORBER, Julien, ZHAO, Liang, HEBACH, Christina, LI, Jialiang, CHENG, Jiashun, VULPETTI, Anna, BROENNIMANN, Valerie, USERA, Aimee, PALERMO, Mark, HOLLINGWORTH, Gregory John, JONES, Darryl
Year of Publication 15.09.2022
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Year of Publication 15.09.2022
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BICYCLIC HETEROARYL COMPOUNDS
DALGARNO, David C, HUANG, Wei-sheng, QI, Jiwei, WANG, Yihan, SAWYER, Tomi K, SUNDARAMOORTHI, Rajeswari, ROMERO, Jan Antoinette C, ZOU, Dong, THOMAS, Mathew R, ZHU, Xiaotian, SHAKESPEARE, William C, METCALF, Chester A, III
Year of Publication 09.12.2020
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Year of Publication 09.12.2020
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BICYCLIC HETEROARYL COMPOUNDS
DALGARNO, David C, HUANG, Wei-sheng, QI, Jiwei, WANG, Yihan, SAWYER, Tomi K, SUNDARAMOORTHI, Rajeswari, ROMERO, Jan Antoinette C, ZOU, Dong, THOMAS, Mathew R, ZHU, Xiaotian, SHAKESPEARE, William C, METCALF, Chester A, III
Year of Publication 12.08.2020
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Year of Publication 12.08.2020
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Bicyclic Heteroaryl Compounds
Metcalf, III, Chester A, Qi, Jiwei, Thomas, R. Mathew, Dalgarno, David C, Romero, Jan Antoinette C, Zhu, Xiaotian, Sawyer, Tomi K, Zou, Dong, Huang, Wei-Sheng, Wang, Yihan, Shakespeare, William C, Sundaramoorthi, Rajeswari
Year of Publication 23.07.2020
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Year of Publication 23.07.2020
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Bicyclic Heteroaryl Compounds
SHAKESPEARE, WILLIAM C, ZHU, XIAOTIAN, HUANG, WEI-SHENG, ROMERO, JAN ANTOINETTE C, DALGARNO, DAVID C, SUNDARAMOORTHI, RAJESWARI, SAWYER, TOMI K, QI, JIWEI, WANG, YIHAN, METCALF, CHESTER A III, THOMAS, MATHEW R, ZOU, DONG
Year of Publication 01.06.2020
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Year of Publication 01.06.2020
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Bicyclic Heteroaryl Compounds
Qi Jiwei, Zhu Xiaotian, Shakespeare William C, Sawyer Tomi K, Romero Jan Antoinette C, Metcalf Chester A III, Zou Dong, Huang Wei-sheng, Thomas Mathew R, Wang Yihan, Sundaramoorthi Rajeswari, Dalgarno David C
Year of Publication 30.04.2020
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Year of Publication 30.04.2020
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