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Published in Proceedings of the National Academy of Sciences - PNAS (26.02.2008)
Published in Proceedings of the National Academy of Sciences - PNAS (26.02.2008)
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Published in Proceedings of the National Academy of Sciences - PNAS (02.04.2013)
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Published in Proceedings of the National Academy of Sciences - PNAS (06.01.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (06.01.2009)
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A family of phosphodiesterase inhibitors discovered by cocrystallography and scaffold-based drug design
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Published in Nature biotechnology (01.02.2005)
Published in Nature biotechnology (01.02.2005)
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RAF inhibitors that evade paradoxical MAPK pathway activation
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Published in Nature (London) (22.10.2015)
Published in Nature (London) (22.10.2015)
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Improved Human Bioavailability of Vemurafenib, a Practically Insoluble Drug, Using an Amorphous Polymer-Stabilized Solid Dispersion Prepared by a Solvent-Controlled Coprecipitation Process
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Published in Journal of pharmaceutical sciences (01.03.2013)
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Characterizing and Overriding the Structural Mechanism of the Quizartinib-Resistant FLT3 "Gatekeeper" F691L Mutation with PLX3397
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Association of Combination of Conformation-Specific KIT Inhibitors With Clinical Benefit in Patients With Refractory Gastrointestinal Stromal Tumors: A Phase 1b/2a Nonrandomized Clinical Trial
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Structural Basis for the Activity of Drugs that Inhibit Phosphodiesterases
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Published in Structure (London) (01.12.2004)
Published in Structure (London) (01.12.2004)
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Published in Journal of the American Chemical Society (01.09.1993)
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Phosphodiesterase-4 as a potential drug target
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Published in Expert opinion on therapeutic targets (01.12.2005)
Published in Expert opinion on therapeutic targets (01.12.2005)
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