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A new family of H3 receptor antagonists based on the natural product Conessine

A new family of H3 receptor antagonists based on the natural product Conessine

by SANTORA, Vincent J, COVEL, Jonathan A, WEBB, Robert R, SAGE, Carleton, REN, Albert, PEREIRA, Guilherme, KNUDSEN, Jens, EDWARDS, Jeffrey E, SUAREZ, Marissa, FRAZER, John, THOMSEN, William, HAUSER, Erin, HAYASHI, Rena, WHELAN, Kevin, GROTTICK, Andrew J, HOFILENA, Brian J, IBARRA, Jason B, PULLEY, Michelle D, WEINHOUSE, Michael I, SENGUPTA, Dipanjan, DUFFIELD, Jonathan J, SEMPLE, Graeme
Published in Bioorganic & medicinal chemistry letters (15.02.2008)

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Journal Article

Identification of biaryl sulfone derivatives as antagonists of the histamine H3 receptor: Discovery of (R)-1-(2-(4′-(3-methoxypropylsulfonyl)biphenyl-4-yl)ethyl)-2-methylpyrrolidine (APD916)

Identification of biaryl sulfone derivatives as antagonists of the histamine H3 receptor: Discovery of (R)-1-(2-(4′-(3-methoxypropylsulfonyl)biphenyl-4-yl)ethyl)-2-methylpyrrolidine (APD916)

by Semple, Graeme, Santora, Vincent J., Smith, Jeffrey M., Covel, Jonathan A., Hayashi, Rena, Gallardo, Charlemagne, Ibarra, Jason B., Schultz, Jeffrey A., Park, Douglas M., Estrada, Scott A., Hofilena, Brian J., Smith, Brian M., Ren, Albert, Suarez, Marissa, Frazer, John, Edwards, Jeffrey E., Hart, Ryan, Hauser, Erin K., Lorea, Jodie, Grottick, Andrew J.
Published in Bioorganic & medicinal chemistry letters (01.01.2012)

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Journal Article

Design and Evaluation of Novel Biphenyl Sulfonamide Derivatives with Potent Histamine H(3) Receptor Inverse Agonist Activity

Design and Evaluation of Novel Biphenyl Sulfonamide Derivatives with Potent Histamine H(3) Receptor Inverse Agonist Activity

by Covel, Jonathan A., Santora, Vincent J., Smith, Jeffrey M., Hayashi, Rena, Gallardo, Charlemagne, Weinhouse, Michael I., Ibarra, Jason B., Schultz, Jeffrey A., Park, Douglas M., Estrada, Scott A., Hofilena, Brian J., Pulley, Michelle D., Smith, Brian M., Ren, Albert, Suarez, Marissa, Frazer, John, Edwards, Jeffrey, Hauser, Erin K., Lorca, Jodie, Semple, Graeme, Grottick, Andrew J.
Published in Journal of medicinal chemistry (24.09.2009)

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Journal Article

Design and Evaluation of Novel Biphenyl Sulfonamide Derivatives with Potent Histamine H3 Receptor Inverse Agonist Activity

Design and Evaluation of Novel Biphenyl Sulfonamide Derivatives with Potent Histamine H3 Receptor Inverse Agonist Activity

by Covel, Jonathan A., Santora, Vincent J., Smith, Jeffrey M., Hayashi, Rena, Gallardo, Charlemagne, Weinhouse, Michael I., Ibarra, Jason B., Schultz, Jeffrey A., Park, Douglas M., Estrada, Scott A., Hofilena, Brian J., Pulley, Michelle D., Smith, Brian M., Ren, Albert, Suarez, Marissa, Frazer, John, Edwards, Jeffrey, Hauser, Erin K., Lorea, Jodie, Semple, Graeme, Grottick, Andrew J.
Published in Journal of medicinal chemistry (24.09.2009)

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Journal Article

Novel H3 receptor antagonists with improved pharmacokinetic profiles

Novel H3 receptor antagonists with improved pharmacokinetic profiles

by SANTORA, Vincent J, COVEL, Jonathan A, EDWARDS, Jeffrey E, SUAREZ, Marissa, FRAZER, John, THOMSEN, William, HAUSER, Erin, LOREA, Jodie, GROTTICK, Andrew J, HAYASHI, Rena, HOFILENA, Brian J, IBARRA, Jason B, PULLEY, Michelle D, WEINHOUSE, Michael I, SEMPLE, Graeme, REN, Albert, PEREIRA, Guilherme
Published in Bioorganic & medicinal chemistry letters (15.07.2008)

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Journal Article

PYRAZOLYL SUBSTITUTED CARBONIC ACID DERIVATIVES AS MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

PYRAZOLYL SUBSTITUTED CARBONIC ACID DERIVATIVES AS MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

by ZOU NING, ULLMAN BRETT, SHIN, YOUNG JUN, TRAN THUY ANH, IBARRA JASON B, ZENG XI
Year of Publication 25.08.2011

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Patent

A new family of H 3 receptor antagonists based on the natural product Conessine

A new family of H 3 receptor antagonists based on the natural product Conessine

by Santora, Vincent J., Covel, Jonathan A., Hayashi, Rena, Hofilena, Brian J., Ibarra, Jason B., Pulley, Michelle D., Weinhouse, Michael I., Sengupta, Dipanjan, Duffield, Jonathan J., Semple, Graeme, Webb, Robert R., Sage, Carleton, Ren, Albert, Pereira, Guilherme, Knudsen, Jens, Edwards, Jeffrey E., Suarez, Marissa, Frazer, John, Thomsen, William, Hauser, Erin, Whelan, Kevin, Grottick, Andrew J.
Published in Bioorganic & medicinal chemistry letters (15.02.2008)

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Journal Article

Identification of biaryl sulfone derivatives as antagonists of the histamine H3 receptor: Discovery of (R)-1-2-(4'-(3-methoxypropylsulfonyl)biphenyl-4-yl)ethyl-2-methylpyrrolidine (APD916)

Identification of biaryl sulfone derivatives as antagonists of the histamine H3 receptor: Discovery of (R)-1-2-(4'-(3-methoxypropylsulfonyl)biphenyl-4-yl)ethyl-2-methylpyrrolidine (APD916)

by SEMPLE, Graeme, SANTORA, Vincent J, HOFILENA, Brian J, SMITH, Brian M, REN, Albert, SUAREZ, Marissa, FRAZER, John, EDWARDS, Jeffrey E, HART, Ryan, HAUSER, Erin K, LOREA, Jodie, GROTTICK, Andrew J, SMITH, Jeffrey M, COVEL, Jonathan A, HAYASHI, Rena, GALLARDO, Charlemagne, IBARRA, Jason B, SCHULTZ, Jeffrey A, PARK, Douglas M, ESTRADA, Scott A
Published in Bioorganic & medicinal chemistry letters (2012)

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Journal Article

Identification of biaryl sulfone derivatives as antagonists of the histamine H3 receptor: Discovery of (R)-1-(2-(4&; prime; -(3-methoxypropylsulfonyl)biphenyl-4-yl)e thyl)-2-methylpyrrolidine (APD916)

Identification of biaryl sulfone derivatives as antagonists of the histamine H3 receptor: Discovery of (R)-1-(2-(4&; prime; -(3-methoxypropylsulfonyl)biphenyl-4-yl)e thyl)-2-methylpyrrolidine (APD916)

by Semple, Graeme, Santora, Vincent J, Smith, Jeffrey M, Covel, Jonathan A, Hayashi, Rena, Gallardo, Charlemagne, Ibarra, Jason B, Schultz, Jeffrey A, Park, Douglas M, Estrada, Scott A, Hofilena, Brian J, Smith, Brian M, Ren, Albert, Suarez, Marissa, Frazer, John, Edwards, Jeffrey E, Hart, Ryan, Hauser, Erin K, Lorea, Jodie, Grottick, Andrew J
Published in Bioorganic & medicinal chemistry letters (01.01.2012)

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Journal Article

Design and Evaluation of Novel Biphenyl Sulfonamide Derivatives with Potent Histamine H 3 Receptor Inverse Agonist Activity

Design and Evaluation of Novel Biphenyl Sulfonamide Derivatives with Potent Histamine H 3 Receptor Inverse Agonist Activity

by Covel, Jonathan A., Santora, Vincent J., Smith, Jeffrey M., Hayashi, Rena, Gallardo, Charlemagne, Weinhouse, Michael I., Ibarra, Jason B., Schultz, Jeffrey A., Park, Douglas M., Estrada, Scott A., Hofilena, Brian J., Pulley, Michelle D., Smith, Brian M., Ren, Albert, Suarez, Marissa, Frazer, John, Edwards, Jeffrey, Hauser, Erin K., Lorea, Jodie, Semple, Graeme, Grottick, Andrew J.
Published in Journal of medicinal chemistry (24.09.2009)

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Journal Article

Novel H 3 receptor antagonists with improved pharmacokinetic profiles

Novel H 3 receptor antagonists with improved pharmacokinetic profiles

by Santora, Vincent J., Covel, Jonathan A., Hayashi, Rena, Hofilena, Brian J., Ibarra, Jason B., Pulley, Michelle D., Weinhouse, Michael I., Semple, Graeme, Ren, Albert, Pereira, Guilherme, Edwards, Jeffrey E., Suarez, Marissa, Frazer, John, Thomsen, William, Hauser, Erin, Lorea, Jodie, Grottick, Andrew J.
Published in Bioorganic & medicinal chemistry letters (15.07.2008)

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Journal Article

Novel H sub(3) receptor antagonists with improved pharmacokinetic profiles

Novel H sub(3) receptor antagonists with improved pharmacokinetic profiles

by Santora, Vincent J, Covel, Jonathan A, Hayashi, Rena, Hofilena, Brian J, Ibarra, Jason B, Pulley, Michelle D, Weinhouse, Michael I, Semple, Graeme, Ren, Albert, Pereira, Guilherme, Edwards, Jeffrey E, Suarez, Marissa, Frazer, John, Thomsen, William, Hauser, Erin, Lorea, Jodie, Grottick, Andrew J
Published in Bioorganic & medicinal chemistry (01.07.2008)

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Journal Article

A new family of H sub(3) receptor antagonists based on the natural product Conessine

A new family of H sub(3) receptor antagonists based on the natural product Conessine

by Santora, Vincent J, Covel, Jonathan A, Hayashi, Rena, Hofilena, Brian J, Ibarra, Jason B, Pulley, Michelle D, Weinhouse, Michael I, Sengupta, Dipanjan, Duffield, Jonathan J, Semple, Graeme, Webb, Robert R, Sage, Carleton, Ren, Albert, Pereira, Guilherme, Knudsen, Jens, Edwards, Jeffrey E, Suarez, Marissa, Frazer, John, Thomsen, William, Hauser, Erin, Whelan, Kevin, Grottick, Andrew J
Published in Bioorganic & medicinal chemistry (01.02.2008)

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Journal Article

Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto

Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto

by Zou, Ning, Shin, Young-Jun, Tran, Thuy-Anh, Ibarra, Jason B, Zeng, Xi, Ullman, Brett
Year of Publication 24.08.2021

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Patent

PYRAZOLYL SUBSTITUTED CARBONIC ACID DERIVATIVES AS MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

PYRAZOLYL SUBSTITUTED CARBONIC ACID DERIVATIVES AS MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

by ULLMAN, Brett, TRAN, Thuy-Anh, IBARRA, Jason B, SHIN, Young-Jun, ZENG, Xi, ZOU, Ning
Year of Publication 14.04.2021

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Patent

PYRAZOLYL SUBSTITUTED CARBONIC ACID DERIVATIVES AS MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

PYRAZOLYL SUBSTITUTED CARBONIC ACID DERIVATIVES AS MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

by ULLMAN, Brett, TRAN, Thuy-Anh, IBARRA, Jason B, SHIN, Young-Jun, ZENG, Xi, ZOU, Ning
Year of Publication 17.12.2020

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Patent

Substituted pyridazines and 1,2,4-triazines as prostacyclin receptor modulators

Substituted pyridazines and 1,2,4-triazines as prostacyclin receptor modulators

by Zou, Ning, Tran, Thuy-Anh, Ibarra, Jason B, Ullman, Brett, Hayashi, Rena
Year of Publication 06.10.2020

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Patent

Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto

Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto

by Zou, Ning, Shin, Young-Jun, Tran, Thuy-Anh, Ibarra, Jason B, Zeng, Xi, Ullman, Brett
Year of Publication 23.06.2020

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Patent

PYRAZOLYL SUBSTITUTED CARBONIC ACID DERIVATIVES AS MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

PYRAZOLYL SUBSTITUTED CARBONIC ACID DERIVATIVES AS MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

by Zou, Ning, Shin, Young-Jun, Tran, Thuy-Anh, Ibarra, Jason B, Zeng, Xi, Ullman, Brett
Year of Publication 05.09.2019

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Patent

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

by Zou, Ning, Tran, Thuy-Anh, Ibarra, Jason B, Ullman, Brett, Hayashi, Rena
Year of Publication 15.08.2019

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Patent

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