Novel p-Arylthio Cinnamides as Antagonists of Leukocyte Function-Associated Antigen-1/Intracellular Adhesion Molecule-1 Interaction. 2. Mechanism of Inhibition and Structure-Based Improvement of Pharmaceutical Properties
Liu, Gang, Huth, Jeffrey R, Olejniczak, Edward T, Mendoza, Renaldo, DeVries, Peter, Leitza, Sandra, Reilly, Edward B, Okasinski, Gregory F, Fesik, Stephen W, von Geldern, Thomas W
Published in Journal of medicinal chemistry (12.04.2001)
Published in Journal of medicinal chemistry (12.04.2001)
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Intracellular folding pathway of human chorionic gonadotropin beta subunit
HUTH, J. R, MOUNTJOY, K, PERINI, F, RUDDON, R. W
Published in The Journal of biological chemistry (05.05.1992)
Published in The Journal of biological chemistry (05.05.1992)
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Disulfide bond mutations affect the folding of the human chorionic gonadotropin-beta subunit in transfected Chinese hamster ovary cells
BEDOWS, E, HUTH, J. R, SUGANUMA, N, BARTELS, C. F, BOIME, I, RUDDON, R. W
Published in The Journal of biological chemistry (05.06.1993)
Published in The Journal of biological chemistry (05.06.1993)
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Domain-dependent protein folding is indicated by the intracellular kinetics of disulfide bond formation of human chorionic gonadotropin beta subunit
Huth, J.R., Mountjoy, K, Perini, F, Bedows, E, Ruddon, R.W.
Published in The Journal of biological chemistry (25.10.1992)
Published in The Journal of biological chemistry (25.10.1992)
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Design of an expression system for detecting folded protein domains and mapping macromolecular interactions by NMR
Huth, Jeffrey R., Bewley, Carole A., Clore, G. Marius, Gronenborn, Angela M., Jackson, Belinda M., Hinnebusch, Alan G.
Published in Protein science (01.11.1997)
Published in Protein science (01.11.1997)
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Discovery of Novel p-Arylthio Cinnamides as Antagonists of Leukocyte Function-Associated Antigen-1/Intercellular Adhesion Molecule-1 Interaction. 4. Structure−Activity Relationship of Substituents on the Benzene Ring of the Cinnamide
Winn, Martin, Reilly, Edward B, Liu, Gang, Huth, Jeffrey R, Jae, Hwan-Soo, Freeman, Jennifer, Pei, Zhonghua, Xin, Zhili, Lynch, John, Kester, Jeff, von Geldern, Thomas W, Leitza, Sandra, DeVries, Peter, Dickinson, Robert, Mussatto, Donna, Okasinski, Gregory F
Published in Journal of medicinal chemistry (06.12.2001)
Published in Journal of medicinal chemistry (06.12.2001)
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Discovery of Potent Antagonists of Leukocyte Function-Associated Antigen-1/Intercellular Adhesion Molecule-1 Interaction. 3. Amide (C-Ring) Structure−Activity Relationship and Improvement of Overall Properties of Arylthio Cinnamides
Pei, Zhonghua, Xin, Zhili, Liu, Gang, Li, Yihong, Reilly, Edward B, Lubbers, Nathan L, Huth, Jeffery R, Link, James T, von Geldern, Thomas W, Cox, Bryan F, Leitza, Sandra, Gao, Yi, Marsh, Kennan C, DeVries, Peter, Okasinski, Greg F
Published in Journal of medicinal chemistry (30.08.2001)
Published in Journal of medicinal chemistry (30.08.2001)
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Protein folding and assembly in vitro parallel intracellular folding and assembly. Catalysis of folding and assembly of the human chorionic gonadotropin alpha beta dimer by protein disulfide isomerase
Huth, J R, Perini, F, Lockridge, O, Bedows, E, Ruddon, R W
Published in The Journal of biological chemistry (05.08.1993)
Published in The Journal of biological chemistry (05.08.1993)
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Druggability Indices for Protein Targets Derived from NMR-Based Screening Data
Hajduk, Philip J, Huth, Jeffrey R, Fesik, Stephen W
Published in Journal of medicinal chemistry (07.04.2005)
Published in Journal of medicinal chemistry (07.04.2005)
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The Wing of the Enhancer-Binding Domain of Mu Phage Transposase is Flexible and is Essential for Efficient Transposition
Clubb, Robert T., Mizuuchi, Michiyo, Huth, Jeffrey R., Omichinski, James G., Savilahti, Harri, Mizuuchi, Kiyoshi, Clore, G. Marius, Gronenborn, Angela M.
Published in Proceedings of the National Academy of Sciences - PNAS (06.02.1996)
Published in Proceedings of the National Academy of Sciences - PNAS (06.02.1996)
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